CY1117706T1 - Παραγωγα οξαζολινης και ισοξαζολινης ως ρυθμιστες crac - Google Patents

Παραγωγα οξαζολινης και ισοξαζολινης ως ρυθμιστες crac

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Publication number
CY1117706T1
CY1117706T1 CY20161100600T CY161100600T CY1117706T1 CY 1117706 T1 CY1117706 T1 CY 1117706T1 CY 20161100600 T CY20161100600 T CY 20161100600T CY 161100600 T CY161100600 T CY 161100600T CY 1117706 T1 CY1117706 T1 CY 1117706T1
Authority
CY
Cyprus
Prior art keywords
crac
isaxazoline
oxazoline
producers
regulators
Prior art date
Application number
CY20161100600T
Other languages
English (en)
Inventor
Nageswara Rao Irlapati
Gokul Keruji Deshmukh
Vijay Pandurang Karche
Santosh Madhukar Jachak
Neelima Sinha
Venkata P Palle
Rajender Kumar Kamboj
Original Assignee
Lupin Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lupin Limited filed Critical Lupin Limited
Publication of CY1117706T1 publication Critical patent/CY1117706T1/el

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
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  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Η παρούσα εφεύρεση αφορά σε ενώσεις του Τύπου (I), μαζί με μεθόδους για παρασκευή αυτών, που είναι χρήσιμες για θεραπεία, πρόληψη ή/και χειρισμό των ασθενειών, διαταραχών, συνδρόμων ή καταστάσεων που σχετίζονται με την ρύθμιση του CRAC. Η εφεύρεση περαιτέρω αφορά σε μεθόδους θεραπείας, πρόληψης, χειρισμού ή/και ελάττωσης των ασθενειών, διαταραχών, συνδρόμων ή καταστάσεων που σχετίζονται με την ρύθμιση CRAC του Τύπου (I).
CY20161100600T 2010-10-30 2016-06-30 Παραγωγα οξαζολινης και ισοξαζολινης ως ρυθμιστες crac CY1117706T1 (el)

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