CY1114975T1 - Σκευασμα εμφυτευματος παλιπεριδονης - Google Patents

Σκευασμα εμφυτευματος παλιπεριδονης

Info

Publication number
CY1114975T1
CY1114975T1 CY20141100156T CY141100156T CY1114975T1 CY 1114975 T1 CY1114975 T1 CY 1114975T1 CY 20141100156 T CY20141100156 T CY 20141100156T CY 141100156 T CY141100156 T CY 141100156T CY 1114975 T1 CY1114975 T1 CY 1114975T1
Authority
CY
Cyprus
Prior art keywords
composition
weeks
polyperidonic
infection preparation
rmakokinitika
Prior art date
Application number
CY20141100156T
Other languages
Greek (el)
English (en)
Inventor
Aduriz Ibon Gutierro
Rodriguez Guillermo Franco
Original Assignee
Laboratorios Farmaceuticos Rovi, S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47074463&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1114975(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Laboratorios Farmaceuticos Rovi, S.A. filed Critical Laboratorios Farmaceuticos Rovi, S.A.
Publication of CY1114975T1 publication Critical patent/CY1114975T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A61K9/0024Solid, semi-solid or solidifying implants, which are implanted or injected in body tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Inorganic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Materials For Medical Uses (AREA)
CY20141100156T 2012-05-31 2014-02-26 Σκευασμα εμφυτευματος παλιπεριδονης CY1114975T1 (el)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP12170366.4A EP2529757B1 (en) 2011-05-31 2012-05-31 Paliperidone implant formulation

Publications (1)

Publication Number Publication Date
CY1114975T1 true CY1114975T1 (el) 2016-12-14

Family

ID=47074463

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20141100156T CY1114975T1 (el) 2012-05-31 2014-02-26 Σκευασμα εμφυτευματος παλιπεριδονης

Country Status (29)

Country Link
EP (1) EP2529757B1 (enExample)
JP (1) JP6430933B2 (enExample)
KR (1) KR101892496B1 (enExample)
CN (2) CN109966239A (enExample)
AU (1) AU2013269546B2 (enExample)
BR (1) BR112014029208B1 (enExample)
CA (1) CA2874702C (enExample)
CL (1) CL2014003215A1 (enExample)
CO (1) CO7160109A2 (enExample)
CY (1) CY1114975T1 (enExample)
DK (1) DK2529757T3 (enExample)
EA (1) EA029921B1 (enExample)
ES (1) ES2456917T3 (enExample)
HR (1) HRP20140158T1 (enExample)
IL (1) IL235850A0 (enExample)
IN (1) IN2014DN10673A (enExample)
MA (1) MA37661B1 (enExample)
MX (1) MX365097B (enExample)
MY (1) MY181549A (enExample)
NZ (1) NZ703319A (enExample)
PH (1) PH12014502668A1 (enExample)
PL (1) PL2529757T3 (enExample)
PT (1) PT2529757E (enExample)
SG (1) SG11201407971QA (enExample)
SI (1) SI2529757T1 (enExample)
SM (1) SMT201400044B (enExample)
UA (1) UA115987C2 (enExample)
WO (1) WO2013178811A1 (enExample)
ZA (1) ZA201409297B (enExample)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2529757B1 (en) * 2011-05-31 2014-01-08 Laboratorios Farmaceuticos Rovi, S.A. Paliperidone implant formulation
US10285936B2 (en) 2010-05-31 2019-05-14 Laboratorios Farmacéuticos Rovi, S.A. Injectable composition with aromatase inhibitor
US10350159B2 (en) 2010-05-31 2019-07-16 Laboratories Farmacéuticos Rovi, S.A. Paliperidone implant formulation
US10335366B2 (en) 2010-05-31 2019-07-02 Laboratorios Farmacéuticos Rovi, S.A. Risperidone or paliperidone implant formulation
US10463607B2 (en) 2010-05-31 2019-11-05 Laboratorios Farmaceutics Rofi S.A. Antipsychotic Injectable Depot Composition
SMT202100679T1 (it) 2010-05-31 2022-01-10 Laboratorios Farmaceuticos Rovi S A Composizioni per impianti biodegradabili in-situ iniettabili
US10881605B2 (en) 2010-05-31 2021-01-05 Laboratorios Farmaceuticos Rovi, S.A. Methods for the preparation of injectable depot compositions
PT2394664T (pt) 2010-05-31 2016-09-06 Farm Rovi Lab Sa Composição depot para injetável antipsicótico
RS62059B1 (sr) * 2011-05-31 2021-07-30 Laboratorios Farmaceuticos Rovi S A Kompozicija implanta risperidona i/ili paliperidona
KR102755145B1 (ko) 2015-04-07 2025-01-14 잔센파마슈티카엔.브이. 장기간 작용형 주사용 팔리페리돈 에스테르에 대한 누락된 용량에 대한 투여 계획
CN106038569A (zh) * 2016-05-26 2016-10-26 湖南赛沃药业有限公司 一种帕利哌酮植入剂及其制备方法
US12097292B2 (en) 2016-08-28 2024-09-24 Mapi Pharma Ltd. Process for preparing microparticles containing glatiramer acetate
SMT202500136T1 (it) * 2016-08-31 2025-05-12 Mapi Pharma Ltd Sistemi a deposito comprendenti glatiramer acetato
US11167003B2 (en) 2017-03-26 2021-11-09 Mapi Pharma Ltd. Methods for suppressing or alleviating primary or secondary progressive multiple sclerosis (PPMS or SPMS) using sustained release glatiramer depot systems
EP3700531B1 (en) * 2017-10-27 2025-06-25 Geneora Pharma (Shijiazhuang) Co., Ltd. Dosage regimen of paliperidone palmitate extended-release injectable suspension
EP3803866A4 (en) 2018-05-24 2022-03-16 Nureva Inc. METHOD, APPARATUS, AND COMPUTER READABLE MATERIALS FOR MANAGING SEMI-CONSTANT (PERSISTENT) SOUND SOURCES IN MICROPHONE CATCH/HOME AREAS
CN111971026A (zh) 2018-05-24 2020-11-20 塞拉尼斯伊娃高性能聚合物公司 用于持续释放大分子药物化合物的可植入器件
BR112020023982A2 (pt) 2018-05-24 2021-02-23 Celanese Eva Performance Polymers Llc dispositivo implantável para liberação prolongada de um composto de fármaco macromolecular
PE20210047A1 (es) 2018-06-12 2021-01-08 Farm Rovi Lab Sa Composicion inyectable
EP4356966A3 (en) 2020-11-30 2024-07-17 JANSSEN Pharmaceutica NV Dosing regimens associated with extended release paliperidone injectable formulations
US11324751B1 (en) 2020-11-30 2022-05-10 Janssen Pharmaceutica Nv Dosing regimens associated with extended release paliperidone injectable formulations
FI4025189T3 (fi) 2020-11-30 2024-07-02 Janssen Pharmaceutica Nv Viivästetysti vapauttavaan injektoitavaan paliperidoniin liittyviä annostusohjelmia
BR112023022439A2 (pt) 2021-04-26 2023-12-26 Celanese Eva Performance Polymers Llc Dispositivo implantável para liberação sustentada de um composto de fármaco macromolecular
US12318387B2 (en) 2021-07-16 2025-06-03 Laboratorios Farmaceuticos Rovi, S.A. Method of treating acute exacerbation of schizophrenia with long-acting injectable depot composition
CN118119394A (zh) 2021-08-20 2024-05-31 詹森药业有限公司 与延长释放帕潘立酮可注射制剂相关的给药方案
TW202313047A (zh) 2021-09-21 2023-04-01 西班牙商禾霏藥品實驗室有限公司 抗精神病可注射儲積型組合物
EP4527389A1 (en) 2022-05-18 2025-03-26 Laboratorios Farmacéuticos Rovi S.A. Prolonged-release injectable compositions for use in treatment with risperidone together with cyp2d6 enzyme inhibitors

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1660039B1 (en) * 2003-07-18 2016-09-28 Oakwood Laboratories L.L.C. Prevention of molecular weight reduction of the polymer, impurity formation and gelling in polymer compositions
AU2005271522B2 (en) 2004-08-04 2011-02-10 Alza Corporation Sustained drug release composition demonstrating an ascending zero order release pattern, methods of manufacturing such a composition
US8852638B2 (en) * 2005-09-30 2014-10-07 Durect Corporation Sustained release small molecule drug formulation
BRPI0809837A2 (pt) 2007-04-19 2014-11-11 Youxin Li "composto para tratamento de distúrbios mentais, saldo do composto para tratamento de distúrbios mentais, composição farmacéutica e uso do composto para tratamento de distúrbios mentais"
MX354603B (es) * 2007-05-25 2018-03-13 Indivior Uk Ltd Formulaciones de transferencia sostenida de compuestos de risperidona.
EP2178872A1 (en) 2007-07-27 2010-04-28 Synthon B.V. Paliperidone derivatives
KR102163196B1 (ko) 2007-12-19 2020-10-12 얀센 파마슈티카 엔.브이. 장기 작용성 주사가능 팔리페리돈 에스테르와 관련된 투여 요법
EP2485712A1 (en) 2009-10-06 2012-08-15 Ascendis Pharma A/S Subcutaneous paliperidone composition
EP2529757B1 (en) * 2011-05-31 2014-01-08 Laboratorios Farmaceuticos Rovi, S.A. Paliperidone implant formulation
PT2394664T (pt) * 2010-05-31 2016-09-06 Farm Rovi Lab Sa Composição depot para injetável antipsicótico
SMT202100679T1 (it) * 2010-05-31 2022-01-10 Laboratorios Farmaceuticos Rovi S A Composizioni per impianti biodegradabili in-situ iniettabili
RS62059B1 (sr) * 2011-05-31 2021-07-30 Laboratorios Farmaceuticos Rovi S A Kompozicija implanta risperidona i/ili paliperidona

Also Published As

Publication number Publication date
PL2529757T3 (pl) 2014-04-30
SMT201400044B (it) 2014-05-07
EP2529757A1 (en) 2012-12-05
MY181549A (en) 2020-12-28
ZA201409297B (en) 2015-12-23
JP6430933B2 (ja) 2018-11-28
PT2529757E (pt) 2014-02-27
CN109966239A (zh) 2019-07-05
EA201401348A1 (ru) 2015-04-30
IN2014DN10673A (enExample) 2015-08-28
ES2456917T3 (es) 2014-04-24
SG11201407971QA (en) 2014-12-30
HRP20140158T1 (hr) 2014-04-25
JP2015518035A (ja) 2015-06-25
AU2013269546B2 (en) 2017-12-14
CO7160109A2 (es) 2015-01-15
SI2529757T1 (sl) 2014-05-30
CN104349792A (zh) 2015-02-11
CA2874702C (en) 2021-05-11
KR20150015020A (ko) 2015-02-09
BR112014029208B1 (pt) 2020-04-07
AU2013269546A1 (en) 2015-01-22
WO2013178811A1 (en) 2013-12-05
KR101892496B1 (ko) 2018-10-04
DK2529757T3 (en) 2014-02-24
EA029921B1 (ru) 2018-05-31
PH12014502668B1 (en) 2015-02-02
BR112014029208A2 (pt) 2017-06-27
MX2014014484A (es) 2015-02-24
MA37661B1 (fr) 2016-12-30
NZ703319A (en) 2016-12-23
MX365097B (es) 2019-05-22
IL235850A0 (en) 2015-01-29
MA37661A1 (fr) 2016-03-31
PH12014502668A1 (en) 2015-02-02
CA2874702A1 (en) 2013-12-05
UA115987C2 (uk) 2018-01-25
CL2014003215A1 (es) 2015-07-10
EP2529757B1 (en) 2014-01-08

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