CY1112815T1 - Ανταγωνιστες υποδοχεα ορμονης απελευθερωσης γοναδοτροπινης και μεθοδοι που σχετιζονται με αυτους - Google Patents

Ανταγωνιστες υποδοχεα ορμονης απελευθερωσης γοναδοτροπινης και μεθοδοι που σχετιζονται με αυτους

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Publication number
CY1112815T1
CY1112815T1 CY20121100499T CY121100499T CY1112815T1 CY 1112815 T1 CY1112815 T1 CY 1112815T1 CY 20121100499 T CY20121100499 T CY 20121100499T CY 121100499 T CY121100499 T CY 121100499T CY 1112815 T1 CY1112815 T1 CY 1112815T1
Authority
CY
Cyprus
Prior art keywords
methods
competitives
gonadotropine
hormones
pharmaceutically acceptable
Prior art date
Application number
CY20121100499T
Other languages
Greek (el)
English (en)
Inventor
Yun-Fei Zhu
Chen Chen
Fabio C Tucci
Zhiqiang Guo
Timothy D Gross
Martin Rowbottom
R Scott Struthers
Original Assignee
Neurocrine Biosciences, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurocrine Biosciences, Inc. filed Critical Neurocrine Biosciences, Inc.
Publication of CY1112815T1 publication Critical patent/CY1112815T1/el

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
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    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/60—Three or more oxygen or sulfur atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
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CY20121100499T 2000-01-25 2012-06-01 Ανταγωνιστες υποδοχεα ορμονης απελευθερωσης γοναδοτροπινης και μεθοδοι που σχετιζονται με αυτους CY1112815T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17793300P 2000-01-25 2000-01-25
US23968300P 2000-10-11 2000-10-11
EP01910362A EP1255738B1 (en) 2000-01-25 2001-01-25 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto

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CY1112815T1 true CY1112815T1 (el) 2016-02-10

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CA2398018A1 (en) 2001-08-02
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AU767585B2 (en) 2003-11-20
US20070208049A1 (en) 2007-09-06
WO2001055119A2 (en) 2001-08-02
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US6608197B2 (en) 2003-08-19
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US7462625B2 (en) 2008-12-09
US20040048884A1 (en) 2004-03-11
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