CY1106973T1 - Παραγωγα θειαζολινης ως εκλεκτικοι διαμορφωται υποδοχεως ανδρογονου (sarms) - Google Patents
Παραγωγα θειαζολινης ως εκλεκτικοι διαμορφωται υποδοχεως ανδρογονου (sarms)Info
- Publication number
- CY1106973T1 CY1106973T1 CY20071101413T CY071101413T CY1106973T1 CY 1106973 T1 CY1106973 T1 CY 1106973T1 CY 20071101413 T CY20071101413 T CY 20071101413T CY 071101413 T CY071101413 T CY 071101413T CY 1106973 T1 CY1106973 T1 CY 1106973T1
- Authority
- CY
- Cyprus
- Prior art keywords
- androgen
- thaizolin
- sarms
- conductors
- products
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/26—Androgens
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Dermatology (AREA)
- Virology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Oncology (AREA)
- Diabetes (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- AIDS & HIV (AREA)
- Urology & Nephrology (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
Η παρούσα εφεύρεσις αναφέρεται εις νέα παράγωγα θειαζολίνης του γενικού τύπου (Ι)˙ εις τον οποίον όλες οι μεταβλητές είναι ως καθορίζονται ενταύθα, φαρμακευτικαί συνθέσεις περιέχουσαι αυτά και χρήσις των εις την θεραπείαν διαταραχών και καταστάσεων διαμορφωμένων υπό του υποδοχέως ανδρογόνου.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US47871203P | 2003-06-13 | 2003-06-13 | |
EP04755044A EP1656360B1 (en) | 2003-06-13 | 2004-06-12 | Thiazoline derivatives as selective androgen receptor modulators (sarms) |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1106973T1 true CY1106973T1 (el) | 2012-09-26 |
Family
ID=33539114
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20071101413T CY1106973T1 (el) | 2003-06-13 | 2007-11-05 | Παραγωγα θειαζολινης ως εκλεκτικοι διαμορφωται υποδοχεως ανδρογονου (sarms) |
Country Status (14)
Country | Link |
---|---|
US (1) | US20050014952A1 (el) |
EP (1) | EP1656360B1 (el) |
JP (1) | JP4898446B2 (el) |
CN (1) | CN1835937B (el) |
AT (1) | ATE370133T1 (el) |
AU (1) | AU2004249697B2 (el) |
CA (1) | CA2528764A1 (el) |
CY (1) | CY1106973T1 (el) |
DE (1) | DE602004008300T2 (el) |
DK (1) | DK1656360T3 (el) |
ES (1) | ES2291906T3 (el) |
PL (1) | PL1656360T3 (el) |
PT (1) | PT1656360E (el) |
WO (1) | WO2004113309A1 (el) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN104803916B (zh) | 2004-11-16 | 2017-08-11 | 詹森药业有限公司 | 用作选择性雄激素受体调节剂(sarms)的杂环衍生物 |
US7709516B2 (en) | 2005-06-17 | 2010-05-04 | Endorecherche, Inc. | Helix 12 directed non-steroidal antiandrogens |
US9284345B2 (en) | 2007-04-12 | 2016-03-15 | Endorecherche, Inc. | 17alpha-substituted steroids as systemic antiandrogens and selective androgen receptor modulators |
EP2802608A4 (en) * | 2012-01-12 | 2015-08-05 | Univ Yale | COMPOUNDS AND METHODS FOR ENHANCED DEGRADATION OF TARGET PROTEINS AND OTHER POLYPEPTIDES BY E3 UBIQUITIN LIGASE |
CN103450112B (zh) * | 2013-08-07 | 2019-09-13 | 华东理工大学 | 一种n-桥连接的含氮五元杂环化合物及其制备与用途 |
US9682960B2 (en) | 2013-12-19 | 2017-06-20 | Endorecherche, Inc. | Non-steroidal antiandrogens and selective androgen receptor modulators with a pyridyl moiety |
CN113811333B (zh) | 2019-05-14 | 2024-03-12 | 诺维逊生物股份有限公司 | 靶向抗癌核激素受体的化合物 |
US11952349B2 (en) | 2019-11-13 | 2024-04-09 | Nuvation Bio Inc. | Anti-cancer nuclear hormone receptor-targeting compounds |
IL306010A (en) | 2021-03-23 | 2023-11-01 | Nuvation Bio Inc | Anticancer compounds against the nuclear hormone receptor |
US12006314B2 (en) | 2021-05-03 | 2024-06-11 | Nuvation Bio Inc. | Anti-cancer nuclear hormone receptor-targeting compounds |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR9506625A (pt) * | 1994-01-24 | 1997-09-30 | Du Pont | Composto composição artropodicida e método para controle de artrópodos |
US6403623B1 (en) * | 1999-05-27 | 2002-06-11 | Unuversity Of Notre Dame Du Lac | Heterocyclic antituberculosis agents |
EA014224B1 (ru) * | 2000-08-24 | 2010-10-29 | Юниверсити Оф Теннесси Рисерч Фаундейшн | Селективные модуляторы андрогенового рецептора и способы их применения |
-
2004
- 2004-06-12 CA CA002528764A patent/CA2528764A1/en not_active Abandoned
- 2004-06-12 US US10/866,591 patent/US20050014952A1/en not_active Abandoned
- 2004-06-12 AT AT04755044T patent/ATE370133T1/de active
- 2004-06-12 AU AU2004249697A patent/AU2004249697B2/en not_active Ceased
- 2004-06-12 JP JP2006533745A patent/JP4898446B2/ja not_active Expired - Fee Related
- 2004-06-12 ES ES04755044T patent/ES2291906T3/es not_active Expired - Lifetime
- 2004-06-12 DE DE602004008300T patent/DE602004008300T2/de not_active Expired - Lifetime
- 2004-06-12 EP EP04755044A patent/EP1656360B1/en not_active Expired - Lifetime
- 2004-06-12 WO PCT/US2004/018665 patent/WO2004113309A1/en active IP Right Grant
- 2004-06-12 PT PT04755044T patent/PT1656360E/pt unknown
- 2004-06-12 CN CN2004800230915A patent/CN1835937B/zh not_active Expired - Fee Related
- 2004-06-12 PL PL04755044T patent/PL1656360T3/pl unknown
- 2004-06-12 DK DK04755044T patent/DK1656360T3/da active
-
2007
- 2007-11-05 CY CY20071101413T patent/CY1106973T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
JP4898446B2 (ja) | 2012-03-14 |
EP1656360B1 (en) | 2007-08-15 |
JP2007501287A (ja) | 2007-01-25 |
CN1835937B (zh) | 2012-07-18 |
AU2004249697B2 (en) | 2010-04-22 |
CN1835937A (zh) | 2006-09-20 |
ES2291906T3 (es) | 2008-03-01 |
DE602004008300T2 (de) | 2008-05-08 |
CA2528764A1 (en) | 2004-12-29 |
DK1656360T3 (da) | 2007-12-27 |
US20050014952A1 (en) | 2005-01-20 |
AU2004249697A1 (en) | 2004-12-29 |
PL1656360T3 (pl) | 2008-01-31 |
DE602004008300D1 (de) | 2007-09-27 |
EP1656360A1 (en) | 2006-05-17 |
ATE370133T1 (de) | 2007-09-15 |
WO2004113309A1 (en) | 2004-12-29 |
PT1656360E (pt) | 2007-10-22 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CY1106973T1 (el) | Παραγωγα θειαζολινης ως εκλεκτικοι διαμορφωται υποδοχεως ανδρογονου (sarms) | |
MY142048A (en) | Novel heterocycle derivatives useful as selective androgen receptor modulators (sarms) | |
TW200621725A (en) | Novel benzimidazole derivatives useful as selective androgen receptor modulators (sarms) | |
SG10201809390QA (en) | Modulators of indoleamine 2,3-dioxygenase and methods of using the same | |
TW200624424A (en) | Novel benzimidazole derivatives useful as selective androgen receptor modulators (sarms) | |
DE60224928D1 (de) | Dermatologische und kosmetische zusammensetzungen enthaltend ein furfurylderivat | |
DE60003863D1 (de) | Dioxocyclopentylhydroxamsäure | |
BR0315547A (pt) | Derivados de quinolina como antagonistas de crth2 | |
MX2007011695A (es) | Derivados de oxindol sustituido, medicamentos que contienen dichos derivados y uso de los mismos. | |
TW200606146A (en) | Novel indole derivatives as selective androgen receptor modulators (SARMS) | |
NO20063821L (no) | Kinolinderivater for anvendelse som mykobakterielle inhibitorer | |
AU2003276028A1 (en) | Pyridine derivatives as cb2 receptor modulators | |
EA201001682A1 (ru) | Производные фенил- и бензодиоксинилзамещенных индазолов | |
MXPA06000921A (es) | Derivados de benzamidazoles como inhibidores de mek. | |
MA32544B1 (fr) | Derives de pyridino-pyridinones, leur preparation et leur application en therapeutique | |
DE602005010401D1 (de) | Imidazolinderivate mit cb1-antagonistischer wirkung | |
NO20082096L (no) | Azaindol-2-karboksamidderivativer | |
MX2007011698A (es) | Derivados de oxindol sustituido, medicamentos que contienen dichos derivados y uso de los mismos. | |
TW200604171A (en) | Novel indole derivatives as selective androgen receptor modulators (SARMs) | |
TW200604170A (en) | Novel indole derivatives as selective androgen receptor modulators (SARMs) | |
ES2335410T8 (es) | Derivados de aminopropanol. | |
MXPA06003363A (es) | Derivados de fenil-piperazina como moduladores de receptores muscarinicos. | |
SE0300456D0 (sv) | Novel compounds | |
CY1109371T1 (el) | Παραγωγα σουλφαμικου βενζοθειοφαινιου ως αναστολεις σουλφατασης στεροειδους | |
ES2345882T3 (es) | Nuevos compuestos y su uso como moduladores de ppar. |