CU20190079A7 - Compuestos derivados de 3-([2-fenoxi]fenoxi)-2-hidroxi-n-bencyl-ciclohexilamina substituidos como inhibidores de la función mitocondrial y composiciones farmacéuticas que los contienen - Google Patents

Compuestos derivados de 3-([2-fenoxi]fenoxi)-2-hidroxi-n-bencyl-ciclohexilamina substituidos como inhibidores de la función mitocondrial y composiciones farmacéuticas que los contienen

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Publication number
CU20190079A7
CU20190079A7 CU2019000079A CU20190079A CU20190079A7 CU 20190079 A7 CU20190079 A7 CU 20190079A7 CU 2019000079 A CU2019000079 A CU 2019000079A CU 20190079 A CU20190079 A CU 20190079A CU 20190079 A7 CU20190079 A7 CU 20190079A7
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Cuba
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phenoxy
inhibitors
pharmaceutical compositions
compositions containing
mitochondrial function
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CU2019000079A
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English (en)
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Michael P Lisanti
Federica Sotgia
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Lunella Biotech Inc
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Publication of CU20190079A7 publication Critical patent/CU20190079A7/es

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    • C07C217/64—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups bound to carbon atoms of at least one six-membered aromatic ring and amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups linked to the six-membered aromatic ring, or to the condensed ring system containing that ring, by carbon chains further substituted by singly-bound oxygen atoms
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Abstract

<p>La presente descripción se refiere a compuestos de mitoribociclina de fórmula</p> <p>ESPACIO PARA LA FÓRMULA</p> <p>composiciones farmacéuticas que los contienen como inhibidores de la función mitocondrial. Tales compuestos tienen propiedades anti-cáncer y antibióticas, para proporcionar beneficios anti-edad, así como anticonceptivo masculino, agente espermistático, y agente inmovilizador del esperma.</p>
CU2019000079A 2017-03-15 2018-03-14 Compuestos derivados de 3-([2-fenoxi]fenoxi)-2-hidroxi-n-bencyl-ciclohexilamina substituidos como inhibidores de la función mitocondrial y composiciones farmacéuticas que los contienen CU20190079A7 (es)

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US201762471688P 2017-03-15 2017-03-15
PCT/US2018/022403 WO2018170109A1 (en) 2017-03-15 2018-03-14 Mitoriboscins: mitochondrial-based therapeutics targeting cancer cells, bacteria, and pathogenic yeast

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CU2019000096A CU20190096A7 (es) 2017-03-15 2018-03-14 Compuestos derivados de 3-metil-3-hidroxi-4-[(n,n-dimetil)amino]-9-[2-(benciloxi)bencil]-1-oxa-9-azaspiro[5,5]undecano substituidos como inhibidores de la función mitocondrial y composiciones farmacéuticas que los contienen
CU2019000079A CU20190079A7 (es) 2017-03-15 2018-03-14 Compuestos derivados de 3-([2-fenoxi]fenoxi)-2-hidroxi-n-bencyl-ciclohexilamina substituidos como inhibidores de la función mitocondrial y composiciones farmacéuticas que los contienen
CU2019000097A CU20190097A7 (es) 2017-03-15 2018-03-14 Compuestos derivados de 2-(benciloxi)-anilina n-substituidos como inhibidores de la función mitocondrial y composiciones farmacéuticas que los contienen

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