CS94391A2 - Carbapenemic compounds and method of their production - Google Patents
Carbapenemic compounds and method of their production Download PDFInfo
- Publication number
- CS94391A2 CS94391A2 CS91943A CS94391A CS94391A2 CS 94391 A2 CS94391 A2 CS 94391A2 CS 91943 A CS91943 A CS 91943A CS 94391 A CS94391 A CS 94391A CS 94391 A2 CS94391 A2 CS 94391A2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- group
- hydrogen
- methyl
- oxo
- formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
- C07D477/10—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D477/12—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
- C07D477/14—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 3
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
- C07D477/26—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 4
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US50613590A | 1990-04-09 | 1990-04-09 |
Publications (1)
Publication Number | Publication Date |
---|---|
CS94391A2 true CS94391A2 (en) | 1991-11-12 |
Family
ID=24013339
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS91943A CS94391A2 (en) | 1990-04-09 | 1991-04-05 | Carbapenemic compounds and method of their production |
Country Status (17)
Country | Link |
---|---|
EP (1) | EP0451764A1 (fi) |
JP (1) | JPH04234884A (fi) |
AU (1) | AU7420591A (fi) |
BR (1) | BR9101418A (fi) |
CA (1) | CA2039987A1 (fi) |
CS (1) | CS94391A2 (fi) |
FI (1) | FI911666A (fi) |
HU (1) | HUT57769A (fi) |
IE (1) | IE911161A1 (fi) |
IL (1) | IL97797A0 (fi) |
MC (1) | MC2262A1 (fi) |
MX (1) | MX25231A (fi) |
NO (1) | NO911357L (fi) |
PT (1) | PT97287A (fi) |
TW (1) | TW216420B (fi) |
YU (1) | YU62991A (fi) |
ZA (1) | ZA912279B (fi) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2001203C (en) * | 1988-10-24 | 2001-02-13 | Thomas P. Demuth, Jr. | Novel antimicrobial dithiocarbamoyl quinolones |
US5328908A (en) * | 1988-10-24 | 1994-07-12 | Procter & Gamble Pharmaceuticals, Inc. | Antimicrobial quinolone thioureas |
EP0997466A1 (en) * | 1988-10-24 | 2000-05-03 | PROCTER & GAMBLE PHARMACEUTICALS, INC. | Novel antimicrobial lactam-quinolones |
US5180719A (en) * | 1988-10-24 | 1993-01-19 | Norwich Eaton Pharmaceuticals, Inc. | Antimicrobial quinolonyl lactam esters |
US5491139A (en) * | 1988-10-24 | 1996-02-13 | The Procter & Gamble Company | Antimicrobial quinolonyl lactams |
US5273973A (en) * | 1988-10-24 | 1993-12-28 | Norwich Eaton Pharmaceuticals, Inc. | Antimicrobial quinolonyl esters |
JPH05506033A (ja) * | 1990-04-18 | 1993-09-02 | ノーウィッチ、イートン、ファーマスーティカルズ、インコーポレーテッド | 抗微生物性キノロニルラクタム類 |
HUT67423A (en) * | 1991-10-01 | 1995-04-28 | Procter & Gamble Pharma | Process for the production of antimicrobal compounds containing quinolone moiety and beta-lactam moiety |
DE4234078A1 (de) * | 1992-10-09 | 1994-04-14 | Bayer Ag | Chinoloncarbonsäuren |
DE4234330A1 (de) * | 1992-10-12 | 1994-04-14 | Bayer Ag | Chinoloncarbonsäuren |
EP0775145A1 (en) * | 1994-08-02 | 1997-05-28 | The Procter & Gamble Company | Process for making quinolonyl lactam antimicrobials and novel intermediate compounds |
ATE190972T1 (de) * | 1994-08-02 | 2000-04-15 | Procter & Gamble | Verfahren zur herstellung von antimikrobiellen verbindungen |
US5607928A (en) * | 1994-08-05 | 1997-03-04 | Zeneca Limited | Carbapenem derivatives containing a bicyclic ketone substituent and their use as anti-infectives |
EP0695753A1 (en) * | 1994-08-05 | 1996-02-07 | Zeneca Limited | Carbapenem derivatives containing a bicyclic substituent, process for their preparation, and their use |
US5973142A (en) * | 1997-01-21 | 1999-10-26 | Yasuda; Nobuyoshi | Process for synthesizing carbapenem intermediates |
CA2276365A1 (en) * | 1997-01-21 | 1998-07-23 | Merck & Co., Inc. | Process for synthesizing carbapenem intermediates |
US6080854A (en) * | 1997-08-25 | 2000-06-27 | Merck & Co., Inc. | Process for synthesizing carbapenem intermediates |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA1179675A (en) * | 1981-01-30 | 1984-12-18 | Erwin Gotschi | 7-oxo-1-azabicyclo ¬3,2,0| heptene-2-derivatives |
US4680292A (en) * | 1984-12-13 | 1987-07-14 | Merck & Co., Inc. | Carbapenems and 1-methylcarbapenems having a 2-heteroaryliumaliphatic substituent |
US4767762A (en) * | 1985-12-23 | 1988-08-30 | Abbott Laboratories | Tricyclic quinoline and naphthyride antibacterials |
EP0997466A1 (en) * | 1988-10-24 | 2000-05-03 | PROCTER & GAMBLE PHARMACEUTICALS, INC. | Novel antimicrobial lactam-quinolones |
EP0366193A3 (en) * | 1988-10-24 | 1992-01-08 | Norwich Eaton Pharmaceuticals, Inc. | Novel antimicrobial quinolonyl lactams |
EP0366641B1 (en) * | 1988-10-24 | 2000-07-05 | Norwich Eaton Pharmaceuticals, Inc. | Novel antimicrobial quinolonyl lactam esters |
-
1991
- 1991-03-26 ZA ZA912279A patent/ZA912279B/xx unknown
- 1991-04-05 JP JP3099750A patent/JPH04234884A/ja active Pending
- 1991-04-05 MC MC932182A patent/MC2262A1/xx unknown
- 1991-04-05 MX MX2523191A patent/MX25231A/es unknown
- 1991-04-05 CS CS91943A patent/CS94391A2/cs unknown
- 1991-04-08 TW TW080102600A patent/TW216420B/zh active
- 1991-04-08 FI FI911666A patent/FI911666A/fi not_active Application Discontinuation
- 1991-04-08 NO NO91911357A patent/NO911357L/no unknown
- 1991-04-08 AU AU74205/91A patent/AU7420591A/en not_active Abandoned
- 1991-04-08 YU YU62991A patent/YU62991A/sh unknown
- 1991-04-08 IL IL97797A patent/IL97797A0/xx unknown
- 1991-04-08 HU HU911132A patent/HUT57769A/hu unknown
- 1991-04-08 CA CA002039987A patent/CA2039987A1/en not_active Abandoned
- 1991-04-08 EP EP91105550A patent/EP0451764A1/en not_active Withdrawn
- 1991-04-08 IE IE116191A patent/IE911161A1/en unknown
- 1991-04-08 PT PT97287A patent/PT97287A/pt not_active Application Discontinuation
- 1991-04-09 BR BR919101418A patent/BR9101418A/pt unknown
Also Published As
Publication number | Publication date |
---|---|
FI911666A (fi) | 1991-10-10 |
EP0451764A1 (en) | 1991-10-16 |
IL97797A0 (en) | 1992-06-21 |
MX25231A (es) | 1993-10-01 |
NO911357L (no) | 1991-10-10 |
MC2262A1 (fr) | 1993-04-26 |
AU7420591A (en) | 1991-10-10 |
PT97287A (pt) | 1992-01-31 |
YU62991A (sh) | 1994-04-05 |
IE911161A1 (en) | 1991-10-09 |
ZA912279B (en) | 1992-02-26 |
HU911132D0 (en) | 1991-10-28 |
FI911666A0 (fi) | 1991-04-08 |
TW216420B (fi) | 1993-11-21 |
JPH04234884A (ja) | 1992-08-24 |
HUT57769A (en) | 1991-12-30 |
CA2039987A1 (en) | 1991-10-10 |
NO911357D0 (no) | 1991-04-08 |
BR9101418A (pt) | 1991-11-26 |
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