CS226907B1 - Alkylamides of carboxyalkanoylpeptides - Google Patents
Alkylamides of carboxyalkanoylpeptides Download PDFInfo
- Publication number
- CS226907B1 CS226907B1 CS815977A CS597781A CS226907B1 CS 226907 B1 CS226907 B1 CS 226907B1 CS 815977 A CS815977 A CS 815977A CS 597781 A CS597781 A CS 597781A CS 226907 B1 CS226907 B1 CS 226907B1
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- alanine
- alanyl
- ethylamide
- formula
- ala
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- C07K5/06165—Dipeptides with the first amino acid being heterocyclic and Pro-amino acid; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06008—Dipeptides with the first amino acid being neutral
- C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
- C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
- C07K5/0806—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Priority Applications (11)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CS815977A CS226907B1 (en) | 1981-08-07 | 1981-08-07 | Alkylamides of carboxyalkanoylpeptides |
IT22506/82A IT1156108B (it) | 1981-08-07 | 1982-07-21 | Alchilamidi di carbossialcanoil peptidi |
FR8213346A FR2510990B1 (fr) | 1981-08-07 | 1982-07-30 | Alcoylamides de carboxyalcanoylpeptides |
JP57134793A JPS5849351A (ja) | 1981-08-07 | 1982-08-03 | カルボキシアルカノイルペプチドのアルキルアミド |
CA000408760A CA1238902A (en) | 1981-08-07 | 1982-08-05 | Alkylamides of carboxyalkanoyl peptides |
GB08222574A GB2104082B (en) | 1981-08-07 | 1982-08-05 | Alkylamides of carboxyalkanoyl peptides |
HU822541A HU193029B (en) | 1981-08-07 | 1982-08-06 | Process for preparing carboxy-alkanoyl-peptide-alkylamide derivatives |
CH4752/82A CH653038A5 (de) | 1981-08-07 | 1982-08-06 | Carboxyalkanoylpeptid-alkylamide. |
US06/406,168 US4554100A (en) | 1981-08-07 | 1982-08-09 | Alkylamides of carboxyalkanoyl peptides and method for preparation thereof |
DE19823229632 DE3229632A1 (de) | 1981-08-07 | 1982-08-09 | Carboxyalkanoylpeptid-alkylamide, ihre herstellung und pharmazeutische mittel |
BE0/208777A BE894065A (fr) | 1981-08-07 | 1982-08-09 | Alkylamides de carboxy-alcanoyl-peptides |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CS815977A CS226907B1 (en) | 1981-08-07 | 1981-08-07 | Alkylamides of carboxyalkanoylpeptides |
Publications (1)
Publication Number | Publication Date |
---|---|
CS226907B1 true CS226907B1 (en) | 1984-04-16 |
Family
ID=5405786
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS815977A CS226907B1 (en) | 1981-08-07 | 1981-08-07 | Alkylamides of carboxyalkanoylpeptides |
Country Status (11)
Country | Link |
---|---|
US (1) | US4554100A (de) |
JP (1) | JPS5849351A (de) |
BE (1) | BE894065A (de) |
CA (1) | CA1238902A (de) |
CH (1) | CH653038A5 (de) |
CS (1) | CS226907B1 (de) |
DE (1) | DE3229632A1 (de) |
FR (1) | FR2510990B1 (de) |
GB (1) | GB2104082B (de) |
HU (1) | HU193029B (de) |
IT (1) | IT1156108B (de) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CS231228B1 (en) * | 1982-10-01 | 1984-10-15 | Evzen Kasafirek | Biologically effective tri and tetrapeptide alkylamide derivatives and their processing method |
DE3481913D1 (de) * | 1983-04-27 | 1990-05-17 | Ici America Inc | Prolin-derivate. |
AU583578B2 (en) * | 1984-12-14 | 1989-05-04 | Australian Commercial Research & Development Limited | Amino acid and peptide inhibitors of human leucocytic elastase |
FR2733995B1 (fr) * | 1995-05-09 | 1997-07-25 | Inst Nat Sante Rech Med | Inhibiteurs de l'inactivation de neuropeptides endogenes notamment la cholecystokinine, leurs procedes de preparation leur utilisation comme medicaments et procede de criblage de medicaments |
ES2828717T3 (es) | 2015-06-24 | 2021-05-27 | Nitto Denko Corp | Compuestos ionizables y composiciones y usos de los mismos |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4029772A (en) * | 1975-12-23 | 1977-06-14 | Merck & Co., Inc. | Peptide carbazates |
US4064236A (en) * | 1975-12-23 | 1977-12-20 | Merck & Co., Inc. | Peptide carbazates and pharmaceutical composition |
CH626872A5 (de) * | 1976-06-21 | 1981-12-15 | Hoffmann La Roche | |
PH14141A (en) * | 1976-06-25 | 1981-03-05 | Hoffmann La Roche | Pharmaceutical composition containing dipeptide derivatives |
FR2381023A1 (fr) * | 1977-02-18 | 1978-09-15 | Delalande Sa | Nouveaux oligopeptides trifluoromethyles derives de la l-alanine, leur procede de preparation et leur application en therapeutique |
IL58849A (en) * | 1978-12-11 | 1983-03-31 | Merck & Co Inc | Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them |
-
1981
- 1981-08-07 CS CS815977A patent/CS226907B1/cs unknown
-
1982
- 1982-07-21 IT IT22506/82A patent/IT1156108B/it active
- 1982-07-30 FR FR8213346A patent/FR2510990B1/fr not_active Expired
- 1982-08-03 JP JP57134793A patent/JPS5849351A/ja active Granted
- 1982-08-05 GB GB08222574A patent/GB2104082B/en not_active Expired
- 1982-08-05 CA CA000408760A patent/CA1238902A/en not_active Expired
- 1982-08-06 CH CH4752/82A patent/CH653038A5/de not_active IP Right Cessation
- 1982-08-06 HU HU822541A patent/HU193029B/hu not_active IP Right Cessation
- 1982-08-09 US US06/406,168 patent/US4554100A/en not_active Expired - Fee Related
- 1982-08-09 BE BE0/208777A patent/BE894065A/fr not_active IP Right Cessation
- 1982-08-09 DE DE19823229632 patent/DE3229632A1/de active Granted
Also Published As
Publication number | Publication date |
---|---|
IT1156108B (it) | 1987-01-28 |
JPS5849351A (ja) | 1983-03-23 |
DE3229632C2 (de) | 1988-06-23 |
CH653038A5 (de) | 1985-12-13 |
GB2104082B (en) | 1984-09-12 |
CA1238902A (en) | 1988-07-05 |
FR2510990B1 (fr) | 1986-05-09 |
BE894065A (fr) | 1982-12-01 |
US4554100A (en) | 1985-11-19 |
HU193029B (en) | 1987-08-28 |
IT8222506A1 (it) | 1984-01-21 |
FR2510990A1 (fr) | 1983-02-11 |
DE3229632A1 (de) | 1983-02-24 |
IT8222506A0 (it) | 1982-07-21 |
JPH0349918B2 (de) | 1991-07-31 |
GB2104082A (en) | 1983-03-02 |
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