CS203184B2 - Process for preparing new pyrroloquinoxalinones and pyrrolobenzodiazepinones - Google Patents
Process for preparing new pyrroloquinoxalinones and pyrrolobenzodiazepinones Download PDFInfo
- Publication number
- CS203184B2 CS203184B2 CS781094A CS109478A CS203184B2 CS 203184 B2 CS203184 B2 CS 203184B2 CS 781094 A CS781094 A CS 781094A CS 109478 A CS109478 A CS 109478A CS 203184 B2 CS203184 B2 CS 203184B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- phenyl
- acid
- dihydro
- calculated
- atom
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
- C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
- C07D241/40—Benzopyrazines
- C07D241/44—Benzopyrazines with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CS792091A CS203185B2 (cs) | 1977-02-25 | 1979-03-29 | Způsob výroby 6-hydroxy-6-fenyl-lH-pyrrolo[1,2,3-de ]- -chinoxalin-2,5 (3H,6H) dionu |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/772,154 US4075206A (en) | 1977-02-25 | 1977-02-25 | Substituted pyrroloquinoxalinones and diones |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS203184B2 true CS203184B2 (en) | 1981-02-27 |
Family
ID=25094096
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS781094A CS203184B2 (en) | 1977-02-25 | 1978-02-21 | Process for preparing new pyrroloquinoxalinones and pyrrolobenzodiazepinones |
Country Status (26)
| Country | Link |
|---|---|
| US (2) | US4075206A (xx) |
| JP (1) | JPS53111095A (xx) |
| AR (1) | AR218056A1 (xx) |
| AT (1) | AT361489B (xx) |
| AU (1) | AU513391B2 (xx) |
| BE (1) | BE864105A (xx) |
| BG (1) | BG28565A3 (xx) |
| CA (1) | CA1097631A (xx) |
| CS (1) | CS203184B2 (xx) |
| DD (1) | DD134871A5 (xx) |
| DE (1) | DE2807145A1 (xx) |
| DK (1) | DK74578A (xx) |
| ES (1) | ES467189A1 (xx) |
| FR (1) | FR2381767A1 (xx) |
| GB (1) | GB1595745A (xx) |
| GR (1) | GR68942B (xx) |
| IL (1) | IL54086A0 (xx) |
| IT (1) | IT1094215B (xx) |
| NL (1) | NL7801927A (xx) |
| NZ (1) | NZ186512A (xx) |
| PH (1) | PH13147A (xx) |
| PL (1) | PL204796A1 (xx) |
| PT (1) | PT67678B (xx) |
| SE (1) | SE7802024L (xx) |
| YU (1) | YU39178A (xx) |
| ZA (1) | ZA78991B (xx) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4262123A (en) * | 1978-09-11 | 1981-04-14 | The Upjohn Company | Quinoxalinones |
| US4242342A (en) * | 1979-05-31 | 1980-12-30 | The Upjohn Company | Quinoxalinones useful for treating atopic eczema and urticaria |
| US4499270A (en) * | 1981-04-16 | 1985-02-12 | Riker Laboratories, Inc. | Substituted pyridoquinoxaline-6-carboxylic acids and derivatives thereof |
| IL93136A (en) * | 1989-02-23 | 1995-01-24 | Janssen Pharmaceutica Nv | History of tetrahydroimidazo [1,4] benzodiazepine-2-thione, their preparation and pharmaceutical preparations containing them |
| NZ235137A (en) * | 1989-09-13 | 1992-02-25 | Janssen Pharmaceutica Nv | Tetrahydroimidazo(1,4)benzodiazepine derivatives, preparation and pharmaceutical compositions thereof |
| JPH05117276A (ja) * | 1991-10-23 | 1993-05-14 | Sumitomo Pharmaceut Co Ltd | 新規な３環性キノキサリンジオン誘導体 |
| TW260660B (xx) * | 1993-04-22 | 1995-10-21 | Sumitomo Pharma | |
| CN114230528B (zh) * | 2021-11-25 | 2024-02-06 | 桂林理工大学 | 一种制备喹喔啉酮衍生物的方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3892746A (en) * | 1969-06-09 | 1975-07-01 | American Home Prod | Pyrrolo{8 1,2,3-de{9 quinoxalin-2(3H)-ones and related compounds |
| US3813392A (en) * | 1969-06-09 | 1974-05-28 | J Sellstedt | Pyrrolo(1,2,3-alpha epsilon)quinoxalin-2(3h)-ones and related compounds |
| US3642821A (en) * | 1969-11-03 | 1972-02-15 | Upjohn Co | Tetrahydropyrrolobenzodiazepines |
| US3579503A (en) * | 1969-11-03 | 1971-05-18 | Upjohn Co | Pyrrolo(3,2,1-jk)(1,4)benzodiazepinones |
-
1977
- 1977-02-25 US US05/772,154 patent/US4075206A/en not_active Expired - Lifetime
- 1977-09-26 US US05/836,830 patent/US4087527A/en not_active Expired - Lifetime
-
1978
- 1978-02-17 GB GB6298/78A patent/GB1595745A/en not_active Expired
- 1978-02-20 DE DE19782807145 patent/DE2807145A1/de not_active Withdrawn
- 1978-02-20 BE BE1008716A patent/BE864105A/xx unknown
- 1978-02-20 PT PT67678A patent/PT67678B/pt unknown
- 1978-02-20 FR FR7804728A patent/FR2381767A1/fr active Pending
- 1978-02-20 IT IT20417/78A patent/IT1094215B/it active
- 1978-02-20 NZ NZ186512A patent/NZ186512A/xx unknown
- 1978-02-20 ZA ZA00780991A patent/ZA78991B/xx unknown
- 1978-02-20 CA CA297,309A patent/CA1097631A/en not_active Expired
- 1978-02-20 AU AU33433/78A patent/AU513391B2/en not_active Expired
- 1978-02-20 IL IL54086A patent/IL54086A0/xx unknown
- 1978-02-20 JP JP1902178A patent/JPS53111095A/ja active Pending
- 1978-02-20 DK DK74578A patent/DK74578A/da unknown
- 1978-02-20 GR GR55496A patent/GR68942B/el unknown
- 1978-02-20 PH PH20799A patent/PH13147A/en unknown
- 1978-02-20 AR AR271156A patent/AR218056A1/es active
- 1978-02-21 DD DD78203784A patent/DD134871A5/xx unknown
- 1978-02-21 CS CS781094A patent/CS203184B2/cs unknown
- 1978-02-21 NL NL7801927A patent/NL7801927A/xx not_active Application Discontinuation
- 1978-02-21 ES ES467189A patent/ES467189A1/es not_active Expired
- 1978-02-21 SE SE7802024A patent/SE7802024L/xx unknown
- 1978-02-21 YU YU00391/78A patent/YU39178A/xx unknown
- 1978-02-21 BG BG038764A patent/BG28565A3/xx unknown
- 1978-02-21 PL PL20479678A patent/PL204796A1/xx unknown
- 1978-02-23 AT AT131578A patent/AT361489B/de not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| US4087527A (en) | 1978-05-02 |
| PL204796A1 (pl) | 1979-04-09 |
| AU513391B2 (en) | 1980-11-27 |
| FR2381767A1 (fr) | 1978-09-22 |
| GR68942B (xx) | 1982-03-29 |
| GB1595745A (en) | 1981-08-19 |
| SE7802024L (sv) | 1978-08-26 |
| IT1094215B (it) | 1985-07-26 |
| AT361489B (de) | 1981-03-10 |
| PT67678B (en) | 1979-07-20 |
| US4075206A (en) | 1978-02-21 |
| AU3343378A (en) | 1979-08-30 |
| CA1097631A (en) | 1981-03-17 |
| BG28565A3 (bg) | 1980-05-15 |
| IL54086A0 (en) | 1978-04-30 |
| BE864105A (fr) | 1978-08-21 |
| NL7801927A (nl) | 1978-08-29 |
| ES467189A1 (es) | 1979-08-16 |
| ZA78991B (en) | 1979-10-31 |
| AR218056A1 (es) | 1980-05-15 |
| DK74578A (da) | 1978-08-26 |
| DE2807145A1 (de) | 1978-08-31 |
| YU39178A (en) | 1983-01-21 |
| NZ186512A (en) | 1981-03-16 |
| DD134871A5 (de) | 1979-03-28 |
| IT7820417A0 (it) | 1978-02-20 |
| PH13147A (en) | 1979-12-18 |
| PT67678A (en) | 1978-03-01 |
| ATA131578A (de) | 1980-08-15 |
| JPS53111095A (en) | 1978-09-28 |
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