CS197217B2 - Method of conversion of penicilin sulphoxide into deacetoxy cephalosporin and lithium salt of the same - Google Patents

Method of conversion of penicilin sulphoxide into deacetoxy cephalosporin and lithium salt of the same Download PDF

Info

Publication number
CS197217B2
CS197217B2 CS733319A CS331973A CS197217B2 CS 197217 B2 CS197217 B2 CS 197217B2 CS 733319 A CS733319 A CS 733319A CS 331973 A CS331973 A CS 331973A CS 197217 B2 CS197217 B2 CS 197217B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
phenyl
acid
group
methyl
Prior art date
Application number
CS733319A
Other languages
Czech (cs)
English (en)
Inventor
Ta-Sen Chou
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Priority to CS773703A priority Critical patent/CS197218B2/cs
Publication of CS197217B2 publication Critical patent/CS197217B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0834—Compounds having one or more O-Si linkage
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/09—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4
    • C07D205/095—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a sulfur atom directly attached in position 4 and with a nitrogen atom directly attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/10—Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage
CS733319A 1972-05-10 1973-05-10 Method of conversion of penicilin sulphoxide into deacetoxy cephalosporin and lithium salt of the same CS197217B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS773703A CS197218B2 (cs) 1972-05-10 1977-06-06 Způsob výroby nových silylesterů azetidin-2-sulíenátů

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25207872A 1972-05-10 1972-05-10
US05/349,876 US3944545A (en) 1972-05-10 1973-04-12 Process for preparing desacetoxycephalosporins

Publications (1)

Publication Number Publication Date
CS197217B2 true CS197217B2 (en) 1980-04-30

Family

ID=26942026

Family Applications (1)

Application Number Title Priority Date Filing Date
CS733319A CS197217B2 (en) 1972-05-10 1973-05-10 Method of conversion of penicilin sulphoxide into deacetoxy cephalosporin and lithium salt of the same

Country Status (21)

Country Link
US (1) US3944545A (ja)
JP (2) JPS5418276B2 (ja)
AR (1) AR203722A1 (ja)
AT (1) AT333424B (ja)
AU (1) AU476568B2 (ja)
BG (2) BG20816A3 (ja)
CA (1) CA1026744A (ja)
CH (2) CH582187A5 (ja)
CS (1) CS197217B2 (ja)
DD (2) DD108302A5 (ja)
DE (1) DE2323395A1 (ja)
ES (1) ES414645A1 (ja)
FR (1) FR2184069B1 (ja)
GB (1) GB1412856A (ja)
HU (2) HU170406B (ja)
IE (1) IE38150B1 (ja)
IL (1) IL42148A (ja)
NL (1) NL7306500A (ja)
PH (1) PH14066A (ja)
SE (2) SE429046B (ja)
YU (1) YU36925B (ja)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA732972B (en) * 1972-05-10 1974-11-27 Lilly Co Eli Process for preparing desacetoxycephalosporins and novel intermediates
GB1465893A (en) * 1973-02-09 1977-03-02 Gist Brocades Nv I-carboxypropenyl-4-iminothio-azetidine-2-one derivatives methods for their preparation and use
US4159266A (en) * 1974-12-24 1979-06-26 Eli Lilly And Company Method of preparation of 3-methylenecephams
AT342197B (de) * 1975-02-20 1978-03-28 Ciba Geigy Ag Neues verfahren zur herstellung von 3-cephemverbindungen
JPS5214789A (en) * 1975-07-22 1977-02-03 Shionogi & Co Ltd Process for preparing 3-substiuted cephem compounds by ring closure
US4536334A (en) * 1979-06-28 1985-08-20 Sumitomo Chemical Company, Limited Preparation of β-lactam derivatives
US5302713A (en) * 1992-03-31 1994-04-12 Industrial Technology Research Institute Method for the preparation of Δ3 -7-substituted amino desacetoxy cephalosporanic acid

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3591585A (en) * 1969-02-14 1971-07-06 Lilly Co Eli Process for making desacetoxycephalosporins
NL159389B (nl) * 1969-03-11 1979-02-15 Glaxo Lab Ltd Werkwijze ter bereiding van 7beta-acylamido-3-methylcef-3-em-4-carbonzuuresters.
US3819622A (en) * 1969-03-11 1974-06-25 Glaxo Lab Ltd Method of producing 7beta-acylamido-3-methylceph-3-em-4-carboxylic acid esters
GB1312233A (en) * 1969-12-05 1973-04-04 Glaxo Lab Ltd Cephalosporin compounds

Also Published As

Publication number Publication date
AT333424B (de) 1976-11-25
DD108302A5 (ja) 1974-09-12
CH580638A5 (ja) 1976-10-15
BG20816A3 (ja) 1975-12-20
CA1026744A (en) 1978-02-21
IL42148A0 (en) 1973-06-29
HU166698B (ja) 1975-05-28
BG20380A3 (ja) 1975-11-05
HU170406B (en) 1977-06-28
IL42148A (en) 1976-08-31
SE429046B (sv) 1983-08-08
ATA410573A (de) 1976-03-15
PH14066A (en) 1981-01-26
IE38150B1 (en) 1978-01-04
CH582187A5 (ja) 1976-11-30
AR203722A1 (es) 1975-10-15
YU36925B (en) 1984-08-31
AU476568B2 (en) 1976-09-30
YU121973A (en) 1982-06-18
SE7604463L (sv) 1976-04-16
FR2184069B1 (ja) 1975-08-22
JPS585917B2 (ja) 1983-02-02
FR2184069A1 (ja) 1973-12-21
GB1412856A (en) 1975-11-05
JPS5418276B2 (ja) 1979-07-06
AU5519773A (en) 1974-11-07
JPS5444657A (en) 1979-04-09
ES414645A1 (es) 1976-06-16
NL7306500A (ja) 1973-11-13
SE429968B (sv) 1983-10-10
IE38150L (en) 1973-11-10
US3944545A (en) 1976-03-16
DE2323395A1 (de) 1973-11-29
DD116617A5 (ja) 1975-12-05
JPS4947388A (ja) 1974-05-08

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