CR8428A - Agente endoparasiticidas para la administracion topica - Google Patents

Agente endoparasiticidas para la administracion topica

Info

Publication number
CR8428A
CR8428A CR8428A CR8428A CR8428A CR 8428 A CR8428 A CR 8428A CR 8428 A CR8428 A CR 8428A CR 8428 A CR8428 A CR 8428A CR 8428 A CR8428 A CR 8428A
Authority
CR
Costa Rica
Prior art keywords
endoparasiticid
agent
topical administration
depsipeptides
praziquantel
Prior art date
Application number
CR8428A
Other languages
English (en)
Inventor
Kanikanti Venkata-Rangarao
Bach Thomas
Altreuther Gertraut
Traubel Michael
Jurgen Hamann Hans
Original Assignee
Bayer Animal Health Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Animal Health Gmbh filed Critical Bayer Animal Health Gmbh
Publication of CR8428A publication Critical patent/CR8428A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • A61K9/0017Non-human animal skin, e.g. pour-on, spot-on
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/04Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15Depsipeptides; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Dermatology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La presente invencion se refiere a agentes de administracion transdermica que contienen depsipeptidos ciclicos y/ o prazicuantel, asi como a su preparacion y uso para combatir endoparasitos.
CR8428A 2003-12-13 2006-06-01 Agente endoparasiticidas para la administracion topica CR8428A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10358525A DE10358525A1 (de) 2003-12-13 2003-12-13 Endoparasitizide Mittel zur topischen Applikation

Publications (1)

Publication Number Publication Date
CR8428A true CR8428A (es) 2006-11-23

Family

ID=34638681

Family Applications (1)

Application Number Title Priority Date Filing Date
CR8428A CR8428A (es) 2003-12-13 2006-06-01 Agente endoparasiticidas para la administracion topica

Country Status (32)

Country Link
US (1) US7763583B2 (es)
EP (1) EP1694291B1 (es)
JP (1) JP4842141B2 (es)
KR (1) KR101272139B1 (es)
CN (1) CN1893919B (es)
AR (1) AR046878A1 (es)
AT (1) ATE447940T1 (es)
AU (1) AU2004296537B2 (es)
BR (1) BRPI0417578B1 (es)
CA (1) CA2548897C (es)
CR (1) CR8428A (es)
DE (2) DE10358525A1 (es)
DK (1) DK1694291T3 (es)
ES (1) ES2334920T3 (es)
GT (1) GT200400264A (es)
HK (1) HK1102915A1 (es)
HR (1) HRP20100056T1 (es)
IL (1) IL176151A (es)
MX (1) MXPA06006594A (es)
MY (1) MY142044A (es)
NO (1) NO20063171L (es)
NZ (1) NZ547837A (es)
PE (1) PE20050919A1 (es)
PL (1) PL1694291T3 (es)
PT (1) PT1694291E (es)
RU (1) RU2401108C2 (es)
SI (1) SI1694291T1 (es)
TW (1) TWI341202B (es)
UA (1) UA85574C2 (es)
UY (1) UY28662A1 (es)
WO (1) WO2005055973A2 (es)
ZA (1) ZA200604744B (es)

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US20070148228A1 (en) * 1999-02-22 2007-06-28 Merrion Research I Limited Solid oral dosage form containing an enhancer
US7658938B2 (en) 1999-02-22 2010-02-09 Merrion Reasearch III Limited Solid oral dosage form containing an enhancer
US8119159B2 (en) 1999-02-22 2012-02-21 Merrion Research Iii Limited Solid oral dosage form containing an enhancer
DE102004055316A1 (de) * 2004-11-16 2006-05-18 Bayer Healthcare Ag Verhinderung vertikaler Endoparasiten-Infektionen
DE102005011779A1 (de) * 2005-03-11 2006-09-14 Bayer Healthcare Ag Endoparasitizide Mittel
US7704977B2 (en) 2006-04-07 2010-04-27 Merrion Research Iii Limited Solid oral dosage form containing an enhancer
EP2040731A4 (en) * 2006-06-09 2010-05-19 Merrion Res Iii Ltd SOLID DOSAGE FORM FOR ORAL ADMINISTRATION CONTAINING AN ACTIVATOR
PE20081406A1 (es) * 2006-12-20 2008-10-17 Schering Plough Ltd Composiciones farmaceuticas de flunixina
WO2009137078A1 (en) * 2008-05-07 2009-11-12 Merrion Research Iii Limited Compositions of peptides and processes of preparation thereof
DE102008022520A1 (de) * 2008-05-07 2009-11-12 Bayer Animal Health Gmbh Feste Arzneimittelformulierung mit verzögerter Freisetzung
ES2617672T3 (es) * 2008-10-08 2017-06-19 Zoetis Services Llc Composiciones antihelmínticas de bencimidazol
US20100215743A1 (en) * 2009-02-25 2010-08-26 Leonard Thomas W Composition and drug delivery of bisphosphonates
DE102009012423A1 (de) 2009-03-10 2010-09-16 Bayer Animal Health Gmbh Zubereitung auf Ölbasis
BRPI1009199A2 (pt) 2009-03-17 2016-03-08 Concert Pharmaceuticals Inc compostos de pirazinoisoquinolina
WO2011013003A2 (en) 2009-07-31 2011-02-03 Shin Nippon Biomedical Laboratories, Ltd. Intranasal granisetron and nasal applicator
US20110182985A1 (en) * 2010-01-28 2011-07-28 Coughlan David C Solid Pharmaceutical Composition with Enhancers and Methods of Preparing thereof
US9089484B2 (en) 2010-03-26 2015-07-28 Merrion Research Iii Limited Pharmaceutical compositions of selective factor Xa inhibitors for oral administration
KR20140026354A (ko) 2011-01-07 2014-03-05 메리온 리서치 Ⅲ 리미티드 경구 투여용 철의 제약 조성물
US8680054B2 (en) * 2011-04-20 2014-03-25 Novartis Ag Suspension type topical formulations comprising cyclic depsipeptide
CN102283843A (zh) * 2011-06-29 2011-12-21 梁晓天 一种吡喹酮外用制剂及其制备方法和应用
MY175307A (en) * 2011-12-21 2020-06-18 Bayer Ip Gmbh Preparations comprising amorphous emodepside
MX350224B (es) * 2012-12-18 2017-08-30 Donaghys Ltd Formulaciones parasiticidas transdermicas.
JP2017505798A (ja) * 2014-02-14 2017-02-23 ディーエスエム アイピー アセッツ ビー.ブイ. 住血吸虫症を予防かつ/または治療するための組成物および方法
JP7211704B2 (ja) 2015-01-29 2023-01-24 ノヴォ ノルディスク アー/エス Glp-1アゴニスト及び腸溶コーティングを含む錠剤
BR112017024773A2 (pt) 2015-05-20 2018-11-06 Merial, Inc. compostos depsipeptídeos anti-helmínticos
CA3009867C (en) 2015-12-28 2022-05-31 Merial, Inc. Anthelmintic cyclic depsipeptide compounds
WO2018093920A1 (en) 2016-11-16 2018-05-24 Merial, Inc. Anthelmintic depsipeptide compounds
EP3480195A1 (en) 2017-11-07 2019-05-08 Bayer Animal Health GmbH Method for the synthesis of cyclic depsipeptides
MX2020004702A (es) 2017-11-07 2020-11-06 Bayer Animal Health Gmbh Metodo para la sintesis de depsipeptidos ciclicos.
CN111346046B (zh) * 2020-03-06 2021-07-09 安徽农业大学 一种含莫西菌素注射用缓释凝胶制剂及制备方法

Family Cites Families (24)

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Publication number Priority date Publication date Assignee Title
US281292A (en) * 1883-07-17 onslow
DE2362539C2 (de) * 1973-12-17 1986-05-07 Merck Patent Gmbh, 6100 Darmstadt 2-Acyl-4-oxo-1,2,3,6,7,11b-hexahydro-4H-pyrazino[2,1-a]isochinoline, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE3619030A1 (de) * 1986-06-06 1987-12-10 Bayer Ag Topisch anwendbare zubereitungen
DE3634755A1 (de) 1986-10-11 1988-04-14 Bayer Ag Dermale behandlung von wurmerkrankungen der katze mit praziquantel
NO176766C (no) 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
US5874479A (en) * 1991-03-01 1999-02-23 Warner-Lambert Company Therapeutic permeation enhanced-wound healing compositions and methods for preparing and using same
DE4317458A1 (de) 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
DE4317432A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4317457A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4400464A1 (de) * 1994-01-11 1995-07-13 Bayer Ag Endoparasitizide Mittel
NZ260018A (en) 1994-03-03 1995-10-26 Bomac Lab Ltd Benzimidazole compositions and anthelmintic compositions
DE19520275A1 (de) * 1995-06-02 1996-12-05 Bayer Ag Endoparasitizide Mittel
US5780487A (en) 1995-08-07 1998-07-14 Amer Moh Samir S-2'- 2-(1-methyl-2-piperidyl) ethyl! cinnamanilide
DE19601263A1 (de) 1996-01-16 1997-07-17 Bayer Ag Anthelmintische Paste
DE19628776A1 (de) 1996-07-17 1998-01-22 Bayer Ag Oral applizierbare Granulate von Hexahydropyrazinderivaten
US5837289A (en) * 1996-07-23 1998-11-17 Grasela; John C. Transdermal delivery of medications using a combination of penetration enhancers
DE19921887A1 (de) 1999-05-12 2000-11-16 Bayer Ag Endoparasitizide Mittel
DE19941024A1 (de) 1999-08-28 2001-03-01 Hartmut Klocke Wirkstoffpräparat für tierärztliche Applikation und Verfahren zu seiner Herstellung
US6340672B1 (en) 2000-02-16 2002-01-22 Phoenix Scientific, Inc. Parasiticidal formulation and a method of making this formulation
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
ATE320812T1 (de) 2000-10-10 2006-04-15 Wyeth Corp Anthelmintika
GB0108485D0 (en) 2001-04-04 2001-05-23 Pfizer Ltd Combination therapy
US6893652B2 (en) 2001-08-27 2005-05-17 Wyeth Endoparasiticidal gel composition
CA2521268C (en) * 2003-04-04 2012-10-16 Merial Ltd. Topical anthelmintic veterinary formulations

Also Published As

Publication number Publication date
PE20050919A1 (es) 2005-12-16
KR101272139B1 (ko) 2013-06-10
CA2548897A1 (en) 2005-06-23
ES2334920T3 (es) 2010-03-17
DK1694291T3 (da) 2010-03-15
RU2006124964A (ru) 2008-01-20
GT200400264A (es) 2005-08-18
CA2548897C (en) 2012-04-10
CN1893919B (zh) 2010-09-29
NO20063171L (no) 2006-07-07
RU2401108C2 (ru) 2010-10-10
JP4842141B2 (ja) 2011-12-21
SI1694291T1 (sl) 2010-03-31
DE10358525A1 (de) 2005-07-07
UA85574C2 (uk) 2009-02-10
AR046878A1 (es) 2005-12-28
ZA200604744B (en) 2007-09-26
DE502004010367D1 (de) 2009-12-24
HK1102915A1 (en) 2007-12-07
MXPA06006594A (es) 2006-08-23
ATE447940T1 (de) 2009-11-15
EP1694291A2 (de) 2006-08-30
BRPI0417578A (pt) 2007-03-20
IL176151A (en) 2013-12-31
UY28662A1 (es) 2005-07-29
AU2004296537B2 (en) 2010-05-13
WO2005055973A2 (de) 2005-06-23
WO2005055973A3 (de) 2005-08-11
KR20060103953A (ko) 2006-10-04
PT1694291E (pt) 2010-01-18
HRP20100056T1 (hr) 2010-03-31
NZ547837A (en) 2010-02-26
AU2004296537A1 (en) 2005-06-23
BRPI0417578B1 (pt) 2015-12-22
MY142044A (en) 2010-08-30
US7763583B2 (en) 2010-07-27
JP2007513903A (ja) 2007-05-31
PL1694291T3 (pl) 2010-04-30
IL176151A0 (en) 2006-10-05
EP1694291B1 (de) 2009-11-11
US20070060509A1 (en) 2007-03-15
CN1893919A (zh) 2007-01-10
TW200533384A (en) 2005-10-16
TWI341202B (en) 2011-05-01

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