CO6420414A2 - Heterociclos microbicidas - Google Patents

Heterociclos microbicidas

Info

Publication number
CO6420414A2
CO6420414A2 CO12022024A CO12022024A CO6420414A2 CO 6420414 A2 CO6420414 A2 CO 6420414A2 CO 12022024 A CO12022024 A CO 12022024A CO 12022024 A CO12022024 A CO 12022024A CO 6420414 A2 CO6420414 A2 CO 6420414A2
Authority
CO
Colombia
Prior art keywords
alkyl
haloalkyl
phenyl
cyano
alkoxy
Prior art date
Application number
CO12022024A
Other languages
English (en)
Inventor
Sarah Sulzer-Mosse
Clemens Lamberth
Respondek Mathias Stephan
Laura Quaranta
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of CO6420414A2 publication Critical patent/CO6420414A2/es

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/761,3-Oxazoles; Hydrogenated 1,3-oxazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/74Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,3
    • A01N43/781,3-Thiazoles; Hydrogenated 1,3-thiazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/82Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with three ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/48Nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/28Radicals substituted by nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/081,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente invención trata acerca de compuestos heterocíclicos de fórmula (I) los cuales tienen actividad microbicida, en particular actividad fungicida, así como acerca de métodos de utilización de los compuestos de fórmula (I) para controlar microbios.en dondeA es x-C(=O)-, x-C(=S)-, x-C(R10R11)-C(=O)-, x-C(R12R13)-C(=S)-, x-O-C(=O)-, x-O-C(=S)-, x-N(R14)-C(=O)-, x-N(R15)-C(=S)-, x-C(R16R17)-SO2- o x-N=C(R26)-, en cada caso x representa el enlace que está conectado a R1;T es CR18 o N;G es O o S;Y1 y Y2 son independientemente CR19 o N;Q es -C(=O)-z, -C(=S)-z, -C(=O)-O-z, -C(=S)-O-z, -C(=O)-N(R20)-z, -C(=S)-N(R21)-z o -SO2-z-, en cada caso z representa el enlace que está conectado a R9 n es 1 o 2;p es 1 o 2, con la condición de que cuando n es 2, p es 1;R1 es fenilo, piridilo, imidazolilo, o pirazolilo; en donde cada uno de los fenilo, piridilo, imidazolilo y pirazolilo están sustituidos opcionalmente con entre 1 y 3 sustituyentes escogidos independientemente entre alquilo C1-C4, haloalquilo C1-C4, halógeno, ciano, hidroxi y amino;R2, R3, R4, R5, R6, R7, R10, R11, R12, R13, R16, R17, R18, R19 y R26 son, cada uno independientemente, hidrógeno, halógeno, ciano, alquilo C1-C4 o haloalquilo C1-C4, R8, R14, R15, R20 y R21 son, cada uno independientemente, hidrógeno, alquilo C1-C4 o alcoxi C1-C4 yR9 es fenilo, bencilo o el grupo (a):en donde cada uno de fenilo, bencilo y el grupo (a) están sustituidos opcionalmente con entre 1 y 3 sustituyentes escogidos independientemente entre alquilo C1-C4, haloalquilo C1-C4, alcoxi C1-C4, haloalcoxi C1-C4, halógeno, ciano, hidroxilo, N(R27)2, SH, alquiltio C1-C4, nitro, fenilsulfonilo y fenilsulfinilo, en donde el fenilsulfonilo y el fenilsulfinilo están sustituidos opcionalmente con entre 1 y 3 sustituyentes escogidos independientemente entre alquilo C1-C4, haloalquilo C1-C4, alcoxi C1-C4, ...
CO12022024A 2009-08-12 2012-02-08 Heterociclos microbicidas CO6420414A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP09167736 2009-08-12

Publications (1)

Publication Number Publication Date
CO6420414A2 true CO6420414A2 (es) 2012-04-16

Family

ID=43016641

Family Applications (1)

Application Number Title Priority Date Filing Date
CO12022024A CO6420414A2 (es) 2009-08-12 2012-02-08 Heterociclos microbicidas

Country Status (25)

Country Link
US (1) US8557821B2 (es)
EP (1) EP2464643A1 (es)
JP (1) JP2013501744A (es)
KR (1) KR20120089644A (es)
CN (1) CN102596943A (es)
AP (1) AP2012006153A0 (es)
AR (1) AR077834A1 (es)
AU (1) AU2010283832A1 (es)
BR (1) BR112012002369A2 (es)
CA (1) CA2769110A1 (es)
CL (1) CL2012000338A1 (es)
CO (1) CO6420414A2 (es)
CR (1) CR20120063A (es)
EA (1) EA021058B1 (es)
GE (1) GEP20146079B (es)
IL (1) IL217289A0 (es)
MA (1) MA33519B1 (es)
MX (1) MX2012001690A (es)
NI (1) NI201200024A (es)
NZ (1) NZ597562A (es)
TW (1) TW201114764A (es)
UA (1) UA104203C2 (es)
UY (1) UY32841A (es)
WO (1) WO2011018401A1 (es)
ZA (1) ZA201109515B (es)

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BR112012027762B1 (pt) 2010-04-28 2018-06-05 Bayer Intellectual Property Gmbh Derivados de cetoheteroarilpiperidina e - piperazina como fungicidas
JP2013528169A (ja) 2010-05-27 2013-07-08 バイエル・クロップサイエンス・アーゲー 殺菌剤としてのピリジニルカルボン酸誘導体
US20120122928A1 (en) 2010-08-11 2012-05-17 Bayer Cropscience Ag Heteroarylpiperidine and -Piperazine Derivatives as Fungicides
US8759527B2 (en) 2010-08-25 2014-06-24 Bayer Cropscience Ag Heteroarylpiperidine and -piperazine derivatives as fungicides
JP5916730B2 (ja) 2010-09-06 2016-05-11 グアンジョウ インスティテュート オブ バイオメディスン アンド ヘルス,チャイニーズ アカデミー オブ サイエンスィズ アミド化合物
CA2815716C (en) 2010-10-27 2019-06-11 Bayer Intellectual Property Gmbh Heteroaryl piperidine and heteroaryl piperazine derivatives as fungicides
US20130317064A1 (en) * 2011-02-10 2013-11-28 Syngenta Participations Ag Microbiocidal pyrazole derivatives
AP3662A (en) * 2011-06-30 2016-04-12 Syngenta Participations Ag Microbiocidal heterocycles
WO2013000941A1 (en) 2011-06-30 2013-01-03 Syngenta Participations Ag Microbiocidal heterocycles
CN103889982A (zh) * 2011-10-18 2014-06-25 先正达参股股份有限公司 杀微生物的吡唑衍生物
WO2013056911A1 (en) * 2011-10-18 2013-04-25 Syngenta Participations Ag Microbiocidal pyrazole derivatives
DK2921492T3 (en) 2011-12-27 2017-12-11 Bayer Ip Gmbh HETEROARYLPIPERIDINE AND ¿PIPERAZINE DERIVATIVES
CN104093715B (zh) 2012-02-02 2017-04-26 埃科特莱茵药品有限公司 4‑(苯并咪唑‑2‑基)‑噻唑化合物及相关氮杂衍生物
WO2014060176A1 (en) 2012-10-16 2014-04-24 Syngenta Participations Ag Microbiocidal pyrazole derivatives
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EP2801575A1 (en) 2013-05-07 2014-11-12 Bayer CropScience AG Heteroaryldihydropyridine derivatives as fungicides
EP3013821B1 (en) 2013-06-24 2018-03-14 Bayer CropScience Aktiengesellschaft Piperidinecarboxylic acid derivatives as fungicides
WO2015011099A1 (en) 2013-07-22 2015-01-29 Actelion Pharmaceuticals Ltd 1-(piperazin-1-yl)-2-([1,2,4]triazol-1-yl)-ethanone derivatives
TWI646095B (zh) 2013-08-28 2019-01-01 拜耳作物科學股份有限公司 作為殺真菌劑之雜芳基哌啶及-哌的丙二酸酯衍生物
AR099789A1 (es) 2014-03-24 2016-08-17 Actelion Pharmaceuticals Ltd Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina
UA117781C2 (uk) 2014-03-24 2018-09-25 Байєр Кропсайєнс Акцієнгезелльшафт Похідні фенілпіперидинкарбоксаміду як фунгіциди
WO2016024350A1 (ja) 2014-08-13 2016-02-18 株式会社エス・ディー・エス バイオテック 縮合11員環化合物及びそれらを含有する農園芸用殺菌剤
TR201900680T4 (tr) 2015-01-15 2019-02-21 Idorsia Pharmaceuticals Ltd CXCR3 Reseptör modülatörleri olarak hidroksialkil- piperazin türevleri.
AR103399A1 (es) 2015-01-15 2017-05-10 Actelion Pharmaceuticals Ltd Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3
JP6407457B2 (ja) 2016-02-08 2018-10-17 株式会社エス・ディー・エス バイオテック 1,2−ベンゼンジメタノール化合物の製造方法
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Also Published As

Publication number Publication date
NZ597562A (en) 2013-10-25
AR077834A1 (es) 2011-09-28
KR20120089644A (ko) 2012-08-13
EA021058B1 (ru) 2015-03-31
CL2012000338A1 (es) 2012-10-12
WO2011018401A1 (en) 2011-02-17
UY32841A (es) 2011-03-31
EA201200262A1 (ru) 2012-09-28
CN102596943A (zh) 2012-07-18
MX2012001690A (es) 2012-02-22
CA2769110A1 (en) 2011-02-17
BR112012002369A2 (pt) 2019-09-24
GEP20146079B (en) 2014-04-25
AU2010283832A1 (en) 2012-02-23
IL217289A0 (en) 2012-02-29
MA33519B1 (fr) 2012-08-01
TW201114764A (en) 2011-05-01
UA104203C2 (en) 2014-01-10
NI201200024A (es) 2012-08-15
EP2464643A1 (en) 2012-06-20
US8557821B2 (en) 2013-10-15
ZA201109515B (en) 2013-01-30
AP2012006153A0 (en) 2012-04-30
US20120142700A1 (en) 2012-06-07
CR20120063A (es) 2012-03-22
JP2013501744A (ja) 2013-01-17

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