CO6140003A2 - Derivados de 4-aza indol y su uso como fungicidas - Google Patents

Derivados de 4-aza indol y su uso como fungicidas

Info

Publication number
CO6140003A2
CO6140003A2 CO09119107A CO09119107A CO6140003A2 CO 6140003 A2 CO6140003 A2 CO 6140003A2 CO 09119107 A CO09119107 A CO 09119107A CO 09119107 A CO09119107 A CO 09119107A CO 6140003 A2 CO6140003 A2 CO 6140003A2
Authority
CO
Colombia
Prior art keywords
optionally substituted
cyano
hydrogen
nr10r11
alkynyl
Prior art date
Application number
CO09119107A
Other languages
English (en)
Inventor
Patrice Selles
Fredrik Cederbaum
Florence Marie-Emilie Bonnaterre
Mafalda Nina
William Guy Whittingham
Original Assignee
Syngenta Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Ltd filed Critical Syngenta Ltd
Publication of CO6140003A2 publication Critical patent/CO6140003A2/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647—Triazoles; Hydrogenated triazoles
    • A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Zoology (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

1.- Un método de prevención y/o control de la infección fúngica en las plantas y/o material de propagación de plantas que comprende aplicar a las plantas o material de propagación de plantas una cantidad efectiva como fungicida de un compuesto de la fórmula (I):donde: X1 es N o CH; X2 es N o CR5;R1 y R2 son independientemente, (i) hidrógeno, halógeno, hidroxilo, ciano o nitro, (ii) alquilo, alquenilo o alquinilo opcionalmente sustituido, (iii) arilo, heteroarilo, ciclilo o heterociclilo opcionalmente sustituido, o (iv) -C(O)R10, -C(O)NR10R11, -C(S)NR10R11, -C(NOR10)R11, -C(O)OR10, -OR10, -SR10, -S(O)R10, -S(O)NR10R11, -S(O)2R10, -NR10R11, -P(O)(OR10)(OR11) u -OP(O)(OR10)(OR11); R3 es: (i) hidrógeno, hidroxilo, ciano o nitro,(ii) alquilo, alquenilo, alenilo, alquinilo o haloalquilo opcionalmente sustituido, (iii) arilo, heteroarilo, ciclilo o heterociclilo o heteroaralquilo opcionalmente sustituido, o (iv) -C(O)R12, -C(O)OR12, -OR12, -OC(O)R12, -S(O)2R12 o -NR12R13; R4 es: (i) hidrógeno, halógeno, hidroxilo, ciano o nitro, (ii) alquenilo, alenilo, alquinilo o haloalquilo opcionalmente sustituido, (iii) arilo, heteroarilo, ciclilo o heterociclilo opcionalmente sustituido o (iv) -C(O)R14, -C(O)OR14, -C(NOR14)R15, -OR14, -SR14, -S(O)NR14R15, -S(O)2R14 o -NR14R15; R5 es: (i) hidrógeno, halógeno, hidroxilo, ciano o nitro,(ii) alquilo, alquenilo, o alquinilo opcionalmente sustituido, (iii) -C(O)R16, -C(O)OR16, -OR16, -SR16, -S(O)R16, -S(O)NR16R17, -S(O)2R16 o NR16R17;R6 es hidrógeno, halógeno, ciano, -C(O)OR18, -SR18, -NR18R19, -C(O)NR18R19, ...
CO09119107A 2007-04-26 2009-10-23 Derivados de 4-aza indol y su uso como fungicidas CO6140003A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0708141.7A GB0708141D0 (en) 2007-04-26 2007-04-26 Improvements in or relating to organic compounds

Publications (1)

Publication Number Publication Date
CO6140003A2 true CO6140003A2 (es) 2010-03-19

Family

ID=38170765

Family Applications (1)

Application Number Title Priority Date Filing Date
CO09119107A CO6140003A2 (es) 2007-04-26 2009-10-23 Derivados de 4-aza indol y su uso como fungicidas

Country Status (20)

Country Link
US (1) US8084395B2 (es)
EP (1) EP2136640A2 (es)
JP (1) JP2010525039A (es)
KR (1) KR20100015918A (es)
CN (1) CN101784191A (es)
AR (1) AR066310A1 (es)
AU (1) AU2008244055A1 (es)
BR (1) BRPI0810679A2 (es)
CA (1) CA2682773A1 (es)
CL (1) CL2008001214A1 (es)
CO (1) CO6140003A2 (es)
CR (1) CR11076A (es)
EC (1) ECSP099699A (es)
GB (1) GB0708141D0 (es)
IL (1) IL201195A0 (es)
MX (1) MX2009011337A (es)
RU (1) RU2009143567A (es)
TW (1) TW200847926A (es)
WO (1) WO2008132434A2 (es)
ZA (1) ZA200906887B (es)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200911807A (en) * 2007-08-29 2009-03-16 Schering Corp 2,3-substituted azaindole derivatives and methods of use thereof
WO2010046215A2 (en) * 2008-10-21 2010-04-29 Syngenta Participations Ag Diaza-indole derivatives and their use as fungicides
DE102008052943A1 (de) * 2008-10-23 2010-04-29 Merck Patent Gmbh Azaindolderivate
EP2198710A1 (de) 2008-12-19 2010-06-23 Bayer CropScience AG Verwendung von 5-Pyridin-4yl-(1,3)Thiazole zur Bekämpfung phytopathogener Pilze
EP2417133A1 (en) * 2009-04-06 2012-02-15 PTC Therapeutics, Inc. Compounds and methods for antiviral treatment
EP2245936A1 (en) * 2009-04-27 2010-11-03 Bayer CropScience AG Use of 4-aza indole derivatives for the reduction of mycotoxin contamination
AR081810A1 (es) 2010-04-07 2012-10-24 Bayer Cropscience Ag Piridinilpirazoles biciclicos
TW201242962A (en) * 2010-12-01 2012-11-01 Sumitomo Chemical Co Pyrimidine compound and use for pest control thereof
WO2012084678A1 (en) * 2010-12-23 2012-06-28 Syngenta Participations Ag Novel imidazoles useful as plant fungicides
EP2487159A1 (en) * 2011-02-11 2012-08-15 MSD Oss B.V. RorgammaT inhibitors
EP2696677B1 (en) 2011-04-13 2021-08-11 BioSafe Technologies, Inc. Insecticide, insect repellant and anti-irritation composition
CN103159663B (zh) * 2011-12-09 2014-09-17 中国科学院大连化学物理研究所 一种由联二烯衍生物制备吡咯衍生物的方法
WO2014026330A1 (en) 2012-08-15 2014-02-20 Merck Sharp & Dohme Corp. 3-AMINOCYCLOALKYL COMPOUNDS AS RORgammaT INHIBITORS AND USES THEREOF
WO2014026329A1 (en) 2012-08-15 2014-02-20 Merck Sharp & Dohme Corp. N-alkylated indole and indazole compounds as rorgammat inhibitors and uses thereof
WO2014026327A1 (en) 2012-08-15 2014-02-20 Merck Sharp & Dohme Corp. 4-heteroaryl substituted benzoic acid compounds as rorgammat inhibitors and uses thereof
JP2016135742A (ja) * 2013-03-29 2016-07-28 日本農薬株式会社 縮合複素環化合物又はその塩類及び該化合物を含有する農園芸用殺虫剤並びにその使用方法
AU2014296261B2 (en) * 2013-07-31 2018-11-15 Merck Patent Gmbh Pyridines, pyrimidines, and pyrazines, as BTK inhibitors and uses thereof
TW201630907A (zh) 2014-12-22 2016-09-01 必治妥美雅史谷比公司 ＴＧＦβＲ拮抗劑
JP2018510135A (ja) 2015-02-11 2018-04-12 メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． ＲＯＲγＴ阻害剤としての置換ピラゾール化合物及びその使用
AU2016344111A1 (en) 2015-10-27 2018-05-10 Merck Sharp & Dohme Corp. Substituted bicyclic pyrazole compounds as RORgammaT inhibitors and uses thereof
JP2018535958A (ja) 2015-10-27 2018-12-06 メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． ＲＯＲγＴ阻害薬としての置換インダゾール化合物及びその使用
EP3368535B1 (en) 2015-10-27 2020-12-02 Merck Sharp & Dohme Corp. Heteroaryl substituted benzoic acids as rorgammat inhibitors and uses thereof
JP6630828B2 (ja) * 2016-07-01 2020-01-15 日本農薬株式会社 Ｎ‐アルキルスルホニル縮合複素環化合物又はその塩類及び該化合物を含有する殺虫剤並びにその使用方法
CA3047896C (en) * 2016-12-27 2021-11-09 Nihon Nohyaku Co., Ltd. 4h-pyrrolopyridine compound or salt thereof, agricultural and horticultural insecticide comprising the compound or the salt, and method for using the insecticide
CN111164081B (zh) * 2017-09-26 2022-08-12 住友化学株式会社 杂环化合物和含有该杂环化合物的有害节肢动物防除剂
MX2020004049A (es) 2017-10-18 2020-07-20 Redag Crop Prot Ltd Compuestos bencimidazol como productos quimicos agricolas.
CN111819176B (zh) 2017-12-18 2023-12-15 百时美施贵宝公司 4-氮杂吲哚化合物
CN110156775A (zh) * 2018-02-12 2019-08-23 新发药业有限公司 一种吡昔替尼的简便制备方法
TWI748194B (zh) 2018-06-28 2021-12-01 德商菲尼克斯 Ｆｘｒ有限責任公司 含有雙環核心部分之新穎lxr調節劑
US20230391769A1 (en) 2020-07-29 2023-12-07 Bayer Aktiengesellschaft Substituted heterocyclic compounds and therapeutic uses thereof
US20230339939A1 (en) 2020-07-29 2023-10-26 Bayer Aktiengesellschaft Substituted 1h-pyrrolo[3,2-b]pyridine compounds and methods of use thereof
CN112661694B (zh) * 2020-12-11 2023-04-11 西安凯立新材料股份有限公司 一种4-(二甲氧基甲基)-哌啶的制备方法
WO2023147015A1 (en) * 2022-01-27 2023-08-03 The Broad Institute, Inc. Substituted heterocyclic csnk1 inhibitors
CN115124527B (zh) * 2022-05-31 2024-03-12 武汉智汇农耀科技有限公司 一种杂环酰胺-氮杂吲哚类化合物及其制备方法和应用、一种除草剂

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2219178C2 (ru) 1997-10-20 2003-12-20 Ф.Хоффманн-Ля Рош Аг Бициклические производные, фармацевтическая композиция на их основе и промежуточные соединения
JP2006502133A (ja) * 2002-08-10 2006-01-19 アステックス、セラピューティックス、リミテッド サイクリン依存キナーゼ（ｃｄｋ）インヒビターとしての３−（カルボニル）１ｈ−インダゾール化合物
EP1978805A1 (en) * 2006-01-30 2008-10-15 Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. Pesticidal composition comprising indole derivates

Also Published As

Publication number Publication date
ECSP099699A (es) 2009-11-30
RU2009143567A (ru) 2011-06-10
BRPI0810679A2 (pt) 2014-10-07
KR20100015918A (ko) 2010-02-12
EP2136640A2 (en) 2009-12-30
CN101784191A (zh) 2010-07-21
WO2008132434A3 (en) 2009-10-15
IL201195A0 (en) 2010-05-17
TW200847926A (en) 2008-12-16
AR066310A1 (es) 2009-08-12
WO2008132434A2 (en) 2008-11-06
AU2008244055A1 (en) 2008-11-06
CA2682773A1 (en) 2008-11-06
CR11076A (es) 2009-12-30
ZA200906887B (en) 2012-03-28
MX2009011337A (es) 2009-11-05
CL2008001214A1 (es) 2008-11-03
US20100184598A1 (en) 2010-07-22
JP2010525039A (ja) 2010-07-22
US8084395B2 (en) 2011-12-27
GB0708141D0 (en) 2007-06-06

Similar Documents

Publication Publication Date Title
CO6140003A2 (es) Derivados de 4-aza indol y su uso como fungicidas
PE20140185A1 (es) Derivados de heteroarilpiperidina y piperazina como fungicidas
CY1119569T1 (el) Μυκητοκτονες ενωσεις και μειγματα
EA200801627A1 (ru) Соединения пиперазина с гербицидным действием
CL2020002423A1 (es) Nuevos compuestos heterocíclicos
UY31148A1 (es) Compuestos de piperazina con accion herbicida (ii)
EA200801904A1 (ru) Способ индуцирования толерантности растений к вирусам
EA201070607A1 (ru) Гербицидные соединения
EA200870299A1 (ru) Гербицидные изоксазольные соединения
BRPI0910178A8 (pt) "composto de fórmula (i), composto de fórmula (vi), composição de fungicidas e método para o controle de fungo fitopatogênico de culturas"
CL2011001385A1 (es) Compuestos derivados de n-oxipiperidinas espiroheterciclicas; su proceso de preparacion; composicion pesticida que comprende a dichos compuestos; metodo para combatir y controlar plagas; y compuestos intermediarios.
BRPI0816132A8 (pt) métodos para controlar pestes invertebradas, e para proteger material de propagação de planta e/ou plantas que crescem a partir dos mesmos, material de propagação de planta, método para tratar ou proteger um animal contra infestação ou infecção por parasitas, composto de pirazol, e, composição agrícola
UY31750A (es) Compuestos y composiciones como inhibidores de quinasa
AR027117A1 (es) Trifluorometilpirrolcarboxamidas y trifluorometilpirroltioamidas como fungicidas
PE20141002A1 (es) Derivados de heteroarilpiperidina y -piperazina como fungicidas
ATE543515T1 (de) Konjugate von hydroxyalkyl-stärke und einer wirksubstanz, hergestellt durch chemische ligation über thiazolidin
CR7864A (es) Piridodiacinas como fungicidas de plantas
BRPI0519292A2 (pt) compostos orgÂnicos
GB0501964D0 (en) Chemical compounds
CR10637A (es) Fungicidas
CL2004000256A1 (es) 2-cloro-n-(4'-clorobifenil-2-il)nicotinamida monociclica; procedimiento de preparacion; util para tratar hongos nocivos, su biotipo o las plantas, superficies, materiales o espacios para mantenerlos libres de ellos.
AR066160A1 (es) DERIVADOS DE ISOTIAZOL Y PIRAZOL SUSTITUíDOS, UNA COMPOSICIoN PARA EL CONTROL DE LAS INFECCIONES FuNGICAS QUE LOS COMPRENDE Y UN METODO PARA TRATAR LAS INFECCIONES FuNGICAS.
UY29879A1 (es) Derivados de 6-heteroarilpiridoindolona, su preparación y su aplicación en terapéutica
UY38303A (es) Compuestos de isoxazolina para controlar plagas de invertebrados
AR076385A1 (es) Uso de derivados de 4-azaindol para reduccion de contaminacion por mico-toxina