CO5540383A2 - UNA COMBINACION FARMACEUTICA QUE COMPRENDE UNO CUALQUIERA DE ACIDO (S)-2-ETOXI-3-(4-(2-(4-METANOSULFONIL OXIFENIL) ETOXI)FENIL) PROPANOICO O ACIDO 3-(4-(2-(4-TERT-BUTOXI CARBONIL-AMINOFENIL)ETOXI)FENIL)-(s)-2-ETOXI PROPANOICO E INSULINA - Google Patents

UNA COMBINACION FARMACEUTICA QUE COMPRENDE UNO CUALQUIERA DE ACIDO (S)-2-ETOXI-3-(4-(2-(4-METANOSULFONIL OXIFENIL) ETOXI)FENIL) PROPANOICO O ACIDO 3-(4-(2-(4-TERT-BUTOXI CARBONIL-AMINOFENIL)ETOXI)FENIL)-(s)-2-ETOXI PROPANOICO E INSULINA

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Publication number
CO5540383A2
CO5540383A2 CO03112112A CO03112112A CO5540383A2 CO 5540383 A2 CO5540383 A2 CO 5540383A2 CO 03112112 A CO03112112 A CO 03112112A CO 03112112 A CO03112112 A CO 03112112A CO 5540383 A2 CO5540383 A2 CO 5540383A2
Authority
CO
Colombia
Prior art keywords
etoxi
phenyl
ethoxy
propanoic
acid
Prior art date
Application number
CO03112112A
Other languages
English (en)
Inventor
Peter Ohman
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of CO5540383A2 publication Critical patent/CO5540383A2/es

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/28Insulins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/325Carbamic acids; Thiocarbamic acids; Anhydrides or salts thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/06Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Zoology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Urology & Nephrology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

1.- Una combinación farmacéutica que comprende uno cualquiera de ácido (S)-2-etoxi-3-[4-(2-{4-metanosulfoniloxifenil)etoxi)fenil] propanoico o 3-{4-[2-(4-tert-butoxicarbonilaminofenil)etoxi]fenil)-(S)-2-etoxi propanoico, o una sal farmacéuticamente aceptable de los mismos y solvatos cualesquiera de uno cualquiera de los mismos e insulina.8.- Una combinación de productos que comprende:(1) una formulación farmacéutica que incluye uno cualquiera de ácido (S)-2-etoxi-3-[4-(2-{4-metano-sulfoniloxifenil}etoxi)fenil] propanoico o ácido 3-{4-[2-(4-tert-butoxicarbonil-aminofenil)-etoxi]fenil}-(S)-2-etoxi propanoico, o una sal farmacéuticamente aceptable de los mismos e insulina, en mezcla con un coadyuvante, diluyente o portador farmacéuticamente aceptables; y(2) un kit de partes que comprende componentes:(a) una formulación farmacéutica que incluye uno cualquiera de ácido (S)-2-etoxi-3-[4-(2-{4-metano-sulfoniloxifenil}etoxi)fenil] propanoico o ácido 3-{4-[2-(4-tert-butoxicarbonil-aminofenil)-etoxi]fenil}-(S)-2-etoxi propanoico, o una sal farmacéuticamente aceptable de los mismos en mezcla con un coadyuvante, diluyente o portador farmacéuticamente aceptables; y(b) una formulación farmacéutica que incluye insulina en mezcla con un coadyuvante, diluyente o portador farmacéuticamente aceptables, los cuales componentes (a) y (b) se proveen cada uno en una forma que es apropiada para administración en conjunción con el otro.
CO03112112A 2001-06-01 2003-12-23 UNA COMBINACION FARMACEUTICA QUE COMPRENDE UNO CUALQUIERA DE ACIDO (S)-2-ETOXI-3-(4-(2-(4-METANOSULFONIL OXIFENIL) ETOXI)FENIL) PROPANOICO O ACIDO 3-(4-(2-(4-TERT-BUTOXI CARBONIL-AMINOFENIL)ETOXI)FENIL)-(s)-2-ETOXI PROPANOICO E INSULINA CO5540383A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE0101981A SE0101981D0 (sv) 2001-06-01 2001-06-01 Pharmaceutical combination

Publications (1)

Publication Number Publication Date
CO5540383A2 true CO5540383A2 (es) 2005-07-29

Family

ID=20284363

Family Applications (1)

Application Number Title Priority Date Filing Date
CO03112112A CO5540383A2 (es) 2001-06-01 2003-12-23 UNA COMBINACION FARMACEUTICA QUE COMPRENDE UNO CUALQUIERA DE ACIDO (S)-2-ETOXI-3-(4-(2-(4-METANOSULFONIL OXIFENIL) ETOXI)FENIL) PROPANOICO O ACIDO 3-(4-(2-(4-TERT-BUTOXI CARBONIL-AMINOFENIL)ETOXI)FENIL)-(s)-2-ETOXI PROPANOICO E INSULINA

Country Status (22)

Country Link
US (1) US20040147600A1 (es)
EP (1) EP1401485A1 (es)
JP (1) JP2004532873A (es)
KR (1) KR20040072027A (es)
CN (1) CN1535155A (es)
BR (1) BR0210129A (es)
CA (1) CA2448637A1 (es)
CO (1) CO5540383A2 (es)
CZ (1) CZ20033233A3 (es)
EE (1) EE200300577A (es)
HU (1) HUP0400964A3 (es)
IL (1) IL159034A0 (es)
IS (1) IS7056A (es)
MX (1) MXPA03011012A (es)
NO (1) NO20035236D0 (es)
NZ (1) NZ529812A (es)
PL (1) PL367704A1 (es)
RU (1) RU2003136156A (es)
SE (1) SE0101981D0 (es)
SK (1) SK14712003A3 (es)
WO (1) WO2002096453A1 (es)
ZA (1) ZA200309261B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE60308390T2 (de) * 2003-11-28 2007-09-06 Merck Santé Behandlung von Hyperurikämie
AR052888A1 (es) * 2005-01-28 2007-04-11 Lilly Co Eli Uso del agonista alfa de ppar para preparar una formulacion farmaceutica, paquete y dosis unitaria de dicha formulacion
CN102036559A (zh) * 2008-05-19 2011-04-27 雀巢产品技术援助有限公司 降低动物脂质吸收的方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9801992D0 (sv) * 1998-06-04 1998-06-04 Astra Ab New 3-aryl-2-hydroxypropionic acid derivative I
SE9801990D0 (sv) * 1998-06-04 1998-06-04 Astra Ab New 3-aryl propionic acid derivatives and analogs
EP1145717B1 (en) * 2000-04-13 2004-05-12 Pfizer Products Inc. Synergistic effect of glyburide and milrinone

Also Published As

Publication number Publication date
NZ529812A (en) 2006-03-31
IL159034A0 (en) 2004-05-12
HUP0400964A2 (hu) 2004-08-30
PL367704A1 (en) 2005-03-07
EE200300577A (et) 2004-02-16
SE0101981D0 (sv) 2001-06-01
MXPA03011012A (es) 2004-02-27
EP1401485A1 (en) 2004-03-31
KR20040072027A (ko) 2004-08-16
BR0210129A (pt) 2004-06-08
NO20035236D0 (no) 2003-11-25
IS7056A (is) 2003-11-28
CZ20033233A3 (cs) 2004-12-15
HUP0400964A3 (en) 2007-11-28
US20040147600A1 (en) 2004-07-29
RU2003136156A (ru) 2005-05-20
ZA200309261B (en) 2005-02-28
CN1535155A (zh) 2004-10-06
CA2448637A1 (en) 2002-12-05
SK14712003A3 (sk) 2004-08-03
JP2004532873A (ja) 2004-10-28
WO2002096453A1 (en) 2002-12-05

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