CO5150174A1 - Bi-pirrolidinilvinil (carba) cefalosporinas - Google Patents

Bi-pirrolidinilvinil (carba) cefalosporinas

Info

Publication number
CO5150174A1
CO5150174A1 CO99075208A CO99075208A CO5150174A1 CO 5150174 A1 CO5150174 A1 CO 5150174A1 CO 99075208 A CO99075208 A CO 99075208A CO 99075208 A CO99075208 A CO 99075208A CO 5150174 A1 CO5150174 A1 CO 5150174A1
Authority
CO
Colombia
Prior art keywords
alkyl
hydrogen
halogen
jpeg
heterocyclyl
Prior art date
Application number
CO99075208A
Other languages
English (en)
Spanish (es)
Inventor
Ingrid Heinze-Kraus
Hans Richter
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CO5150174A1 publication Critical patent/CO5150174A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D463/00Heterocyclic compounds containing 1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D463/10Heterocyclic compounds containing 1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D463/14Heterocyclic compounds containing 1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hetero atoms directly attached in position 7
    • C07D463/16Nitrogen atoms
    • C07D463/18Nitrogen atoms further acylated by radicals derived from carboxylic acids or by nitrogen or sulfur analogues thereof
    • C07D463/20Nitrogen atoms further acylated by radicals derived from carboxylic acids or by nitrogen or sulfur analogues thereof with the acylating radicals further substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D463/22Nitrogen atoms further acylated by radicals derived from carboxylic acids or by nitrogen or sulfur analogues thereof with the acylating radicals further substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen further substituted by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CO99075208A 1998-12-03 1999-11-30 Bi-pirrolidinilvinil (carba) cefalosporinas CO5150174A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP98122965 1998-12-03
EP99119895 1999-10-07

Publications (1)

Publication Number Publication Date
CO5150174A1 true CO5150174A1 (es) 2002-04-29

Family

ID=26149851

Family Applications (1)

Application Number Title Priority Date Filing Date
CO99075208A CO5150174A1 (es) 1998-12-03 1999-11-30 Bi-pirrolidinilvinil (carba) cefalosporinas

Country Status (5)

Country Link
AR (1) AR023065A1 (fr)
AU (1) AU1654900A (fr)
CO (1) CO5150174A1 (fr)
PE (1) PE20001402A1 (fr)
WO (1) WO2000032605A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE60035925T2 (de) * 1999-07-05 2008-05-15 Basilea Pharmaceutica Ag Verfahren zur Herstellung von Cephalosporin-Derivaten
AU6267100A (en) * 1999-07-07 2001-01-30 F. Hoffmann-La Roche Ag Vinylpyrrolidinone derivatives with substituted thiazole ring

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5883247A (en) * 1996-06-10 1999-03-16 Hoffmann-La Roche Inc. Preparation of cephem and isooxacephem derivatives
EP0831093A1 (fr) * 1996-09-23 1998-03-25 F. Hoffmann-La Roche Ag Dérivés de 1-carba-(déthia)-céphalosporine
EP0838465A1 (fr) * 1996-10-22 1998-04-29 F. Hoffmann-La Roche Ag Dérivés de (lactamylvinyl)cephalosporin pyridinium substitués, leur préparation et leur utilisation comme antibiotiques
ATE354577T1 (de) * 1996-11-06 2007-03-15 Basilea Pharmaceutica Ag Vinylpyrrolidinon-cephalosporin-derivate
TW415949B (en) * 1996-12-19 2000-12-21 Hoffmann La Roche Vinyl pyrrolidine cephalosporin derivatives with basic substituents
US6150350A (en) * 1997-09-15 2000-11-21 Hoffman-La Roche Inc. Antimicrobial compositions

Also Published As

Publication number Publication date
WO2000032605A1 (fr) 2000-06-08
AR023065A1 (es) 2002-09-04
AU1654900A (en) 2000-06-19
PE20001402A1 (es) 2000-12-15

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