CO2022011593A2 - Método de preparación de derivados de amina heterocíclica - Google Patents

Método de preparación de derivados de amina heterocíclica

Info

Publication number
CO2022011593A2
CO2022011593A2 CONC2022/0011593A CO2022011593A CO2022011593A2 CO 2022011593 A2 CO2022011593 A2 CO 2022011593A2 CO 2022011593 A CO2022011593 A CO 2022011593A CO 2022011593 A2 CO2022011593 A2 CO 2022011593A2
Authority
CO
Colombia
Prior art keywords
heterocyclic amine
preparation
amine derivatives
amine derivative
heterocyclic
Prior art date
Application number
CONC2022/0011593A
Other languages
English (en)
Inventor
Wol-Young Kim
Qing Ri Li
Deok Ki Eom
Hyae Jung Hyun
Joon Seok Park
Original Assignee
Daewoong Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from KR1020210025655A external-priority patent/KR102531088B1/ko
Application filed by Daewoong Pharmaceutical Co Ltd filed Critical Daewoong Pharmaceutical Co Ltd
Publication of CO2022011593A2 publication Critical patent/CO2022011593A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Método para preparar un derivado de amina heterocíclica, y el método de preparación según la presente divulgación tiene la ventaja de que puede prepararse un derivado de amina heterocíclica que tiene un contenido de impurezas reducido con un alto rendimiento.
CONC2022/0011593A 2020-02-26 2022-08-17 Método de preparación de derivados de amina heterocíclica CO2022011593A2 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR20200023899 2020-02-26
KR1020210025655A KR102531088B1 (ko) 2020-02-26 2021-02-25 헤테로사이클릭아민 유도체의 제조 방법
PCT/KR2021/002440 WO2021172922A1 (ko) 2020-02-26 2021-02-26 헤테로사이클릭아민 유도체의 제조 방법

Publications (1)

Publication Number Publication Date
CO2022011593A2 true CO2022011593A2 (es) 2022-08-30

Family

ID=77490106

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2022/0011593A CO2022011593A2 (es) 2020-02-26 2022-08-17 Método de preparación de derivados de amina heterocíclica

Country Status (9)

Country Link
US (1) US20230094404A1 (es)
EP (1) EP4112617A4 (es)
JP (1) JP7447291B2 (es)
CN (1) CN115151537B (es)
BR (1) BR112022016729A2 (es)
CO (1) CO2022011593A2 (es)
JO (1) JOP20220199A1 (es)
MX (1) MX2022010391A (es)
WO (1) WO2021172922A1 (es)

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE318812T1 (de) 2000-12-21 2006-03-15 Bristol Myers Squibb Co Thiazolyl-inhibitoren von tyrosinkinasen der tec- familie
WO2005056785A2 (en) 2003-12-05 2005-06-23 Vertex Pharmaceuticals, Inc. Crystal structure of interleukin-2 tyrosine kinase (itk) and binding pockets thereof
WO2005066335A1 (en) 2003-12-30 2005-07-21 Boehringer Ingelheim Pharmaceuticals, Inc. Crystal structure of the interleukin-2-inducible cell kinase (itk) kinase domain
EP2532235A1 (en) 2006-09-22 2012-12-12 Pharmacyclics, Inc. Inhibitors of bruton's tyrosine kinase
WO2012035055A1 (en) * 2010-09-17 2012-03-22 Glaxo Group Limited Novel compounds
WO2014036016A1 (en) 2012-08-31 2014-03-06 Principia Biopharma Inc. Benzimidazole derivatives as itk inhibitors
WO2014055934A2 (en) 2012-10-04 2014-04-10 University Of Utah Research Foundation Substituted n-(3-(pyrimidin-4-yl)phenyl)acrylamide analogs as tyrosine receptor kinase btk inhibitors
WO2015061247A2 (en) 2013-10-21 2015-04-30 Merck Patent Gmbh Heteroaryl compounds as btk inhibitors and uses thereof
CN104628657A (zh) * 2013-11-06 2015-05-20 韩冰 一类治疗缺血性脑损伤的化合物及其用途
EP3715346B1 (en) * 2014-10-22 2024-01-03 Dana-Farber Cancer Institute, Inc. Thiazolyl-containing compounds for treating proliferative diseases
KR102613433B1 (ko) * 2017-10-11 2023-12-13 주식회사 대웅제약 신규한 페닐피리딘 유도체 및 이를 포함하는 약학 조성물
KR102328682B1 (ko) * 2018-08-27 2021-11-18 주식회사 대웅제약 신규한 헤테로사이클릭아민 유도체 및 이를 포함하는 약학 조성물

Also Published As

Publication number Publication date
JOP20220199A1 (ar) 2023-01-30
US20230094404A1 (en) 2023-03-30
JP2023515197A (ja) 2023-04-12
BR112022016729A2 (pt) 2022-10-11
EP4112617A4 (en) 2024-03-13
CN115151537B (zh) 2024-09-06
JP7447291B2 (ja) 2024-03-11
CN115151537A (zh) 2022-10-04
EP4112617A1 (en) 2023-01-04
WO2021172922A1 (ko) 2021-09-02
MX2022010391A (es) 2022-09-05

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