BR112015031820A2 - composto, composição farmacêutica, intermediário, processo para a preparação de um composto e métodos - Google Patents
composto, composição farmacêutica, intermediário, processo para a preparação de um composto e métodosInfo
- Publication number
- BR112015031820A2 BR112015031820A2 BR112015031820A BR112015031820A BR112015031820A2 BR 112015031820 A2 BR112015031820 A2 BR 112015031820A2 BR 112015031820 A BR112015031820 A BR 112015031820A BR 112015031820 A BR112015031820 A BR 112015031820A BR 112015031820 A2 BR112015031820 A2 BR 112015031820A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- methods
- pharmaceutical composition
- preparing
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4192—1,2,3-Triazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/20—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by nitrogen atoms not being part of nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
- C07C279/20—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylguanidines
- C07C279/24—Y being a hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Immunology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
composto, composição farmacêutica, intermediário, processo para a preparação de um composto e métodos the present invention relates to macrocyclic amidinourea derivatives, methods of preparation and uses thereof, pharmaceutical compositions in particular to be used as chitinase inhibitors.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201361836401P | 2013-06-18 | 2013-06-18 | |
PCT/EP2014/062896 WO2014202697A1 (en) | 2013-06-18 | 2014-06-18 | New macrocyclic amidinourea derivatives, methods of preparation and uses thereof as chitinase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
BR112015031820A2 true BR112015031820A2 (pt) | 2017-07-25 |
Family
ID=50979767
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR112015031820A BR112015031820A2 (pt) | 2013-06-18 | 2014-06-18 | composto, composição farmacêutica, intermediário, processo para a preparação de um composto e métodos |
Country Status (10)
Country | Link |
---|---|
US (1) | US10071975B2 (pt) |
EP (1) | EP3010896B1 (pt) |
JP (1) | JP6586416B2 (pt) |
CN (1) | CN105612147B (pt) |
AU (1) | AU2014283281C1 (pt) |
BR (1) | BR112015031820A2 (pt) |
CA (1) | CA2915767A1 (pt) |
MX (1) | MX363622B (pt) |
PT (1) | PT3010896T (pt) |
WO (1) | WO2014202697A1 (pt) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9135200B2 (en) | 2013-06-28 | 2015-09-15 | Futurewei Technologies, Inc. | System and method for extended peripheral component interconnect express fabrics |
EP3854789A1 (en) | 2020-01-22 | 2021-07-28 | Cygnet Biosciences B.V. | Macrocyclic compounds useful as chitinase inhibitors |
CN113773233B (zh) * | 2021-09-18 | 2022-05-06 | 中国农业大学 | 一种甲基胍基脲衍生物及其制备方法与应用 |
CN115754090B (zh) * | 2022-12-15 | 2023-08-29 | 华夏生生药业(北京)有限公司 | 一种lc-ms检测氟康唑相关杂质的方法 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1114155A (en) * | 1964-08-24 | 1968-05-15 | Evans Medical Ltd | Guanidino derivatives |
WO2009113033A2 (en) * | 2008-03-13 | 2009-09-17 | Università Degli Studi Di Siena | Linear and cyclic guanidine derivatives, method of preparation and uses thereof |
-
2014
- 2014-06-18 PT PT147316251T patent/PT3010896T/pt unknown
- 2014-06-18 CN CN201480045663.3A patent/CN105612147B/zh not_active Expired - Fee Related
- 2014-06-18 JP JP2016520477A patent/JP6586416B2/ja not_active Expired - Fee Related
- 2014-06-18 CA CA2915767A patent/CA2915767A1/en not_active Abandoned
- 2014-06-18 WO PCT/EP2014/062896 patent/WO2014202697A1/en active Application Filing
- 2014-06-18 EP EP14731625.1A patent/EP3010896B1/en not_active Not-in-force
- 2014-06-18 US US14/899,872 patent/US10071975B2/en not_active Expired - Fee Related
- 2014-06-18 BR BR112015031820A patent/BR112015031820A2/pt active Search and Examination
- 2014-06-18 AU AU2014283281A patent/AU2014283281C1/en not_active Ceased
- 2014-06-18 MX MX2015017446A patent/MX363622B/es unknown
Also Published As
Publication number | Publication date |
---|---|
CA2915767A1 (en) | 2014-12-24 |
EP3010896B1 (en) | 2017-11-01 |
PT3010896T (pt) | 2018-03-07 |
JP6586416B2 (ja) | 2019-10-02 |
AU2014283281A1 (en) | 2016-02-04 |
JP2016522236A (ja) | 2016-07-28 |
MX363622B (es) | 2019-03-28 |
AU2014283281B2 (en) | 2018-10-04 |
AU2014283281C1 (en) | 2019-01-24 |
CN105612147A (zh) | 2016-05-25 |
MX2015017446A (es) | 2016-08-12 |
US20160137617A1 (en) | 2016-05-19 |
EP3010896A1 (en) | 2016-04-27 |
US10071975B2 (en) | 2018-09-11 |
CN105612147B (zh) | 2018-06-05 |
WO2014202697A1 (en) | 2014-12-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B07D | Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette] | ||
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B07E | Notice of approval relating to section 229 industrial property law [chapter 7.5 patent gazette] |
Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI |
|
B06T | Formal requirements before examination [chapter 6.20 patent gazette] | ||
B06A | Notification to applicant to reply to the report for non-patentability or inadequacy of the application [chapter 6.1 patent gazette] | ||
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B11D | Dismissal acc. art. 38, par 2 of ipl - failure to pay fee after grant in time | ||
B350 | Update of information on the portal [chapter 15.35 patent gazette] |