CO2021012061A2 - Procedimiento para preparar un compuesto tricíclico fusionado, e intermedio del mismo - Google Patents

Procedimiento para preparar un compuesto tricíclico fusionado, e intermedio del mismo

Info

Publication number
CO2021012061A2
CO2021012061A2 CONC2021/0012061A CO2021012061A CO2021012061A2 CO 2021012061 A2 CO2021012061 A2 CO 2021012061A2 CO 2021012061 A CO2021012061 A CO 2021012061A CO 2021012061 A2 CO2021012061 A2 CO 2021012061A2
Authority
CO
Colombia
Prior art keywords
preparing
procedure
fused tricyclic
tricyclic compound
intermediates
Prior art date
Application number
CONC2021/0012061A
Other languages
English (en)
Inventor
Zhenhua Huang
Pengfei Guo
Cheng Li
Original Assignee
Kbp Biosciences Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kbp Biosciences Co Ltd filed Critical Kbp Biosciences Co Ltd
Publication of CO2021012061A2 publication Critical patent/CO2021012061A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/54Improvements relating to the production of bulk chemicals using solvents, e.g. supercritical solvents or ionic liquids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

La presente solicitud describe un procedimiento para preparar un compuesto tricíclico fusionado y un intermedio del mismo, se refiere específicamente a un procedimiento para preparar un compuesto de quinolina (3S,3aR)-3-ciclopentil-3,3a,4,5-tetrahidro-2H-pirazolo[3,4-f], intermedios en dicho procedimiento y métodos para preparar dichos intermedios.
CONC2021/0012061A 2019-03-01 2021-09-15 Procedimiento para preparar un compuesto tricíclico fusionado, e intermedio del mismo CO2021012061A2 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201910155700 2019-03-01
CN201910187667 2019-03-13
PCT/CN2020/077413 WO2020177658A1 (zh) 2019-03-01 2020-03-02 一种三并环化合物的制备方法及其中间体

Publications (1)

Publication Number Publication Date
CO2021012061A2 true CO2021012061A2 (es) 2021-09-30

Family

ID=72337678

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2021/0012061A CO2021012061A2 (es) 2019-03-01 2021-09-15 Procedimiento para preparar un compuesto tricíclico fusionado, e intermedio del mismo

Country Status (18)

Country Link
US (1) US20220144824A1 (es)
EP (1) EP3932920A4 (es)
JP (1) JP7291426B2 (es)
KR (1) KR20210136046A (es)
CN (1) CN113874371B (es)
AU (1) AU2020230627B2 (es)
BR (1) BR112021017276A2 (es)
CA (1) CA3132075A1 (es)
CL (1) CL2021002287A1 (es)
CO (1) CO2021012061A2 (es)
IL (1) IL286015A (es)
MX (1) MX2021010511A (es)
PE (1) PE20212179A1 (es)
SG (1) SG11202109564UA (es)
TW (1) TWI728727B (es)
UA (1) UA127368C2 (es)
WO (1) WO2020177658A1 (es)
ZA (1) ZA202106376B (es)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH08301850A (ja) * 1995-05-01 1996-11-19 Sagami Chem Res Center 光学活性5,9−メタノシクロオクタ[b]ピリジン誘導体の製造方法
JPH11322635A (ja) * 1998-05-07 1999-11-24 Kankyo Kagaku Center:Kk 光学活性化合物及び光学分割剤からなる分子化合物の生成方法
JP5212740B2 (ja) * 2009-10-29 2013-06-19 東レ・ファインケミカル株式会社 1,2−ジアミノシクロヘキサンの製造法
CN102372710A (zh) * 2010-08-18 2012-03-14 山东轩竹医药科技有限公司 作为盐皮质激素受体拮抗剂的并环类化合物
AU2013362400B2 (en) * 2012-12-22 2016-07-28 Novo Nordisk A/S Crystal form of compound used as mineralocorticoid receptor antagonist and preparation method therefor
CN103694253A (zh) * 2013-11-04 2014-04-02 湖南华腾制药有限公司 一种噻吩并三唑并[4,3-a][1,4]二氮杂卓类化合物的制备方法
WO2017063307A1 (zh) * 2015-10-13 2017-04-20 山东轩竹医药科技有限公司 1,4-二氢吡啶-3,5-二羧酸酯衍生物的制备方法及中间体
CN109983022B (zh) * 2016-09-27 2022-06-07 默沙东公司 作为mGluR2负性别构调节剂的色满、异色满和二氢异苯并呋喃衍生物、组合物及其用途

Also Published As

Publication number Publication date
JP7291426B2 (ja) 2023-06-15
WO2020177658A1 (zh) 2020-09-10
ZA202106376B (en) 2022-07-27
EP3932920A1 (en) 2022-01-05
AU2020230627B2 (en) 2023-01-19
SG11202109564UA (en) 2021-10-28
AU2020230627A1 (en) 2021-09-30
US20220144824A1 (en) 2022-05-12
TW202039492A (zh) 2020-11-01
CA3132075A1 (en) 2020-09-10
IL286015A (en) 2021-10-31
UA127368C2 (uk) 2023-07-26
CN113874371B (zh) 2024-04-16
MX2021010511A (es) 2021-11-17
CL2021002287A1 (es) 2022-04-22
KR20210136046A (ko) 2021-11-16
TWI728727B (zh) 2021-05-21
CN113874371A (zh) 2021-12-31
PE20212179A1 (es) 2021-11-09
JP2022522489A (ja) 2022-04-19
EP3932920A4 (en) 2022-12-14
BR112021017276A2 (pt) 2021-11-09

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