CN1823065A - 用于对映选择性制备亚砜衍生物的方法 - Google Patents

用于对映选择性制备亚砜衍生物的方法 Download PDF

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Publication number
CN1823065A
CN1823065A CN 200480008537 CN200480008537A CN1823065A CN 1823065 A CN1823065 A CN 1823065A CN 200480008537 CN200480008537 CN 200480008537 CN 200480008537 A CN200480008537 A CN 200480008537A CN 1823065 A CN1823065 A CN 1823065A
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CN
China
Prior art keywords
methyl
amino
methoxyl group
pyridyl
chemical formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN 200480008537
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English (en)
Chinese (zh)
Inventor
亚伯拉罕·科亨
苏济·沙尔比
弗朗索瓦·舒策
弗雷德里克·马蒂内
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sidem Pharma SA
Original Assignee
Sidem Pharma SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sidem Pharma SA filed Critical Sidem Pharma SA
Publication of CN1823065A publication Critical patent/CN1823065A/zh
Pending legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B45/00—Formation or introduction of functional groups containing sulfur
    • C07B45/04—Formation or introduction of functional groups containing sulfur of sulfonyl or sulfinyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
CN 200480008537 2003-03-28 2004-03-26 用于对映选择性制备亚砜衍生物的方法 Pending CN1823065A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR0303914A FR2852956B1 (fr) 2003-03-28 2003-03-28 Procede de preparation enantioselective de derives de sulfoxydes
FR0303914 2003-03-28
FR0314679 2003-12-15

Publications (1)

Publication Number Publication Date
CN1823065A true CN1823065A (zh) 2006-08-23

Family

ID=32947286

Family Applications (1)

Application Number Title Priority Date Filing Date
CN 200480008537 Pending CN1823065A (zh) 2003-03-28 2004-03-26 用于对映选择性制备亚砜衍生物的方法

Country Status (2)

Country Link
CN (1) CN1823065A (fr)
FR (1) FR2852956B1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102471290A (zh) * 2009-07-16 2012-05-23 拜尔农作物科学股份公司 手性3-三唑基亚砜衍生物的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE7804231L (sv) * 1978-04-14 1979-10-15 Haessle Ab Magsyrasekretionsmedel
DE3336751A1 (de) * 1983-10-08 1985-04-18 Bayer Ag, 5090 Leverkusen Verfahren zur herstellung von aminobenzol-alkylsulfonen bzw. -sulfoxiden
DK171989B1 (da) * 1987-08-04 1997-09-08 Takeda Chemical Industries Ltd Fremgangsmåde til fremstilling af 2-(2-pyridylmethylsulfinyl)-benzimidazoler
SE504459C2 (sv) * 1994-07-15 1997-02-17 Astra Ab Förfarande för framställning av substituerade sulfoxider
AU2003262375A1 (en) * 2002-04-22 2003-11-03 Sun Pharmaceutical Industries Limited Optically active substituted pyridinylmethyl-sulphinyl-benzimidazole and salts

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102471290A (zh) * 2009-07-16 2012-05-23 拜尔农作物科学股份公司 手性3-三唑基亚砜衍生物的制备方法
CN102471290B (zh) * 2009-07-16 2016-02-03 拜耳知识产权有限责任公司 手性3-三唑基亚砜衍生物的制备方法

Also Published As

Publication number Publication date
FR2852956A1 (fr) 2004-10-01
FR2852956B1 (fr) 2006-08-04

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Open date: 20060823