CN1410059A - 治疗方法和包含促生长激素分泌剂的药盒 - Google Patents
治疗方法和包含促生长激素分泌剂的药盒 Download PDFInfo
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- CN1410059A CN1410059A CN02143349A CN02143349A CN1410059A CN 1410059 A CN1410059 A CN 1410059A CN 02143349 A CN02143349 A CN 02143349A CN 02143349 A CN02143349 A CN 02143349A CN 1410059 A CN1410059 A CN 1410059A
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- oxo
- alkyl
- pyridine
- ethyl
- growth hormone
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- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
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Cited By (1)
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| CN102333545A (zh) * | 2009-02-27 | 2012-01-25 | 赫尔辛医疗（美国）有限公司 | 基于生长激素释放肽模拟物的增强的偏头痛治疗 |
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| EP1529533A1 (en) * | 2003-11-06 | 2005-05-11 | Sahltech I Göteborg AB | Use of GH secretagogues in hypoxic-ischemic brain injury |
| EP1986508B1 (en) * | 2006-01-26 | 2014-05-21 | Hill's Pet Nutrition, Inc. | Methods and compositions for treating feline hyperthyroidism |
| CA2677045C (en) | 2007-01-31 | 2016-10-18 | Dana-Farber Cancer Institute, Inc. | Stabilized p53 peptides and uses thereof |
| WO2008100448A2 (en) * | 2007-02-13 | 2008-08-21 | Helsinn Therapeutics (U.S.), Inc. | Method of treating cell proliferative disorders using growth hormone secretagogues |
| KR20160061439A (ko) | 2007-03-28 | 2016-05-31 | 프레지던트 앤드 펠로우즈 오브 하바드 칼리지 | 스티칭된 폴리펩티드 |
| CA2691010A1 (en) * | 2007-06-28 | 2008-12-31 | Merck Frosst Canada Ltd. | Substituted fused pyrimidines as antagonists of gpr105 activity |
| US8759289B2 (en) * | 2010-02-03 | 2014-06-24 | Orbis Health Solutions Llc | Method for sensitizing cancer stem cells to cancer therapy |
| MX355543B (es) | 2010-08-13 | 2018-04-20 | Aileron Therapeutics Inc Star | Macrociclos peptidomiméticos. |
| RU2639523C2 (ru) | 2011-10-18 | 2017-12-21 | Эйлерон Терапьютикс, Инк. | Пептидомиметические макроциклы и их применение |
| JP6450191B2 (ja) | 2012-02-15 | 2019-01-09 | エイルロン セラピューティクス，インコーポレイテッド | ペプチドミメティック大環状化合物 |
| HK1205454A1 (en) | 2012-02-15 | 2015-12-18 | Aileron Therapeutics, Inc. | Triazole-crosslinked and thioether-crosslinked peptidomimetic macrocycles |
| US9604919B2 (en) | 2012-11-01 | 2017-03-28 | Aileron Therapeutics, Inc. | Disubstituted amino acids and methods of preparation and use thereof |
| US9119832B2 (en) | 2014-02-05 | 2015-09-01 | The Regents Of The University Of California | Methods of treating mild brain injury |
| SG11201702223UA (en) | 2014-09-24 | 2017-04-27 | Aileron Therapeutics Inc | Peptidomimetic macrocycles and uses thereof |
| EP3294318A4 (en) | 2015-03-20 | 2019-04-03 | Aileron Therapeutics, Inc. | PEPTIDOMIMETIC MACROCYCLES AND USES THEREOF |
| US20220152032A1 (en) * | 2020-11-13 | 2022-05-19 | Pharma America Holding Inc. | Sexual therapy formulation and method of treatment |
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| US4411890A (en) * | 1981-04-14 | 1983-10-25 | Beckman Instruments, Inc. | Synthetic peptides having pituitary growth hormone releasing activity |
| US4060615A (en) * | 1976-02-18 | 1977-11-29 | Mead Johnson & Company | 2-Piperazinyl-6,7-dimethoxyquinazolines |
| DE3046719C2 (de) * | 1980-12-11 | 1983-02-17 | Klinge Pharma GmbH, 8000 München | 1,1,2-Triphenyl-but-1-en-Derivate, Verfahren zu ihrer Herstellung und Arzneimittel |
| US4418068A (en) * | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
| JPS6094992A (ja) * | 1983-10-28 | 1985-05-28 | Sankyo Co Ltd | グリゼオ−ル酸誘導体 |
| US4783532A (en) * | 1983-10-28 | 1988-11-08 | Sankyo Company Limited | Process for preparing griseolic acid derivatives |
| US4666908A (en) * | 1985-04-05 | 1987-05-19 | Warner-Lambert Company | 5-Substituted pyrazolo[4,3-d]pyrimidine-7-ones and methods of use |
| FI94133C (fi) * | 1985-04-19 | 1995-07-25 | Sankyo Co | Menetelmä lääkeaineina käyttökelpoisten griseoliinihapon johdannaisten valmistamiseksi |
| CA1303037C (en) * | 1987-02-02 | 1992-06-09 | Smith Kline & French Laboratories Limited | Purinone derivatives as bronchodilators vasodilators and anti-allergic agents |
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| EP0347146B1 (en) * | 1988-06-16 | 1993-09-01 | Smith Kline & French Laboratories Limited | Fused pyrimidine derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them |
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-
2002
- 2002-09-13 EP EP02256371A patent/EP1312363A1/en not_active Withdrawn
- 2002-09-19 IL IL15183502A patent/IL151835A0/xx unknown
- 2002-09-25 ZA ZA200207677A patent/ZA200207677B/xx unknown
- 2002-09-25 BR BR0203886-2A patent/BR0203886A/pt not_active IP Right Cessation
- 2002-09-26 CN CN02143349A patent/CN1410059A/zh active Pending
- 2002-09-26 CA CA002405342A patent/CA2405342A1/en not_active Abandoned
- 2002-09-27 US US10/256,567 patent/US20030105114A1/en not_active Abandoned
- 2002-09-27 PL PL02356364A patent/PL356364A1/xx not_active Application Discontinuation
- 2002-09-27 HU HU0203243A patent/HUP0203243A2/hu unknown
- 2002-09-27 JP JP2002282958A patent/JP2003160508A/ja not_active Withdrawn
- 2002-09-28 KR KR1020020059118A patent/KR20030027865A/ko not_active Ceased
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102333545A (zh) * | 2009-02-27 | 2012-01-25 | 赫尔辛医疗（美国）有限公司 | 基于生长激素释放肽模拟物的增强的偏头痛治疗 |
| CN102333545B (zh) * | 2009-02-27 | 2014-03-19 | 赫尔辛医疗（美国）有限公司 | 基于生长激素释放肽模拟物的增强的偏头痛治疗 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP1312363A1 (en) | 2003-05-21 |
| CA2405342A1 (en) | 2003-03-28 |
| PL356364A1 (en) | 2003-04-07 |
| US20030105114A1 (en) | 2003-06-05 |
| KR20030027865A (ko) | 2003-04-07 |
| IL151835A0 (en) | 2003-04-10 |
| HUP0203243A2 (en) | 2008-03-28 |
| ZA200207677B (en) | 2004-03-25 |
| BR0203886A (pt) | 2003-09-16 |
| JP2003160508A (ja) | 2003-06-03 |
| HU0203243D0 (cg-RX-API-DMAC7.html) | 2002-11-28 |
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