CN1252061A - 4-氨基烷氧基-1,3-二氢苯咪唑-2-硫酮衍生物、它们的制备方法以及它们作为多巴胺自身受体(d2)激动剂的用途 - Google Patents
4-氨基烷氧基-1,3-二氢苯咪唑-2-硫酮衍生物、它们的制备方法以及它们作为多巴胺自身受体(d2)激动剂的用途 Download PDFInfo
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- CN1252061A CN1252061A CN98804120A CN98804120A CN1252061A CN 1252061 A CN1252061 A CN 1252061A CN 98804120 A CN98804120 A CN 98804120A CN 98804120 A CN98804120 A CN 98804120A CN 1252061 A CN1252061 A CN 1252061A
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- dihydro
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- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/28—Sulfur atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- H—ELECTRICITY
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- H04N—PICTORIAL COMMUNICATION, e.g. TELEVISION
- H04N19/00—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals
- H04N19/10—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding
- H04N19/102—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the element, parameter or selection affected or controlled by the adaptive coding
- H04N19/124—Quantisation
- H04N19/126—Details of normalisation or weighting functions, e.g. normalisation matrices or variable uniform quantisers
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- H04N19/134—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the element, parameter or criterion affecting or controlling the adaptive coding
- H04N19/154—Measured or subjectively estimated visual quality after decoding, e.g. measurement of distortion
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- H04N19/17—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the coding unit, i.e. the structural portion or semantic portion of the video signal being the object or the subject of the adaptive coding the unit being an image region, e.g. an object
- H04N19/172—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the coding unit, i.e. the structural portion or semantic portion of the video signal being the object or the subject of the adaptive coding the unit being an image region, e.g. an object the region being a picture, frame or field
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- H04N19/169—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the coding unit, i.e. the structural portion or semantic portion of the video signal being the object or the subject of the adaptive coding
- H04N19/182—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the coding unit, i.e. the structural portion or semantic portion of the video signal being the object or the subject of the adaptive coding the unit being a pixel
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- H04N19/00—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals
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- H04N19/61—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using transform coding in combination with predictive coding
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- H04N19/85—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using pre-processing or post-processing specially adapted for video compression
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- H04N19/00—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals
- H04N19/10—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding
- H04N19/102—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the element, parameter or selection affected or controlled by the adaptive coding
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- H04N19/00—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals
- H04N19/10—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding
- H04N19/102—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the element, parameter or selection affected or controlled by the adaptive coding
- H04N19/132—Sampling, masking or truncation of coding units, e.g. adaptive resampling, frame skipping, frame interpolation or high-frequency transform coefficient masking
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- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04N—PICTORIAL COMMUNICATION, e.g. TELEVISION
- H04N19/00—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals
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- H04N19/134—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the element, parameter or criterion affecting or controlling the adaptive coding
- H04N19/146—Data rate or code amount at the encoder output
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- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04N—PICTORIAL COMMUNICATION, e.g. TELEVISION
- H04N19/00—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals
- H04N19/10—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding
- H04N19/134—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the element, parameter or criterion affecting or controlling the adaptive coding
- H04N19/146—Data rate or code amount at the encoder output
- H04N19/149—Data rate or code amount at the encoder output by estimating the code amount by means of a model, e.g. mathematical model or statistical model
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04N—PICTORIAL COMMUNICATION, e.g. TELEVISION
- H04N19/00—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals
- H04N19/10—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding
- H04N19/134—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the element, parameter or criterion affecting or controlling the adaptive coding
- H04N19/146—Data rate or code amount at the encoder output
- H04N19/15—Data rate or code amount at the encoder output by monitoring actual compressed data size at the memory before deciding storage at the transmission buffer
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- H04N19/00—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals
- H04N19/10—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding
- H04N19/134—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using adaptive coding characterised by the element, parameter or criterion affecting or controlling the adaptive coding
- H04N19/146—Data rate or code amount at the encoder output
- H04N19/152—Data rate or code amount at the encoder output by measuring the fullness of the transmission buffer
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- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04N—PICTORIAL COMMUNICATION, e.g. TELEVISION
- H04N19/00—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals
- H04N19/60—Methods or arrangements for coding, decoding, compressing or decompressing digital video signals using transform coding
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Signal Processing (AREA)
- Multimedia (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Addiction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US80265197A | 1997-02-18 | 1997-02-18 | |
US08/802,651 | 1997-02-18 |
Publications (1)
Publication Number | Publication Date |
---|---|
CN1252061A true CN1252061A (zh) | 2000-05-03 |
Family
ID=25184324
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN98804120A Pending CN1252061A (zh) | 1997-02-18 | 1998-01-13 | 4-氨基烷氧基-1,3-二氢苯咪唑-2-硫酮衍生物、它们的制备方法以及它们作为多巴胺自身受体(d2)激动剂的用途 |
Country Status (12)
Country | Link |
---|---|
EP (1) | EP0964854A1 (fr) |
JP (1) | JP2001511803A (fr) |
KR (1) | KR20000071124A (fr) |
CN (1) | CN1252061A (fr) |
AR (1) | AR011139A1 (fr) |
AU (1) | AU5915298A (fr) |
BR (1) | BR9807840A (fr) |
CA (1) | CA2278718A1 (fr) |
HU (1) | HUP0001942A2 (fr) |
IL (1) | IL131157A0 (fr) |
WO (1) | WO1998035947A1 (fr) |
ZA (1) | ZA981308B (fr) |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1986001204A1 (fr) * | 1984-08-15 | 1986-02-27 | Schering Aktiengesellschaft | Nouveaux derives de dopamine, procede pour leur production et leur utilisation comme produits medicinaux |
EP1123933A1 (fr) * | 1994-10-14 | 2001-08-16 | MERCK PATENT GmbH | 2-[5-(4-fluorophényl)-3-pyridylméthylaminométhyl]chromane agissant sur le système nerveux central |
ZA9610745B (en) * | 1995-12-22 | 1997-06-24 | Warner Lambert Co | 4-Subsituted piperidine analogs and their use as subtype selective nmda receptor antagonists |
-
1998
- 1998-01-13 IL IL13115798A patent/IL131157A0/xx unknown
- 1998-01-13 HU HU0001942A patent/HUP0001942A2/hu unknown
- 1998-01-13 JP JP53572698A patent/JP2001511803A/ja active Pending
- 1998-01-13 ZA ZA981308A patent/ZA981308B/xx unknown
- 1998-01-13 AU AU59152/98A patent/AU5915298A/en not_active Abandoned
- 1998-01-13 KR KR1019997007412A patent/KR20000071124A/ko not_active Application Discontinuation
- 1998-01-13 WO PCT/US1998/000612 patent/WO1998035947A1/fr not_active Application Discontinuation
- 1998-01-13 CN CN98804120A patent/CN1252061A/zh active Pending
- 1998-01-13 EP EP98902512A patent/EP0964854A1/fr not_active Withdrawn
- 1998-01-13 CA CA002278718A patent/CA2278718A1/fr not_active Abandoned
- 1998-01-13 BR BR9807840-2A patent/BR9807840A/pt not_active Application Discontinuation
- 1998-02-11 AR ARP980100621A patent/AR011139A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
JP2001511803A (ja) | 2001-08-14 |
KR20000071124A (ko) | 2000-11-25 |
ZA981308B (en) | 1999-08-17 |
AR011139A1 (es) | 2000-08-02 |
HUP0001942A2 (hu) | 2000-11-28 |
WO1998035947A1 (fr) | 1998-08-20 |
CA2278718A1 (fr) | 1998-08-20 |
BR9807840A (pt) | 2000-09-19 |
AU5915298A (en) | 1998-09-08 |
EP0964854A1 (fr) | 1999-12-22 |
IL131157A0 (en) | 2001-01-28 |
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CN1252061A (zh) | 4-氨基烷氧基-1,3-二氢苯咪唑-2-硫酮衍生物、它们的制备方法以及它们作为多巴胺自身受体(d2)激动剂的用途 |
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C02 | Deemed withdrawal of patent application after publication (patent law 2001) | ||
WD01 | Invention patent application deemed withdrawn after publication |