CN1161345C - 作为cck-a受体激动剂的1,5-苯并二氮杂�衍生物 - Google Patents
作为cck-a受体激动剂的1,5-苯并二氮杂�衍生物 Download PDFInfo
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- CN1161345C CN1161345C CNB008099324A CN00809932A CN1161345C CN 1161345 C CN1161345 C CN 1161345C CN B008099324 A CNB008099324 A CN B008099324A CN 00809932 A CN00809932 A CN 00809932A CN 1161345 C CN1161345 C CN 1161345C
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Classifications
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- C07—ORGANIC CHEMISTRY
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- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/12—1,5-Benzodiazepines; Hydrogenated 1,5-benzodiazepines
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
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- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Endocrinology (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Gastroenterology & Hepatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9910366.5A GB9910366D0 (en) | 1999-05-06 | 1999-05-06 | 1,5-Benzodiazepine Derivatives |
| GB9910366.5 | 1999-05-06 | ||
| GB0008179.4 | 2000-04-05 | ||
| GBGB0008179.4A GB0008179D0 (en) | 2000-04-05 | 2000-04-05 | Chemical process |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN1362949A CN1362949A (zh) | 2002-08-07 |
| CN1161345C true CN1161345C (zh) | 2004-08-11 |
Family
ID=26244033
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB008099324A Expired - Fee Related CN1161345C (zh) | 1999-05-06 | 2000-05-04 | 作为cck-a受体激动剂的1,5-苯并二氮杂�衍生物 |
Country Status (21)
| Country | Link |
|---|---|
| EP (1) | EP1212305A2 (pt) |
| JP (1) | JP2002544200A (pt) |
| KR (1) | KR20020012567A (pt) |
| CN (1) | CN1161345C (pt) |
| AR (1) | AR022044A1 (pt) |
| AU (1) | AU4754800A (pt) |
| BR (1) | BR0010338A (pt) |
| CA (1) | CA2370801A1 (pt) |
| CO (1) | CO5170461A1 (pt) |
| CZ (1) | CZ20013988A3 (pt) |
| HK (1) | HK1046138A1 (pt) |
| HU (1) | HUP0201181A3 (pt) |
| IL (1) | IL146124A0 (pt) |
| MX (1) | MXPA01011267A (pt) |
| MY (1) | MY138319A (pt) |
| NO (1) | NO20015397L (pt) |
| NZ (1) | NZ515048A (pt) |
| PE (1) | PE20010110A1 (pt) |
| PL (1) | PL351546A1 (pt) |
| TR (1) | TR200103169T2 (pt) |
| WO (1) | WO2000068209A2 (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005035793A2 (en) * | 2003-10-09 | 2005-04-21 | Decode Genetics Ehf. | Cckar markers and haplotypes associated with extreme weight conditions |
| EP1753766A1 (en) | 2004-05-25 | 2007-02-21 | Pfizer Products Inc. | Tetraazabenzo(e)azulene derivatives and analogs thereof |
| AU2020363377A1 (en) | 2019-10-07 | 2022-04-21 | Kallyope, Inc. | GPR119 agonists |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9307833D0 (en) * | 1993-04-15 | 1993-06-02 | Glaxo Inc | Modulators of cholecystokinin and gastrin |
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2000
- 2000-05-03 AR ARP000102119A patent/AR022044A1/es unknown
- 2000-05-04 CZ CZ20013988A patent/CZ20013988A3/cs unknown
- 2000-05-04 AU AU47548/00A patent/AU4754800A/en not_active Abandoned
- 2000-05-04 PL PL00351546A patent/PL351546A1/xx not_active Application Discontinuation
- 2000-05-04 MX MXPA01011267A patent/MXPA01011267A/es not_active Application Discontinuation
- 2000-05-04 BR BR0010338-1A patent/BR0010338A/pt not_active IP Right Cessation
- 2000-05-04 PE PE2000000415A patent/PE20010110A1/es not_active Application Discontinuation
- 2000-05-04 MY MYPI20001917A patent/MY138319A/en unknown
- 2000-05-04 IL IL14612400A patent/IL146124A0/xx unknown
- 2000-05-04 CO CO00031982A patent/CO5170461A1/es not_active Application Discontinuation
- 2000-05-04 HU HU0201181A patent/HUP0201181A3/hu unknown
- 2000-05-04 JP JP2000617189A patent/JP2002544200A/ja active Pending
- 2000-05-04 TR TR2001/03169T patent/TR200103169T2/xx unknown
- 2000-05-04 NZ NZ515048A patent/NZ515048A/xx unknown
- 2000-05-04 EP EP00929488A patent/EP1212305A2/en not_active Withdrawn
- 2000-05-04 CA CA002370801A patent/CA2370801A1/en not_active Abandoned
- 2000-05-04 CN CNB008099324A patent/CN1161345C/zh not_active Expired - Fee Related
- 2000-05-04 KR KR1020017014075A patent/KR20020012567A/ko not_active Application Discontinuation
- 2000-05-04 WO PCT/EP2000/003982 patent/WO2000068209A2/en not_active Application Discontinuation
-
2001
- 2001-11-05 NO NO20015397A patent/NO20015397L/no not_active Application Discontinuation
-
2002
- 2002-10-23 HK HK02107684.4A patent/HK1046138A1/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AR022044A1 (es) | 2002-09-04 |
| MY138319A (en) | 2009-05-29 |
| IL146124A0 (en) | 2002-07-25 |
| WO2000068209A3 (en) | 2001-03-01 |
| EP1212305A2 (en) | 2002-06-12 |
| NZ515048A (en) | 2004-01-30 |
| NO20015397D0 (no) | 2001-11-05 |
| CA2370801A1 (en) | 2000-11-16 |
| PE20010110A1 (es) | 2001-03-05 |
| MXPA01011267A (es) | 2002-05-06 |
| NO20015397L (no) | 2001-11-05 |
| TR200103169T2 (tr) | 2002-04-22 |
| PL351546A1 (en) | 2003-05-05 |
| HK1046138A1 (zh) | 2002-12-27 |
| KR20020012567A (ko) | 2002-02-16 |
| HUP0201181A2 (hu) | 2002-12-28 |
| WO2000068209A2 (en) | 2000-11-16 |
| HUP0201181A3 (en) | 2003-10-28 |
| CO5170461A1 (es) | 2002-06-27 |
| JP2002544200A (ja) | 2002-12-24 |
| CN1362949A (zh) | 2002-08-07 |
| AU4754800A (en) | 2000-11-21 |
| BR0010338A (pt) | 2002-02-13 |
| CZ20013988A3 (cs) | 2002-02-13 |
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