CN116120314A - 用于调节毛发生长的组合物和方法 - Google Patents

用于调节毛发生长的组合物和方法 Download PDF

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CN116120314A
CN116120314A CN202310059843.8A CN202310059843A CN116120314A CN 116120314 A CN116120314 A CN 116120314A CN 202310059843 A CN202310059843 A CN 202310059843A CN 116120314 A CN116120314 A CN 116120314A
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nmr
acid
dmso
jxl
compound
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Chinese (zh)
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W·E·劳瑞
M·E·荣格
H·克里斯托夫
X·刘
A·弗洛雷斯
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University of California San Diego UCSD
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K8/492—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with one nitrogen as the only hetero atom having five membered rings, e.g. pyrrolidone carboxylic acid having condensed rings, e.g. indol
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    • C07C255/41—Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by carboxyl groups, other than cyano groups
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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  • Chemical Kinetics & Catalysis (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
CN202310059843.8A 2017-06-30 2018-06-29 用于调节毛发生长的组合物和方法 Pending CN116120314A (zh)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US201762527775P 2017-06-30 2017-06-30
US62/527,775 2017-06-30
US201862654095P 2018-04-06 2018-04-06
US62/654,095 2018-04-06
CN201880043696.2A CN110944634A (zh) 2017-06-30 2018-06-29 用于调节毛发生长的组合物和方法
PCT/US2018/040385 WO2019006359A1 (en) 2017-06-30 2018-06-29 COMPOSITIONS AND METHODS FOR MODULATION OF HAIR GROWTH

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MX389692B (es) 2017-02-24 2025-03-20 Univ California Composiciones y métodos para promover el crecimiento del cabello con inhibidores de mpc.
CN116120314A (zh) 2017-06-30 2023-05-16 加利福尼亚大学董事会 用于调节毛发生长的组合物和方法
US20210161968A1 (en) * 2018-04-13 2021-06-03 North Carolina State University Use of microneedle patch to promote hair growth
CN113631555A (zh) * 2019-01-02 2021-11-09 加利福尼亚大学董事会 用于调节毛发生长的组合物和方法
CA3164224A1 (en) * 2019-12-20 2021-06-24 The Regent Of The University Of California Synthesis of compounds to promote hair growth
FR3105222B1 (fr) * 2019-12-20 2022-06-03 Nunii Laboratoire Inhibiteur du transporteur MCT7/SLC16A6 pour son utilisation pour la régulation de la pigmentation cutanée et une composition comprenant ledit inhibiteur
WO2021253013A2 (en) * 2020-06-12 2021-12-16 Rekindle Therapeutics Inc. Modulators of e3 ligases
US20240327400A1 (en) * 2020-06-30 2024-10-03 The Regents Of The University Of California Compositions and methods for modulating hair growth
WO2022006040A1 (en) * 2020-06-30 2022-01-06 The Regents Of The University Of California Compositions and methods for modulating hair growth
AU2022424022A1 (en) * 2021-12-29 2024-07-18 Pelage Pharmaceuticals, Inc. Compounds for treatment of hair loss
WO2023129854A1 (en) 2021-12-29 2023-07-06 Pelage Pharmaceuticals, Inc. Compounds for treatment of hair loss
WO2023191515A1 (ko) * 2022-03-29 2023-10-05 연세대학교 산학협력단 인디루빈 유도체 및 대사활성화제를 포함하는 탈모 방지 또는 발모 촉진용 조성물
WO2024145369A1 (en) * 2022-12-27 2024-07-04 Pelage Pharmaceuticals, Inc. Compounds for treatment of hair loss
CN116251086A (zh) * 2023-02-15 2023-06-13 江西中医药大学 乳酸及其衍生物在促毛发生长及缓解脱发中的应用
CN121005682A (zh) * 2024-05-24 2025-11-25 上海医药工业研究院有限公司 一种2-苯基-吡咯类化合物、其制备方法及其应用

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