CN113149983B - 酪氨酸激酶抑制剂 - Google Patents
酪氨酸激酶抑制剂 Download PDFInfo
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- CN113149983B CN113149983B CN202011284728.3A CN202011284728A CN113149983B CN 113149983 B CN113149983 B CN 113149983B CN 202011284728 A CN202011284728 A CN 202011284728A CN 113149983 B CN113149983 B CN 113149983B
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- amino
- oxo
- imidazo
- phenoxyphenyl
- dihydro
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Landscapes
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| CN201680000891.8A CN106459049B (zh) | 2015-06-03 | 2016-06-02 | 酪氨酸激酶抑制剂 |
| CN202011284728.3A CN113149983B (zh) | 2015-06-03 | 2016-06-02 | 酪氨酸激酶抑制剂 |
| PCT/US2016/035588 WO2016196840A1 (en) | 2015-06-03 | 2016-06-02 | Tyrosine kinase inhibitors |
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| WO2013130619A1 (en) | 2012-02-27 | 2013-09-06 | O-Ray Pharma, Inc. | Solid drug implants for intracochlear delivery of therapeutics for the treatment of otic disorders |
| SG11201501815UA (en) | 2012-09-10 | 2015-05-28 | Principia Biopharma Inc | Pyrazolopyrimidine compounds as kinase inhibitors |
| EP3075681B1 (en) | 2013-11-29 | 2021-06-02 | Daizo Corporation | Content-accommodating container, content-accommodating product using same, discharging product, and discharging device |
| KR20160117614A (ko) | 2014-02-21 | 2016-10-10 | 프린시피아 바이오파마, 인코퍼레이티드 | Btk 억제제의 염 및 고체 형태 |
| AU2015364335B2 (en) | 2014-12-18 | 2020-11-26 | Principia Biopharma Inc. | Treatment of pemphigus |
| SG10201912443XA (en) * | 2015-06-03 | 2020-02-27 | Principia Biopharma Inc | Tyrosine kinase inhibitors |
| EP3313839A1 (en) | 2015-06-24 | 2018-05-02 | Principia Biopharma Inc. | Tyrosine kinase inhibitors |
| CN105753863B (zh) * | 2015-09-11 | 2018-07-31 | 东莞市真兴贝特医药技术有限公司 | 氧代二氢咪唑并吡啶类化合物及其应用 |
| EP3414234B1 (en) * | 2015-10-14 | 2022-06-29 | Zibo Biopolar Changsheng Pharmaceutical Co. Ltd. | Bruton's tyrosine kinase inhibitors |
| IL293621B2 (en) | 2016-06-29 | 2023-09-01 | Principia Biopharma Inc | Modified release formulations of 2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)pyrazolo[4,3-d]pyrimidin-1-yl]piperidine-1-carbonyl]-4 -Methyl-4-[4-(oxane-3-yl)piperazine-1-yl)penta-2-ananitrile |
| ES2899114T3 (es) * | 2016-07-25 | 2022-03-10 | Nerviano Medical Sciences Srl | Análogos de purina y 3-deazapurina como inhibidores de colina cinasa |
| EP3585789A1 (en) * | 2017-02-24 | 2020-01-01 | Gilead Sciences, Inc. | Inhibitors of bruton's tyrosine kinase |
| WO2019208805A1 (ja) * | 2018-04-27 | 2019-10-31 | 小野薬品工業株式会社 | Ｂｔｋ阻害活性を有する化合物を有効成分として含む自己免疫疾患の予防および／または治療剤 |
| JP7555327B2 (ja) | 2018-07-25 | 2024-09-24 | ノバルティス アーゲー | Ｎｌｒｐ３インフラマソーム阻害剤 |
| KR102612513B1 (ko) | 2018-07-31 | 2023-12-12 | 록쏘 온콜로지, 인코포레이티드 | (s)-5-아미노-3-(4-((5-플루오로-2-메톡시벤즈아미도)메틸)페닐)-1-(1,1,1-트리플루오로프로판-2-일)-1h-피라졸-4-카르복스아미드의 분무-건조된 분산물 및 제제 |
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