CN1126988A - 二氟平衡酮类似物 - Google Patents
二氟平衡酮类似物 Download PDFInfo
- Publication number
- CN1126988A CN1126988A CN94192700A CN94192700A CN1126988A CN 1126988 A CN1126988 A CN 1126988A CN 94192700 A CN94192700 A CN 94192700A CN 94192700 A CN94192700 A CN 94192700A CN 1126988 A CN1126988 A CN 1126988A
- Authority
- CN
- China
- Prior art keywords
- alkyl
- phenyl
- amino
- benzene
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/28—Radicals substituted by singly-bound oxygen or sulphur atoms
- C07D213/30—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- C07C271/08—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms
- C07C271/10—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C271/22—Esters of carbamic acids having oxygen atoms of carbamate groups bound to acyclic carbon atoms with the nitrogen atoms of the carbamate groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/36—Radicals substituted by singly-bound nitrogen atoms
- C07D213/40—Acylated substituent nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/54—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/56—Amides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/084—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/088—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
- Saccharide Compounds (AREA)
- Phenolic Resins Or Amino Resins (AREA)
- Air Bags (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP93401785.6 | 1993-07-08 | ||
| EP93401785 | 1993-07-08 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN1126988A true CN1126988A (zh) | 1996-07-17 |
Family
ID=8214732
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN94192700A Pending CN1126988A (zh) | 1993-07-08 | 1994-06-07 | 二氟平衡酮类似物 |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US5717093A (enExample) |
| EP (1) | EP0707564B1 (enExample) |
| JP (1) | JPH08512319A (enExample) |
| KR (1) | KR100316864B1 (enExample) |
| CN (1) | CN1126988A (enExample) |
| AT (1) | ATE196465T1 (enExample) |
| AU (1) | AU680009B2 (enExample) |
| CA (1) | CA2166693C (enExample) |
| DE (1) | DE69425971T2 (enExample) |
| ES (1) | ES2152982T3 (enExample) |
| FI (1) | FI120389B (enExample) |
| HU (1) | HUT73411A (enExample) |
| IL (1) | IL110227A0 (enExample) |
| NO (1) | NO306343B1 (enExample) |
| NZ (1) | NZ268202A (enExample) |
| TW (1) | TW288005B (enExample) |
| WO (1) | WO1995001958A1 (enExample) |
| ZA (1) | ZA944818B (enExample) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE179167T1 (de) * | 1993-09-09 | 1999-05-15 | Merrell Pharma Inc | Antivirale analoge von difluorostaton |
| TW200910648A (en) | 2007-08-31 | 2009-03-01 | Isotech Products Inc | Forming process of resin lens of an LED component |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5066643A (en) * | 1985-02-19 | 1991-11-19 | Sandoz Ltd. | Fluorine and chlorine statine or statone containing peptides and method of use |
| CH672792A5 (enExample) * | 1985-02-19 | 1989-12-29 | Sandoz Ag | |
| WO1986006379A1 (en) * | 1985-04-19 | 1986-11-06 | The Upjohn Company | Dihalo-statine substituted renin inhibitors |
| GB8619182D0 (en) * | 1986-08-06 | 1986-09-17 | Sandoz Ltd | Peptides & derivatives |
| NZ223148A (en) * | 1987-01-16 | 1989-10-27 | Merrell Dow Pharma | Peptide derivatives having peptidase inhibition activity |
| BE1002213A5 (fr) * | 1987-04-23 | 1990-10-16 | Sandoz Sa | Nouveaux derives peptidiques, leur preparation et leur utilisation comme medicaments. |
| GB2212158A (en) * | 1987-12-15 | 1989-07-19 | Sandoz Ltd | Trialkylsilymethyl-substituted peptides; renin inhibitors |
| JPH03505875A (ja) * | 1988-07-08 | 1991-12-19 | スミスクライン・ベックマン・コーポレイション | レトロウイルス・プロテアーゼ結合ペプチド |
| IL90872A0 (en) * | 1988-07-08 | 1990-02-09 | Smithkline Beckman Corp | Retroviral protease binding peptides |
| CA2010531A1 (en) * | 1989-03-06 | 1990-09-06 | Werner Neidhart | Amino acid derivatives |
| US5151438A (en) * | 1989-05-23 | 1992-09-29 | Abbott Laboratories | Retroviral protease inhibiting compounds |
| HU210647B (en) * | 1991-01-02 | 1995-06-28 | Merrell Dow Pharma | Process for producing antiviral difluoro-statone derivatives and pharmaceutical compositions containing them |
| CA2131154A1 (en) * | 1992-03-25 | 1993-09-30 | Colin W. Greengrass | Antiviral peptides |
| GB9210744D0 (en) * | 1992-05-20 | 1992-07-08 | Pfizer Ltd | Antiviral peptides |
| EP0957093A3 (en) * | 1992-05-21 | 2000-04-12 | Monsanto Company | Retrovial protease inhibitors |
| CN1152910A (zh) * | 1994-07-15 | 1997-06-25 | 默里尔药物公司 | 二氟斯塔酮抗病毒剂 |
| AU2014214806B2 (en) | 2013-02-08 | 2017-02-16 | Tait Towers Manufacturing, LLC | Visually flying platform with visually transparent flexible support members |
-
1994
- 1994-06-07 CA CA002166693A patent/CA2166693C/en not_active Expired - Fee Related
- 1994-06-07 DE DE69425971T patent/DE69425971T2/de not_active Expired - Lifetime
- 1994-06-07 JP JP7504027A patent/JPH08512319A/ja active Pending
- 1994-06-07 EP EP94920095A patent/EP0707564B1/en not_active Expired - Lifetime
- 1994-06-07 ES ES94920095T patent/ES2152982T3/es not_active Expired - Lifetime
- 1994-06-07 HU HU9503706A patent/HUT73411A/hu unknown
- 1994-06-07 NZ NZ268202A patent/NZ268202A/en unknown
- 1994-06-07 AU AU71008/94A patent/AU680009B2/en not_active Ceased
- 1994-06-07 US US08/578,698 patent/US5717093A/en not_active Expired - Lifetime
- 1994-06-07 WO PCT/US1994/006376 patent/WO1995001958A1/en not_active Ceased
- 1994-06-07 AT AT94920095T patent/ATE196465T1/de not_active IP Right Cessation
- 1994-06-07 CN CN94192700A patent/CN1126988A/zh active Pending
- 1994-06-07 KR KR1019960700062A patent/KR100316864B1/ko not_active Expired - Fee Related
- 1994-07-04 ZA ZA944818A patent/ZA944818B/xx unknown
- 1994-07-05 TW TW083106128A patent/TW288005B/zh active
- 1994-07-06 IL IL11022794A patent/IL110227A0/xx unknown
-
1996
- 1996-01-05 NO NO960048A patent/NO306343B1/no not_active IP Right Cessation
- 1996-01-05 FI FI960051A patent/FI120389B/fi not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| ES2152982T3 (es) | 2001-02-16 |
| AU7100894A (en) | 1995-02-06 |
| KR960703844A (ko) | 1996-08-31 |
| DE69425971D1 (de) | 2000-10-26 |
| NO960048D0 (no) | 1996-01-05 |
| HUT73411A (en) | 1996-07-29 |
| HU9503706D0 (en) | 1996-02-28 |
| US5717093A (en) | 1998-02-10 |
| FI960051L (fi) | 1996-03-07 |
| EP0707564B1 (en) | 2000-09-20 |
| FI960051A0 (fi) | 1996-01-05 |
| WO1995001958A1 (en) | 1995-01-19 |
| CA2166693C (en) | 1999-08-24 |
| DE69425971T2 (de) | 2001-05-23 |
| NO306343B1 (no) | 1999-10-25 |
| AU680009B2 (en) | 1997-07-17 |
| IL110227A0 (en) | 1994-10-21 |
| ATE196465T1 (de) | 2000-10-15 |
| EP0707564A1 (en) | 1996-04-24 |
| JPH08512319A (ja) | 1996-12-24 |
| ZA944818B (en) | 1995-02-22 |
| CA2166693A1 (en) | 1995-01-09 |
| FI120389B (fi) | 2009-10-15 |
| NO960048L (no) | 1996-03-05 |
| NZ268202A (en) | 1997-09-22 |
| KR100316864B1 (ko) | 2002-11-13 |
| TW288005B (enExample) | 1996-10-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C06 | Publication | ||
| PB01 | Publication | ||
| C10 | Entry into substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C02 | Deemed withdrawal of patent application after publication (patent law 2001) | ||
| WD01 | Invention patent application deemed withdrawn after publication |