CN112533897B - 赖氨酰氧化酶的卤代烯丙胺砜衍生抑制剂及其用途 - Google Patents

赖氨酰氧化酶的卤代烯丙胺砜衍生抑制剂及其用途 Download PDF

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CN112533897B
CN112533897B CN201980051571.9A CN201980051571A CN112533897B CN 112533897 B CN112533897 B CN 112533897B CN 201980051571 A CN201980051571 A CN 201980051571A CN 112533897 B CN112533897 B CN 112533897B
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cycloalkyl
cancer
fibrosis
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CN112533897A (zh
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艾莉森·桃乐丝·芬得利
克雷格·伊旺·特纳
曼达·迪奥达
强纳森·史都华·甫特
沃尔夫冈·杰洛利梅克
周文斌
A·布森
A·E·格雷克
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Pharmaxis Ltd
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CN201980051571.9A 2018-08-03 2019-08-02 赖氨酰氧化酶的卤代烯丙胺砜衍生抑制剂及其用途 Active CN112533897B (zh)

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Application Number Priority Date Filing Date Title
AU2018902829 2018-08-03
AU2018902829A AU2018902829A0 (en) 2018-08-03 Haloallylamine sulfone derivative inhibitors of lysyl oxidases and uses thereof
PCT/AU2019/050811 WO2020024017A1 (en) 2018-08-03 2019-08-02 Haloallylamine sulfone derivative inhibitors of lysyl oxidases and uses thereof

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CN112533897B true CN112533897B (zh) 2023-07-14

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US12233056B2 (en) * 2022-04-06 2025-02-25 Syntara Limited Lysyl oxidase inhibitors for treating myeloid malignancies
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WO2009066152A2 (en) * 2007-11-21 2009-05-28 Pharmaxis Ltd. Haloallylamine inhibitors of ssao/vap-1 and uses therefor
CN104520268A (zh) * 2012-05-02 2015-04-15 法马克西斯制药公司 Ssao的取代的3-卤代烯丙基胺抑制剂及其用途
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