CN111094252B - 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物 - Google Patents

5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物 Download PDF

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CN111094252B
CN111094252B CN201880059865.1A CN201880059865A CN111094252B CN 111094252 B CN111094252 B CN 111094252B CN 201880059865 A CN201880059865 A CN 201880059865A CN 111094252 B CN111094252 B CN 111094252B
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mixture
solution
crystalline form
crystalline
composition
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CN111094252A (zh
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迈克尔·格劳鲍历克
加仑·苏伊士
佐顿·内梅
萨马·阿拉斯比
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Adamaksim Co ltd
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00—Fungicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CN201880059865.1A 2017-07-17 2018-07-16 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物 Active CN111094252B (zh)

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CN202410543394.9A CN118515619A (zh) 2017-07-17 2018-07-16 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物

Applications Claiming Priority (3)

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US201762533509P 2017-07-17 2017-07-17
US62/533,509 2017-07-17
PCT/IB2018/000875 WO2019038583A1 (en) 2017-07-17 2018-07-16 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2-ONE POLYMORPHS

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CN202410543394.9A Division CN118515619A (zh) 2017-07-17 2018-07-16 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物

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CN111094252B true CN111094252B (zh) 2024-05-24

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CN202410543394.9A Pending CN118515619A (zh) 2017-07-17 2018-07-16 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物
CN201880059865.1A Active CN111094252B (zh) 2017-07-17 2018-07-16 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物

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US (1) US11632954B2 (enExample)
EP (1) EP3655396A1 (enExample)
JP (3) JP2020527563A (enExample)
CN (2) CN118515619A (enExample)
AR (1) AR112276A1 (enExample)
AU (1) AU2018320492C1 (enExample)
CA (1) CA3069619A1 (enExample)
IL (5) IL271950B2 (enExample)
MA (1) MA49639A (enExample)
WO (1) WO2019038583A1 (enExample)
ZA (1) ZA202000411B (enExample)

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AU2023227455A1 (en) 2022-03-03 2024-09-19 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AU2023275068A1 (en) 2022-05-26 2024-11-28 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AR130107A1 (es) 2022-08-03 2024-11-06 Adama Makhteshim Ltd 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona para hongos resistentes a fungicidas
AU2024233301A1 (en) 2023-03-09 2025-09-18 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
WO2024189563A1 (en) 2023-03-14 2024-09-19 Adama Makhteshim Ltd. Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber
AR132381A1 (es) 2023-04-11 2025-06-18 Adama Makhteshim Ltd Compuestos y procesos relativos a flumetilsulforim
AR133680A1 (es) 2023-08-31 2025-10-22 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
WO2025114931A1 (en) 2023-11-28 2025-06-05 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof

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WO2019038583A1 (en) 2019-02-28
IL323266A (en) 2025-11-01
NZ761039A (en) 2023-09-29
JP2023145572A (ja) 2023-10-11
IL323268A (en) 2025-11-01
EP3655396A1 (en) 2020-05-27
AU2018320492C1 (en) 2023-07-13
AU2018320492A1 (en) 2020-02-13
IL271950B1 (en) 2024-02-01
IL271950B2 (en) 2024-06-01
MA49639A (fr) 2020-05-27
US20200229437A1 (en) 2020-07-23
US11632954B2 (en) 2023-04-25
IL309708B1 (en) 2025-10-01
AR112276A1 (es) 2019-10-09
IL309708A (en) 2024-02-01
IL323267A (en) 2025-11-01
CN118515619A (zh) 2024-08-20
JP2025163080A (ja) 2025-10-28
IL271950A (en) 2020-02-27
BR112020000953A2 (pt) 2020-07-14
CA3069619A1 (en) 2019-02-28
CN111094252A (zh) 2020-05-01
JP2020527563A (ja) 2020-09-10
AU2018320492B2 (en) 2022-12-01
ZA202000411B (en) 2023-10-25

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