AU2018320492C1 - Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one - Google Patents

Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one Download PDF

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AU2018320492C1
AU2018320492C1 AU2018320492A AU2018320492A AU2018320492C1 AU 2018320492 C1 AU2018320492 C1 AU 2018320492C1 AU 2018320492 A AU2018320492 A AU 2018320492A AU 2018320492 A AU2018320492 A AU 2018320492A AU 2018320492 C1 AU2018320492 C1 AU 2018320492C1
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solution
crystalline form
compound
crystalline
filtering
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AU2018320492A1 (en
AU2018320492B2 (en
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Samaa ALASIBI
Michael Grabarnick
Zoltán NEMET
Gal SUEZ
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Adama Makhteshim Ltd
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Adama Makhteshim Ltd
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00—Fungicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Environmental Sciences (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2018320492A 2017-07-17 2018-07-16 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one Active AU2018320492C1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762533509P 2017-07-17 2017-07-17
US62/533,509 2017-07-17
PCT/IB2018/000875 WO2019038583A1 (en) 2017-07-17 2018-07-16 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2-ONE POLYMORPHS

Publications (3)

Publication Number Publication Date
AU2018320492A1 AU2018320492A1 (en) 2020-02-13
AU2018320492B2 AU2018320492B2 (en) 2022-12-01
AU2018320492C1 true AU2018320492C1 (en) 2023-07-13

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AU2018320492A Active AU2018320492C1 (en) 2017-07-17 2018-07-16 Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one

Country Status (11)

Country Link
US (1) US11632954B2 (enExample)
EP (1) EP3655396A1 (enExample)
JP (3) JP2020527563A (enExample)
CN (2) CN118515619A (enExample)
AR (1) AR112276A1 (enExample)
AU (1) AU2018320492C1 (enExample)
CA (1) CA3069619A1 (enExample)
IL (5) IL271950B2 (enExample)
MA (1) MA49639A (enExample)
WO (1) WO2019038583A1 (enExample)
ZA (1) ZA202000411B (enExample)

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IL321760A (en) 2019-07-22 2025-08-01 Adama Makhteshim Ltd Fungicidal combinations, mixtures and compositions and uses thereof
US12466796B2 (en) * 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound
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CA3206570A1 (en) 2021-01-27 2022-08-04 Alexandra ROSENMUND 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1 h)-one for controlling plant diseases
CA3216622A1 (en) 2021-05-04 2022-11-10 Stefano Luca Giaffreda Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof
AU2023227455A1 (en) 2022-03-03 2024-09-19 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AU2023275068A1 (en) 2022-05-26 2024-11-28 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
AR130107A1 (es) 2022-08-03 2024-11-06 Adama Makhteshim Ltd 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona para hongos resistentes a fungicidas
AU2024233301A1 (en) 2023-03-09 2025-09-18 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof
WO2024189563A1 (en) 2023-03-14 2024-09-19 Adama Makhteshim Ltd. Liquid compositions containing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1h)-one and derivatives thereof and a uv absorber
AR132381A1 (es) 2023-04-11 2025-06-18 Adama Makhteshim Ltd Compuestos y procesos relativos a flumetilsulforim
AR133680A1 (es) 2023-08-31 2025-10-22 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
WO2025114931A1 (en) 2023-11-28 2025-06-05 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof

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WO2019038583A1 (en) 2019-02-28
IL323266A (en) 2025-11-01
NZ761039A (en) 2023-09-29
JP2023145572A (ja) 2023-10-11
IL323268A (en) 2025-11-01
EP3655396A1 (en) 2020-05-27
AU2018320492A1 (en) 2020-02-13
IL271950B1 (en) 2024-02-01
IL271950B2 (en) 2024-06-01
MA49639A (fr) 2020-05-27
US20200229437A1 (en) 2020-07-23
US11632954B2 (en) 2023-04-25
IL309708B1 (en) 2025-10-01
AR112276A1 (es) 2019-10-09
IL309708A (en) 2024-02-01
IL323267A (en) 2025-11-01
CN118515619A (zh) 2024-08-20
JP2025163080A (ja) 2025-10-28
IL271950A (en) 2020-02-27
BR112020000953A2 (pt) 2020-07-14
CN111094252B (zh) 2024-05-24
CA3069619A1 (en) 2019-02-28
CN111094252A (zh) 2020-05-01
JP2020527563A (ja) 2020-09-10
AU2018320492B2 (en) 2022-12-01
ZA202000411B (en) 2023-10-25

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