CN107669534A - 具有消除眼袋功效的美容霜的制备方法 - Google Patents
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Abstract
本发明涉及具有消除眼袋功效的美容霜的制备方法,属于化妆品领域。本发明的具有消除眼袋功效的美容霜的制备方法通过以下方法制备而成:(1)制备水相:按重量份将艾纳香提取物2‑5份,卷柏提取物3‑6份,仙鹤草提取物1‑4份,石榴皮鞣花酸1‑4份,月桂醇硫酸酯三乙醇胺盐10‑16份,椰油酰胺丙基甜菜碱12‑20份和燕麦β-葡聚糖5‑10份加入纯化水中,搅拌均匀,加热至80‑85℃;(2)制备油相:按重量份将四‑(二丁基羟基氢化肉桂酸)季戊四醇酯0.1‑0.2份,十六烷基二甲基硅氧烷共聚物1‑5份,2,6‑二叔丁基羟基甲苯0.01‑0.05份,PEG‑40氢化蓖麻油0.2‑0.5份,玫瑰香精0.1‑0.5份,丙二醇15‑18份和辛二醇10‑15份混合均匀,加热至80‑85℃;(3)将水相和油相混合均匀,冷却至室温,即得。本发明的美容霜经临床验证消除眼袋效果显著,取得了优异的技术效果。
Description
技术领域
本发明涉及化妆品领域,具体涉及一种具有消除眼袋功效的美容霜的制备方法。
背景技术
眼部肌肤是人体最薄肌肤,同时又是活动最频繁的部位,而且还是化妆中拉扯皮肤次数最多的地方,非常容易长出皱纹,并且一旦长出就很难消。
眼霜属于护肤类化妆产品,有滋润功效,除了可以减低黑眼圈、眼袋问题外,同时也具备改善皱纹、细纹的功效。眼霜是用来保护眼睛周围比较薄的这一层皮肤的,对眼袋、黑眼圈、鱼尾纹等都有一定的效用,但是不同的眼霜有不同的作用。眼霜的种类很多,大致分为眼膜、眼胶、眼部啫喱、眼贴、眼霜等;从功能上分为滋润眼霜、紧实眼霜、抗老化眼霜、抗敏眼霜等等。
艾纳香(Blumeabalsamifera(L.)DC.)为菊科艾纳香属BlumeabalsamiferaDC,苗药名档窝凯Diangdvobbvid植物,药用为枝叶、嫩枝根、别名:大风艾、客家人叫法(大毛风)艾纳香冰片艾、家风艾、大毛药、大艾等。具有温中活血,祛风除湿,杀虫。治寒湿泻痢,腹痛肠鸣,肿胀,筋骨疼痛,跌打损伤,癣疮,通诸窍散郁火,消肿止痛等功效。
卷柏〔Selaginellatamariscina(P.Beauv.)Spring〕,卷柏科卷柏属土生或石生复苏植物,呈垫状。靠孢子繁殖。卷柏又名九死还魂草,根能自行从土壤分离,蜷缩似拳状,随风移动,遇水而荣,根重新再钻到土壤里寻找水份。因其耐旱力极强,在长期干旱后只要根系在水中浸泡后就又可舒展,故而得名。卷柏全草含苏铁双黄酮(sotetsuflavone),穗花杉双黄酮(amentoflavone),扁柏双黄酮(hinokiflavone),异柳杉双黄酮(isocryptomerin),柳杉双黄酮(cryptomerin)B,芹菜素(apigenin)和海藻糖(trehalose)等活性成分。具有抗癌作用、止血作用、抑菌作用(100%卷柏煎剂用平板打洞法,对金黄色葡萄球菌有抑制作用)和解痉作用。
仙鹤草别名脱力草、瓜香草、老牛筋、狼芽草。来源为蔷薇科植物龙芽草Agrimoniapilosa Ledeb.的地上部分。全草夏、秋季采收。芽冬、春季新株萌发前采收。植物形态多年生草本,高达1m,全株具白色长毛。根茎短,常生1或数个根芽(越冬芽)。茎直立,被疏柔毛及腺毛。羽状复叶互生,小叶大小不等,间隔排列,卵圆形至倒卵圆形,长2.5~7cm,宽1.5~3.5cm,边缘有锯齿,两面均被柔毛;托叶近卵形。总状花序顶生;花萼倒圆锥形,5裂,裂片基部生多数钩状刚毛,宿存;花瓣5,黄色;雄蕊5~15;子房半下位,花柱突出。萼筒于果熟时增厚,下垂,顶端有一轮直立钩刺,外有较深纵沟。极似仙鹤头部,因而称仙鹤草。含仙鹤草酚(agrimophol)、仙鹤草内酯(agrimonolide),并含木犀草甙(luteoloside)、仙鹤草甲、乙、丙素(agrimoninA,B,C)、赛仙鹤草酚A~E(agrimolA~E),另含鞣质、甾醇、皂甙及挥发油。性味性平,味苦、涩。具有止血,促进血液凝固,强心,调整心率,大量服用能使心搏徐缓,抗菌和驱虫功效。
发明内容
本发明的目的是充分利用艾纳香、卷柏和仙鹤草,提供一种具有消除眼袋功效的美容霜的制备方法。
本发明解决该技术问题的技术方案是:
一种具有消除眼袋功效的美容霜的制备方法,其通过以下方法制备而成:
(1)制备水相:按重量份将艾纳香提取物2-5份,卷柏提取物3-6份,仙鹤草提取物1-4份,石榴皮鞣花酸1-4份,月桂醇硫酸酯三乙醇胺盐10-16份,椰油酰胺丙基甜菜碱12-20份和燕麦β-葡聚糖5-10份加入纯化水中,搅拌均匀,加热至80-85℃;
(2)制备油相:按重量份将四-(二丁基羟基氢化肉桂酸)季戊四醇酯0.1-0.2份,十六烷基二甲基硅氧烷共聚物1-5份,2,6-二叔丁基羟基甲苯0.01-0.05份,PEG-40氢化蓖麻油0.2-0.5份,玫瑰香精0.1-0.5份,丙二醇15-18份和辛二醇10-15份混合均匀,加热至80-85℃;
(3)将水相和油相混合均匀,冷却至室温,即得。
所述步骤(1)中各组分的重量份数优选为:艾纳香提取物3份,卷柏提取物4份,仙鹤草提取物3份,石榴皮鞣花酸3份,月桂醇硫酸酯三乙醇胺盐12份,椰油酰胺丙基甜菜碱15份和燕麦β-葡聚糖8份。
所述步骤(2)中各组分的重量份数优选为:四-(二丁基羟基氢化肉桂酸)季戊四醇酯0.1份,十六烷基二甲基硅氧烷共聚物3份,2,6-二叔丁基羟基甲苯0.03份,PEG-40氢化蓖麻油0.3份,玫瑰香精0.3份,丙二醇16份和辛二醇12份。
所述步骤(1)和步骤(2)的加热温度优选为85℃。
所述艾纳香提取物、卷柏提取物和仙鹤草提取物可以通过本领域常规水提和醇提方法制备,例如所述艾纳香提取物的制备方法为:取艾纳香枝叶干燥粉碎,加入石油醚脱脂后用50%乙醇按料液比1:(20-30)于30-40℃提取1-2h,重复提取三次,合并滤液,于90℃旋转蒸发得稠膏,干燥,粉碎,即得;所述卷柏提取物的制备方法为:将卷柏干燥全草粉碎过80目,至于10-12倍量的蒸馏水中,超声提取后过滤,1500r/min离心2-3h,浓缩,干燥,即得;所述仙鹤草提取物的制备方法为:按料液比1:12-15加入60%乙醇,用超声波辅助提取3次,每次1h,过滤,收集合并滤液,减压浓缩,干燥即得。
本发明的美容霜经临床验证消除眼袋效果显著,取得了优异的技术效果。
具体实施方式
实施例1
(1)取艾纳香枝叶干燥粉碎,加入石油醚脱脂后用50%乙醇按料液比1:25于35℃提取2h,重复提取三次,合并滤液,于90℃旋转蒸发得稠膏,干燥,粉碎,即得艾纳香提取物;将卷柏干燥全草粉碎过80目,至于10倍量的蒸馏水中,超声提取后过滤,1500r/min离心2h,浓缩,干燥,即得卷柏提取物;按料液比1:12在仙鹤草中加入60%乙醇,用超声波辅助提取3次,每次1h,过滤,收集合并滤液,减压浓缩,干燥即得;
(2)制备水相:按重量份将艾纳香提取物3份,卷柏提取物3份,仙鹤草提取物2份,石榴皮鞣花酸2份,月桂醇硫酸酯三乙醇胺盐12份,椰油酰胺丙基甜菜碱15份和燕麦β-葡聚糖6份加入纯化水中,搅拌均匀,加热至80℃;
(3)制备油相:按重量份将四-(二丁基羟基氢化肉桂酸)季戊四醇酯0.1份,十六烷基二甲基硅氧烷共聚物2份,2,6-二叔丁基羟基甲苯0.02份,PEG-40氢化蓖麻油0.2份,玫瑰香精0.2份,丙二醇16份和辛二醇12份混合均匀,加热至80℃;
(4)将水相和油相混合均匀,冷却至室温,即得。
实施例2
(1)制备水相:按重量份将实施例1的艾纳香提取物4份,卷柏提取物4份,仙鹤草提取物3份,石榴皮鞣花酸3份,月桂醇硫酸酯三乙醇胺盐13份,椰油酰胺丙基甜菜碱15份和燕麦β-葡聚糖8份加入纯化水中,搅拌均匀,加热至80℃;
(2)制备油相:按重量份将四-(二丁基羟基氢化肉桂酸)季戊四醇酯0.2份,十六烷基二甲基硅氧烷共聚物3份,2,6-二叔丁基羟基甲苯0.03份,PEG-40氢化蓖麻油0.3份,玫瑰香精0.3份,丙二醇16份和辛二醇13份混合均匀,加热至80℃;
(3)将水相和油相混合均匀,冷却至室温,即得。
实施例3
(1)制备水相:按重量份将实施例1的艾纳香提取物5份,卷柏提取物6份,仙鹤草提取物4份,石榴皮鞣花酸4份,月桂醇硫酸酯三乙醇胺盐16份,椰油酰胺丙基甜菜碱20份和燕麦β-葡聚糖10份加入纯化水中,搅拌均匀,加热至85℃;
(2)制备油相:按重量份将四-(二丁基羟基氢化肉桂酸)季戊四醇酯0.2份,十六烷基二甲基硅氧烷共聚物5份,2,6-二叔丁基羟基甲苯0.05份,PEG-40氢化蓖麻油0.5份,玫瑰香精0.5份,丙二醇18份和辛二醇15份混合均匀,加热至85℃;
(3)将水相和油相混合均匀,冷却至室温,即得。
试验例1本发明的美容霜消除眼袋的效果研究
选用180名受试者,男78名,女102名,年龄在18-42岁之间,其中60名有单纯皮肤松弛型眼袋,症状普遍为下睑及外眦皮肤松弛,无眶隔松弛,无眶隔脂肪突出,眼周出现细小皱纹,60名有单纯眼轮匝肌肥厚型眼袋,症状普遍表现为靠近下睑缘,呈弧形连续分布,皮肤并不松弛,60名有下睑膨隆型眼袋,症状普遍表现为皮肤、眼轮匝肌及眶隔松弛。受试者每日使用本发明实施例1的美容霜2次,早晚各一次,历时两个月,经专家检验效果,停止使用1个月之后,再次检验是否复发,各种检查标准为:
有效:眼袋全部消除,未复发;
良好:眼袋基本消除,未复发
基本有效:眼袋基本消除,复发
无效:眼袋明显
检测结果如表1所示:
表1本发明美容霜的消除眼袋效果研究
单纯皮肤松弛型眼袋 | 单纯眼轮匝肌肥厚型眼袋 | 下睑膨隆型眼袋 | |
有效 | 53 | 48 | 50 |
良好 | 2 | 10 | 6 |
基本有效 | 3 | 2 | 3 |
无效 | 2 | 0 | 1 |
结果显示,本发明的美容霜对于单纯皮肤松弛型眼袋的有效率高达88%,良好有效率高达92%,对于单纯眼轮匝肌肥厚型眼袋的有效率高达80%,良好有效率高达97%,对于下睑膨隆型眼袋的有效率高达83%,良好有效率高达93%,表明本发明的美容霜消除眼袋效果显著。
Claims (5)
1.具有消除眼袋功效的美容霜的制备方法,其特征在于,其通过以下方法制备而成:
(1)制备水相:按重量份将艾纳香提取物2-5份,卷柏提取物3-6份,仙鹤草提取物1-4份,石榴皮鞣花酸1-4份,月桂醇硫酸酯三乙醇胺盐10-16份,椰油酰胺丙基甜菜碱12-20份和燕麦β-葡聚糖5-10份加入纯化水中,搅拌均匀,加热至80-85℃;
(2)制备油相:按重量份将四-(二丁基羟基氢化肉桂酸)季戊四醇酯0.1-0.2份,十六烷基二甲基硅氧烷共聚物1-5份,2,6-二叔丁基羟基甲苯0.01-0.05份,PEG-40氢化蓖麻油0.2-0.5份,玫瑰香精0.1-0.5份,丙二醇15-18份和辛二醇10-15份混合均匀,加热至80-85℃;
(3)将水相和油相混合均匀,冷却至室温,即得。
2.根据权利要求1所述的具有消除眼袋功效的美容霜的制备方法,其特征在于,所述步骤(1)中各组分的重量份数优选为:艾纳香提取物3份,卷柏提取物4份,仙鹤草提取物3份,石榴皮鞣花酸3份,月桂醇硫酸酯三乙醇胺盐12份,椰油酰胺丙基甜菜碱15份和燕麦β-葡聚糖8份。
3.根据权利要求1所述的具有消除眼袋功效的美容霜的制备方法,其特征在于,所述步骤(2)中各组分的重量份数优选为:四-(二丁基羟基氢化肉桂酸)季戊四醇酯0.1份,十六烷基二甲基硅氧烷共聚物3份,2,6-二叔丁基羟基甲苯0.03份,PEG-40氢化蓖麻油0.3份,玫瑰香精0.3份,丙二醇16份和辛二醇12份。
4.根据权利要求1所述的具有消除眼袋功效的美容霜的制备方法,其特征在于,所述步骤(1)和步骤(2)的加热温度优选为85℃。
5.根据权利要求1-4任一项所述的具有消除眼袋功效的美容霜的制备方法,其特征在于,所述艾纳香提取物的制备方法为:取艾纳香枝叶干燥粉碎,加入石油醚脱脂后用50%乙醇按料液比1:(20-30)于30-40℃提取1-2h,重复提取三次,合并滤液,于90℃旋转蒸发得稠膏,干燥,粉碎,即得;所述卷柏提取物的制备方法为:将卷柏干燥全草粉碎过80目,至于10-12倍量的蒸馏水中,超声提取后过滤,1500r/min离心2-3h,浓缩,干燥,即得;所述仙鹤草提取物的制备方法为:按料液比1:12-15加入60%乙醇,用超声波辅助提取3次,每次1h,过滤,收集合并滤液,减压浓缩,干燥即得。
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CN105920379A (zh) * | 2015-12-31 | 2016-09-07 | 青岛安倍康生物医药技术有限公司 | 一种缓解眼袋的中药眼霜及其制备方法 |
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