CN1072413A - 氨基酸衍生物 - Google Patents

氨基酸衍生物 Download PDF

Info

Publication number
CN1072413A
CN1072413A CN92113665A CN92113665A CN1072413A CN 1072413 A CN1072413 A CN 1072413A CN 92113665 A CN92113665 A CN 92113665A CN 92113665 A CN92113665 A CN 92113665A CN 1072413 A CN1072413 A CN 1072413A
Authority
CN
China
Prior art keywords
cyclopropyl
pyridyl
triazolo
pyrazine
pyridylmethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN92113665A
Other languages
English (en)
Chinese (zh)
Inventor
H·施塔德勒
E·维尔拉
W·沃斯尔
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=25691089&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN1072413(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of CN1072413A publication Critical patent/CN1072413A/zh
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CN92113665A 1991-11-19 1992-11-18 氨基酸衍生物 Pending CN1072413A (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CH337491 1991-11-19
CH3374/91 1991-11-19
CH2665/92 1992-08-28
CH266592 1992-08-28

Publications (1)

Publication Number Publication Date
CN1072413A true CN1072413A (zh) 1993-05-26

Family

ID=25691089

Family Applications (1)

Application Number Title Priority Date Filing Date
CN92113665A Pending CN1072413A (zh) 1991-11-19 1992-11-18 氨基酸衍生物

Country Status (12)

Country Link
EP (1) EP0543245A1 (enExample)
JP (1) JPH05239059A (enExample)
CN (1) CN1072413A (enExample)
AU (1) AU2841392A (enExample)
BG (1) BG97094A (enExample)
CA (1) CA2081236A1 (enExample)
FI (1) FI925068L (enExample)
HU (1) HU9203580D0 (enExample)
IL (1) IL103743A0 (enExample)
IS (1) IS3947A (enExample)
NO (1) NO924423L (enExample)
TW (1) TW275630B (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2615284B2 (ja) * 1991-08-19 1997-05-28 三菱重工業 株式会社 アルミニウム複合品の製造方法
US5481008A (en) * 1993-09-13 1996-01-02 Hoffmann-La Roche Inc. Process for the preparation of optically active compounds
JP4794446B2 (ja) * 2003-09-23 2011-10-19 メルク・シャープ・エンド・ドーム・コーポレイション イソキノリン系カリウムチャンネル阻害薬

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1328333C (en) * 1988-03-04 1994-04-05 Quirico Branca Amino acid derivatives
AU629867B2 (en) * 1988-11-17 1992-10-15 Imperial Chemical Industries Plc Triazolo (4,3a) pyrazine derivatives
CA2044564A1 (en) * 1990-06-28 1991-12-29 Quirico Branca Amino acid derivatives

Also Published As

Publication number Publication date
BG97094A (bg) 1993-12-24
HU9203580D0 (en) 1993-01-28
FI925068A0 (fi) 1992-11-09
AU2841392A (en) 1993-05-20
NO924423L (no) 1993-05-20
CA2081236A1 (en) 1993-04-24
IL103743A0 (en) 1993-04-04
EP0543245A1 (de) 1993-05-26
JPH05239059A (ja) 1993-09-17
TW275630B (enExample) 1996-05-11
FI925068A7 (fi) 1993-05-20
NO924423D0 (no) 1992-11-17
FI925068L (fi) 1993-05-20
IS3947A (is) 1993-05-20

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Legal Events

Date Code Title Description
C06 Publication
PB01 Publication
C01 Deemed withdrawal of patent application (patent law 1993)
WD01 Invention patent application deemed withdrawn after publication