CN105916500A - 用于治疗炎性疾病的化合物、药物组合物和方法 - Google Patents
用于治疗炎性疾病的化合物、药物组合物和方法 Download PDFInfo
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- CN105916500A CN105916500A CN201480073506.3A CN201480073506A CN105916500A CN 105916500 A CN105916500 A CN 105916500A CN 201480073506 A CN201480073506 A CN 201480073506A CN 105916500 A CN105916500 A CN 105916500A
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- pyrrolidine
- chlorophenyl
- carboxylic acid
- biphenyl
- carbonyl
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- 0 CC(*)(C1)C(*)(*)C(*)(C(O*)=O)N(*IC[Al]*)C1(C)I* Chemical compound CC(*)(C1)C(*)(*)C(*)(C(O*)=O)N(*IC[Al]*)C1(C)I* 0.000 description 4
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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- Engineering & Computer Science (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Immunology (AREA)
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- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Diabetes (AREA)
- Virology (AREA)
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- Pain & Pain Management (AREA)
- AIDS & HIV (AREA)
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- Neurology (AREA)
- Molecular Biology (AREA)
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- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202210539668.8A CN114773249B (zh) | 2013-11-27 | 2014-11-27 | 用于治疗炎性疾病的化合物、药物组合物和方法 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP13194730.1 | 2013-11-27 | ||
| EP13194730 | 2013-11-27 | ||
| PCT/EP2014/075768 WO2015078949A1 (en) | 2013-11-27 | 2014-11-27 | Compounds, pharmaceutical composition and methods for use in treating inflammatory diseases |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202210539668.8A Division CN114773249B (zh) | 2013-11-27 | 2014-11-27 | 用于治疗炎性疾病的化合物、药物组合物和方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN105916500A true CN105916500A (zh) | 2016-08-31 |
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Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN201480073506.3A Pending CN105916500A (zh) | 2013-11-27 | 2014-11-27 | 用于治疗炎性疾病的化合物、药物组合物和方法 |
| CN202210539668.8A Active CN114773249B (zh) | 2013-11-27 | 2014-11-27 | 用于治疗炎性疾病的化合物、药物组合物和方法 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202210539668.8A Active CN114773249B (zh) | 2013-11-27 | 2014-11-27 | 用于治疗炎性疾病的化合物、药物组合物和方法 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US9770435B2 (https=) |
| EP (2) | EP3610872A1 (https=) |
| JP (2) | JP6854126B2 (https=) |
| KR (1) | KR102259934B1 (https=) |
| CN (2) | CN105916500A (https=) |
| AU (1) | AU2014356460B2 (https=) |
| BR (1) | BR112016011917B1 (https=) |
| CA (1) | CA2929436C (https=) |
| DK (1) | DK3074008T3 (https=) |
| EA (1) | EA032271B9 (https=) |
| ES (1) | ES2755332T3 (https=) |
| MX (1) | MX2016006975A (https=) |
| WO (1) | WO2015078949A1 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN113816818A (zh) * | 2021-09-17 | 2021-12-21 | 哈尔滨工业大学(深圳) | 一种铜催化不对称烯丙基烷基化反应方法及手性化合物 |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10550091B2 (en) | 2016-03-25 | 2020-02-04 | St. Jude Children's Research Hospital | 1,4,5-substituted 1,2,3-triazole analogues as antagonists of the pregnane X receptor |
| BR102018007822A2 (pt) | 2017-04-20 | 2018-11-06 | Gilead Sciences, Inc. | composto, métodos para inibir pd-1, pd-l1 e/ou interação de pd-1/pd-l1 e para tratamento de câncer, composição farmacêutica, e, kit para tratamento de ou prevenção de câncer ou uma doença ou condição |
| TWI707849B (zh) | 2018-02-13 | 2020-10-21 | 美商基利科學股份有限公司 | Pd‐1/pd‐l1抑制劑 |
| KR102591947B1 (ko) | 2018-04-19 | 2023-10-25 | 길리애드 사이언시즈, 인코포레이티드 | Pd-1/pd-l1 억제제 |
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| EA032271B1 (ru) | 2019-05-31 |
| ES2755332T3 (es) | 2020-04-22 |
| EP3074008A1 (en) | 2016-10-05 |
| US9770435B2 (en) | 2017-09-26 |
| EA201690783A1 (ru) | 2016-08-31 |
| CN114773249A (zh) | 2022-07-22 |
| MX2016006975A (es) | 2016-10-12 |
| WO2015078949A1 (en) | 2015-06-04 |
| US20160303075A1 (en) | 2016-10-20 |
| EA032271B9 (ru) | 2019-08-30 |
| JP2019178152A (ja) | 2019-10-17 |
| AU2014356460A1 (en) | 2016-05-19 |
| HK1224184A1 (en) | 2017-08-18 |
| BR112016011917A2 (https=) | 2017-08-08 |
| KR20160079907A (ko) | 2016-07-06 |
| EP3610872A1 (en) | 2020-02-19 |
| CA2929436A1 (en) | 2015-06-04 |
| CN114773249B (zh) | 2024-08-16 |
| DK3074008T3 (da) | 2019-10-21 |
| AU2014356460B2 (en) | 2020-01-16 |
| KR102259934B1 (ko) | 2021-06-03 |
| CA2929436C (en) | 2021-06-15 |
| JP6854126B2 (ja) | 2021-04-07 |
| JP2017503758A (ja) | 2017-02-02 |
| BR112016011917B1 (pt) | 2022-10-11 |
| EP3074008B1 (en) | 2019-09-04 |
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