CN104292229A - 2-苯氧基嘧啶酮类似物 - Google Patents
2-苯氧基嘧啶酮类似物 Download PDFInfo
- Publication number
- CN104292229A CN104292229A CN201410468406.2A CN201410468406A CN104292229A CN 104292229 A CN104292229 A CN 104292229A CN 201410468406 A CN201410468406 A CN 201410468406A CN 104292229 A CN104292229 A CN 104292229A
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- CN
- China
- Prior art keywords
- compound
- fluorophenyl
- hydrate
- pharmaceutically acceptable
- purin
- Prior art date
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Classifications
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US82325806P | 2006-08-23 | 2006-08-23 | |
| US60/823,258 | 2006-08-23 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNA2007800309530A Division CN101506210A (zh) | 2006-08-23 | 2007-08-22 | 2-苯氧基嘧啶酮类似物 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN104292229A true CN104292229A (zh) | 2015-01-21 |
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ID=39107411
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNA2007800309530A Pending CN101506210A (zh) | 2006-08-23 | 2007-08-22 | 2-苯氧基嘧啶酮类似物 |
| CN201410468406.2A Pending CN104292229A (zh) | 2006-08-23 | 2007-08-22 | 2-苯氧基嘧啶酮类似物 |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
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| CNA2007800309530A Pending CN101506210A (zh) | 2006-08-23 | 2007-08-22 | 2-苯氧基嘧啶酮类似物 |
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| GB0509573D0 (en) * | 2005-05-11 | 2005-06-15 | Merck Sharp & Dohme | Therapeutic compounds |
| WO2008024438A2 (en) | 2006-08-23 | 2008-02-28 | Neurogen Corporation | 2-phenoxy pyrimidinone analogues |
| EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
| EP3417851B1 (en) | 2013-09-09 | 2020-07-22 | Peloton Therapeutics, Inc. | Aryl ethers and uses thereof |
| JP6667093B2 (ja) * | 2014-08-11 | 2020-03-18 | ハイドラ・バイオサイエンシーズ・リミテッド・ライアビリティ・カンパニーＨｙｄｒａ Ｂｉｏｓｃｉｅｎｃｅｓ， ＬＬＣ | ピリド［２，３−ｄ］ピリミジン−２，４（１Ｈ，３Ｈ）−ジオン誘導体 |
| US10155726B2 (en) | 2015-03-11 | 2018-12-18 | Peloton Therapeutics, Inc. | Substituted pyridines and uses thereof |
| WO2016144825A1 (en) | 2015-03-11 | 2016-09-15 | Peloton Therapeutics, Inc. | Aromatic compounds and uses thereof |
| WO2016145045A1 (en) | 2015-03-11 | 2016-09-15 | Peloton Therapeutics, Inc. | Compositions for use in treating glioblastoma |
| EP3267792A4 (en) | 2015-03-11 | 2018-09-26 | Peloton Therapeutics, Inc. | Compositions for use in treating pulmonary arterial hypertension |
| US10335388B2 (en) | 2015-04-17 | 2019-07-02 | Peloton Therapeutics, Inc. | Combination therapy of a HIF-2-alpha inhibitor and an immunotherapeutic agent and uses thereof |
| EP3908308A4 (en) * | 2019-01-08 | 2023-03-22 | Texas Tech University System | SMALL MOLECULE ANALOGUES OF PROTEIN E4ORF1 FOR THE TREATMENT AND PREVENTION OF METABOLIC DISORDERS |
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| WO2005049613A1 (en) * | 2003-11-14 | 2005-06-02 | Merck Sharp & Dohme Limited | Bicyclic pyrimidin-4-(3h)-ones and analogues and derivatives thereof which modulate the function of the vanilloid-1 receptor (vr1) |
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Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2005049613A1 (en) * | 2003-11-14 | 2005-06-02 | Merck Sharp & Dohme Limited | Bicyclic pyrimidin-4-(3h)-ones and analogues and derivatives thereof which modulate the function of the vanilloid-1 receptor (vr1) |
Also Published As
| Publication number | Publication date |
|---|---|
| SV2009003173A (es) | 2010-08-10 |
| US8759361B2 (en) | 2014-06-24 |
| NO20091182L (no) | 2009-05-14 |
| MX2009002066A (es) | 2009-03-06 |
| WO2008024438A2 (en) | 2008-02-28 |
| CA2660957A1 (en) | 2008-02-28 |
| EP2061794B1 (en) | 2012-12-05 |
| GT200900040A (es) | 2010-03-16 |
| EP2061794A4 (en) | 2010-09-08 |
| US8003656B2 (en) | 2011-08-23 |
| AU2007288203B2 (en) | 2013-01-17 |
| NI200900023A (es) | 2010-03-05 |
| CN101506210A (zh) | 2009-08-12 |
| KR20090043583A (ko) | 2009-05-06 |
| CO6150167A2 (es) | 2010-04-20 |
| ES2399928T3 (es) | 2013-04-04 |
| CR10675A (es) | 2009-04-17 |
| WO2008024438A3 (en) | 2008-11-27 |
| ZA200901163B (en) | 2010-08-25 |
| US20120208829A1 (en) | 2012-08-16 |
| TW200825089A (en) | 2008-06-16 |
| BRPI0716582A2 (pt) | 2013-10-08 |
| AU2007288203A1 (en) | 2008-02-28 |
| US20090069347A1 (en) | 2009-03-12 |
| EP2061794A2 (en) | 2009-05-27 |
| EA200900330A1 (ru) | 2009-08-28 |
| IL197043A0 (en) | 2009-11-18 |
| MA30720B1 (fr) | 2009-09-01 |
| JP5421108B2 (ja) | 2014-02-19 |
| JP2010502576A (ja) | 2010-01-28 |
| CA2660957C (en) | 2016-10-11 |
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