CN103717239B - 适合于吸入的氧化抗生物素蛋白的药物组合物 - Google Patents

适合于吸入的氧化抗生物素蛋白的药物组合物 Download PDF

Info

Publication number
CN103717239B
CN103717239B CN201280037217.9A CN201280037217A CN103717239B CN 103717239 B CN103717239 B CN 103717239B CN 201280037217 A CN201280037217 A CN 201280037217A CN 103717239 B CN103717239 B CN 103717239B
Authority
CN
China
Prior art keywords
biotinylation
oxavidin
lung
avidin
oxidized avidin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CN201280037217.9A
Other languages
English (en)
Chinese (zh)
Other versions
CN103717239A (zh
Inventor
R·德·桑德斯
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Alpha Sigma Co Ltd
Original Assignee
Sigma Tau Industrie Farmaceutiche Riunite SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sigma Tau Industrie Farmaceutiche Riunite SpA filed Critical Sigma Tau Industrie Farmaceutiche Riunite SpA
Publication of CN103717239A publication Critical patent/CN103717239A/zh
Application granted granted Critical
Publication of CN103717239B publication Critical patent/CN103717239B/zh
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0078Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a nebulizer such as a jet nebulizer, ultrasonic nebulizer, e.g. in the form of aqueous drug solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/1703Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/42Proteins; Polypeptides; Degradation products thereof; Derivatives thereof, e.g. albumin, gelatin or zein
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/62Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
    • A61K47/66Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid the modifying agent being a pre-targeting system involving a peptide or protein for targeting specific cells
    • A61K47/665Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid the modifying agent being a pre-targeting system involving a peptide or protein for targeting specific cells the pre-targeting system, clearing therapy or rescue therapy involving biotin-(strept) avidin systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K51/00Preparations containing radioactive substances for use in therapy or testing in vivo
    • A61K51/02Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04Organic compounds
    • A61K51/041Heterocyclic compounds
    • A61K51/044Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0453Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B82NANOTECHNOLOGY
    • B82YSPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pulmonology (AREA)
  • Molecular Biology (AREA)
  • Nanotechnology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Optics & Photonics (AREA)
  • Immunology (AREA)
  • Dispersion Chemistry (AREA)
  • Otolaryngology (AREA)
  • Physics & Mathematics (AREA)
  • Marine Sciences & Fisheries (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • General Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Biotechnology (AREA)
  • Inorganic Chemistry (AREA)
  • Medical Informatics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Cell Biology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CN201280037217.9A 2011-08-02 2012-07-25 适合于吸入的氧化抗生物素蛋白的药物组合物 Active CN103717239B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11006338 2011-08-02
EP11006338.5 2011-08-02
PCT/EP2012/064576 WO2013017494A1 (en) 2011-08-02 2012-07-25 Pharmaceutical composition of oxidised avidin suitable for inhalation

Publications (2)

Publication Number Publication Date
CN103717239A CN103717239A (zh) 2014-04-09
CN103717239B true CN103717239B (zh) 2017-08-01

Family

ID=46581966

Family Applications (1)

Application Number Title Priority Date Filing Date
CN201280037217.9A Active CN103717239B (zh) 2011-08-02 2012-07-25 适合于吸入的氧化抗生物素蛋白的药物组合物

Country Status (19)

Country Link
US (1) US9872831B2 (enExample)
EP (1) EP2739314B1 (enExample)
JP (1) JP6019118B2 (enExample)
KR (1) KR101966630B1 (enExample)
CN (1) CN103717239B (enExample)
AU (1) AU2012292229B2 (enExample)
BR (1) BR112014002593B1 (enExample)
CA (1) CA2842276C (enExample)
DK (1) DK2739314T3 (enExample)
EA (1) EA026453B1 (enExample)
ES (1) ES2729549T3 (enExample)
IL (1) IL230597A0 (enExample)
MX (1) MX355177B (enExample)
PH (1) PH12014500193A1 (enExample)
PL (1) PL2739314T3 (enExample)
PT (1) PT2739314T (enExample)
UA (1) UA114482C2 (enExample)
WO (1) WO2013017494A1 (enExample)
ZA (1) ZA201401921B (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2941243A4 (en) 2013-01-04 2016-09-14 Massachusetts Inst Technology SURFACE BINDING IN THE ADMINISTRATION OF A MEDICAMENT ON NANOPARTICLE BASE IN A TISSUE
EP3458097A4 (en) * 2016-05-19 2020-01-08 University of Miami TARGETED DELIVERY OF THERAPEUTIC AGENTS AND IMAGING REAGENTS TO CANCER PANCREAS CELLS

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2106806A1 (en) * 2008-03-31 2009-10-07 Fraunhofer-Gesellschaft zur Förderung der Angewandten Forschung e.V. Nanoparticles for targeted delivery of active agents to the lung
CN101772353A (zh) * 2007-08-02 2010-07-07 希格马托制药工业公司 在受治疗组织中展现高停留时间的氧化的抗生物素蛋白

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5384128A (en) * 1993-03-02 1995-01-24 University Of Alabama Research Foundation Method of and compounds for treatment for cystic fibrosis
JPH09501418A (ja) 1993-07-19 1997-02-10 アムジエン・インコーポレーテツド エアゾル化タンパク質の安定化
DE69830305T2 (de) * 1997-02-20 2006-02-02 Dime, David S., Toronto Ortsspezifische arzneimittel verabreichung
HK1042234A1 (zh) * 1999-04-13 2002-08-09 Nektar Therapeutics 向肺部施加乾粉配方以治疗不育症
US7001994B2 (en) * 2001-01-18 2006-02-21 Genzyme Corporation Methods for introducing mannose 6-phosphate and other oligosaccharides onto glycoproteins
ITRM20010079A1 (it) 2001-02-16 2002-08-16 Sigma Tau Ind Farmaceuti Amminoderivati della biotina e loro coniugati con chelanti macrociclici.
ITRM20030196A1 (it) * 2003-04-24 2004-10-25 Sigma Tau Ind Farmaceuti Uso di reagenti per la preparazione di un medicamento
EP2311793A1 (en) * 2004-12-17 2011-04-20 Cipla Ltd. Crystalline levosalbutamol sulphate (Form II)
GB0602778D0 (en) * 2006-02-10 2006-03-22 Glaxo Group Ltd Novel compound
TW201031436A (en) * 2009-02-16 2010-09-01 Univ Nat Taiwan Pharmaceutical composition for inhalation delivery and fabrication method thereof

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101772353A (zh) * 2007-08-02 2010-07-07 希格马托制药工业公司 在受治疗组织中展现高停留时间的氧化的抗生物素蛋白
EP2106806A1 (en) * 2008-03-31 2009-10-07 Fraunhofer-Gesellschaft zur Förderung der Angewandten Forschung e.V. Nanoparticles for targeted delivery of active agents to the lung

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
Pretargeted Radioimmunotherapy of Cancer: Progress Step by Step;Otto C. Boerman et al.;《The Journal of Nuclear Medicine》;20030331;第44卷(第3期);第400-411页 *

Also Published As

Publication number Publication date
EP2739314A1 (en) 2014-06-11
ES2729549T3 (es) 2019-11-04
PL2739314T3 (pl) 2019-09-30
EA026453B1 (ru) 2017-04-28
MX355177B (es) 2018-04-09
CN103717239A (zh) 2014-04-09
BR112014002593A2 (pt) 2017-03-01
ZA201401921B (en) 2015-05-27
PH12014500193A1 (en) 2014-03-24
US20140134106A1 (en) 2014-05-15
CA2842276C (en) 2020-11-24
AU2012292229A1 (en) 2014-02-13
JP6019118B2 (ja) 2016-11-02
US9872831B2 (en) 2018-01-23
CA2842276A1 (en) 2013-02-07
KR20140047668A (ko) 2014-04-22
NZ620202A (en) 2016-05-27
EP2739314B1 (en) 2019-05-22
DK2739314T3 (da) 2019-06-24
KR101966630B1 (ko) 2019-04-09
IL230597A0 (en) 2014-03-31
MX2014001176A (es) 2014-07-14
EA201490401A1 (ru) 2014-05-30
WO2013017494A1 (en) 2013-02-07
BR112014002593B1 (pt) 2022-11-29
UA114482C2 (uk) 2017-06-26
PT2739314T (pt) 2019-06-21
AU2012292229B2 (en) 2017-08-03
JP2014521675A (ja) 2014-08-28

Similar Documents

Publication Publication Date Title
Li et al. Nanomedicine embraces cancer radio-immunotherapy: mechanism, design, recent advances, and clinical translation
CN111989138B (zh) 人源化抗前列腺特异性膜抗原(psma)抗体药物缀合物
Groneberg et al. Molecular mechanisms of pulmonary peptidomimetic drug and peptide transport
US20070231408A1 (en) Colloidal metal compositions and methods
US20110064652A1 (en) Nanoparticles for targeted delivery of active agents to the lung
CN111954531A (zh) α聚谷氨酸化培美曲塞及其用途
CN111954529A (zh) α聚谷氨酸化氨甲蝶呤及其用途
CN111936146A (zh) α聚谷氨酸化四氢叶酸及其用途
Maillet et al. The airways, a novel route for delivering monoclonal antibodies to treat lung tumors
RS61961B1 (sr) Morfogenetski proteini kosti
CN103717239B (zh) 适合于吸入的氧化抗生物素蛋白的药物组合物
Zarogoulidis et al. 2-diethylaminoethyl-dextran methyl methacrylate copolymer nonviral vector: still a long way toward the safety of aerosol gene therapy
CN118766874B (zh) 一种吸入式制剂、迭代优化流程及其应用
JP2001512831A (ja) 生物学的薬剤組成物を同定する方法
JPWO2020071448A1 (ja) 吸入粉末剤、その評価方法及びその用途
HK1194002A (en) Pharmaceutical composition of oxidised avidin suitable for inhalation
HK1194002B (en) Pharmaceutical composition of oxidised avidin suitable for inhalation
NZ620202B2 (en) Pharmaceutical composition of oxidised avidin suitable for inhalation
US10912791B2 (en) Compositions comprising antisense-encoded erythropoietin receptor and use thereof
Siddhanta et al. Inhalable perfluorocarbon RNA nanocapsules overcome biological barriers to treat lung metastases
US20180177724A1 (en) Site-targeted nano-liposomal nitroglycerin therapeutics
Li Development of an Aerosol-Based Immunotherapy for Non-Small Cell Lung Cancer
Huayamares et al. Current Research in Biotechnology
Gaber et al. In vivo pharmacodynamics of lactoferrin-coupled lipid nanocarriers for lung carcinoma: intravenous versus powder for inhalation
Zarogoulidis et al. Airway local endoscopic pharmacological treatment; current applications and future concepts

Legal Events

Date Code Title Description
C06 Publication
PB01 Publication
C10 Entry into substantive examination
SE01 Entry into force of request for substantive examination
REG Reference to a national code

Ref country code: HK

Ref legal event code: DE

Ref document number: 1194002

Country of ref document: HK

GR01 Patent grant
GR01 Patent grant
TR01 Transfer of patent right
TR01 Transfer of patent right

Effective date of registration: 20180118

Address after: Milan Italy

Patentee after: Alpha Sigmar joint-stock company

Address before: Rome Italy

Patentee before: Sigma-Tau Industrie Farmaceutiche Riunite S. P. A.

CP03 Change of name, title or address
CP03 Change of name, title or address

Address after: Bologna, Italy

Patentee after: Alpha sigma Co., Ltd

Address before: Milan Italy

Patentee before: Alpha Sigmar JSC