CN103327981A - 用于治疗视网膜疾病的方法 - Google Patents
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- CN103327981A CN103327981A CN2011800652550A CN201180065255A CN103327981A CN 103327981 A CN103327981 A CN 103327981A CN 2011800652550 A CN2011800652550 A CN 2011800652550A CN 201180065255 A CN201180065255 A CN 201180065255A CN 103327981 A CN103327981 A CN 103327981A
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
- A61P39/06—Free radical scavengers or antioxidants
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- Ophthalmology & Optometry (AREA)
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| US41966010P | 2010-12-03 | 2010-12-03 | |
| US61/419,660 | 2010-12-03 | ||
| PCT/US2011/061370 WO2012074788A1 (en) | 2010-12-03 | 2011-11-18 | Methods for treating diseases of the retina |
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| CN103327981A true CN103327981A (zh) | 2013-09-25 |
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| CN2011800652550A Pending CN103327981A (zh) | 2010-12-03 | 2011-11-18 | 用于治疗视网膜疾病的方法 |
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| US (2) | US9018202B2 (https=) |
| EP (1) | EP2646034A1 (https=) |
| JP (1) | JP2013544838A (https=) |
| KR (1) | KR20130122958A (https=) |
| CN (1) | CN103327981A (https=) |
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| CA (1) | CA2819616A1 (https=) |
| RU (1) | RU2013129748A (https=) |
| WO (1) | WO2012074788A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10752593B2 (en) | 2018-12-28 | 2020-08-25 | Endogena Therapeutics, Inc. | Compounds for use as therapeutically active substances in the treatment of retinal diseases |
| JP6864327B2 (ja) | 2017-07-06 | 2021-04-28 | 山田 健一 | 脂質過酸化誘発性疾患の治療薬およびそのスクリーニング方法 |
| US10807973B2 (en) | 2018-12-28 | 2020-10-20 | Endogena Therapeutics, Inc. | Compounds for use as therapeutically active substances in the treatment of retinal diseases |
| EP3919052A4 (en) * | 2019-01-09 | 2022-10-05 | Fuso Pharmaceutical Industries, Ltd. | Pharmaceutical composition for intraocular or oral administration for treatment of retinal diseases |
| US20250170143A1 (en) * | 2022-04-14 | 2025-05-29 | Mayo Foundation For Medical Education And Research | Methods of treating ocular fibrotic pathologies |
Citations (4)
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| US5744468A (en) * | 1996-10-23 | 1998-04-28 | Tong-Ho Lin | Hypotensive intraocular pressure activity of clozapine and sulpiride |
| WO2003070249A1 (de) * | 2002-02-19 | 2003-08-28 | Nowak Goetz | Kombination von trapidil mit serotoninantagonisten wie cyproheptadin oder pizotifen zur hemmung der angiogenese |
| WO2004103263A2 (en) * | 2003-05-22 | 2004-12-02 | Yeda Research And Development Co. Ltd. | Dopamine and agonists and antagonists thereof for treatment of neurodegenerative diseases |
| CN101437478A (zh) * | 2004-10-04 | 2009-05-20 | Qlt美国有限公司 | 聚合送递制剂的眼部送递 |
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| HK1004520A1 (en) | 1992-05-13 | 1998-11-27 | Novartis Ag | Ophthalmic compositions containing a cyclosporin |
| US5474979A (en) | 1994-05-17 | 1995-12-12 | Allergan, Inc. | Nonirritating emulsions for sensitive tissue |
| US5631250A (en) | 1995-03-24 | 1997-05-20 | Eli Lilly And Company | Process and solvate of 2-methyl-thieno-benzodiazepine |
| JPH10175865A (ja) * | 1996-12-11 | 1998-06-30 | Towa Rin | 抗眼圧活性製剤 |
| US7160898B2 (en) * | 2001-12-14 | 2007-01-09 | Board Of Trustees Of The University Of Illinois | Pharmacological treatment for sleep apnea |
| JP2002530340A (ja) * | 1998-11-23 | 2002-09-17 | セプラコール， インク． | オランザピン−ｎ−オキサイドを含む医薬組成物 |
| JP2006515628A (ja) * | 2003-01-23 | 2006-06-01 | アカディア ファーマシューティカルズ，インコーポレーテッド | ヒト神経精神疾患を処置するためのｎ−デスメチルクロザピンの使用 |
| US20050059583A1 (en) | 2003-09-15 | 2005-03-17 | Allergan, Inc. | Methods of providing therapeutic effects using cyclosporin components |
| US20050277584A1 (en) | 2004-06-09 | 2005-12-15 | Allergan, Inc. | Pharmaceutical compositions comprising cyclosporins |
| US20060035887A1 (en) | 2004-07-02 | 2006-02-16 | Dr. Reddy's Laboratories Limited | Process for preparing olanzapine |
| AU2005271513A1 (en) * | 2004-08-05 | 2006-02-16 | Acadia Pharmaceuticals Inc. | Use of N-desmethylclozapine to treat human neuropsychiatric disease |
| MX2007003789A (es) | 2004-10-04 | 2007-07-20 | Qlt Usa Inc | Suministro ocular de formulaciones polimericas para suministro. |
| US7297679B2 (en) | 2005-07-13 | 2007-11-20 | Allergan, Inc. | Cyclosporin compositions |
| US20070015691A1 (en) | 2005-07-13 | 2007-01-18 | Allergan, Inc. | Cyclosporin compositions |
| WO2008111497A1 (ja) * | 2007-03-08 | 2008-09-18 | Santen Pharmaceutical Co., Ltd. | トリテルペノイドを有効成分として含有する酸化ストレスが関連する眼疾患の予防又は治療剤 |
| CN101711236B (zh) * | 2007-04-12 | 2012-10-31 | Nsab神经研究瑞典公司分公司 | 表现出改善的心血管副作用特性的多巴胺受体稳定剂/调节剂的n-氧化物和/或二-n-氧化物衍生物 |
-
2011
- 2011-11-16 US US13/298,028 patent/US9018202B2/en active Active
- 2011-11-18 WO PCT/US2011/061370 patent/WO2012074788A1/en not_active Ceased
- 2011-11-18 CA CA 2819616 patent/CA2819616A1/en not_active Abandoned
- 2011-11-18 JP JP2013542043A patent/JP2013544838A/ja active Pending
- 2011-11-18 KR KR20137017036A patent/KR20130122958A/ko not_active Ceased
- 2011-11-18 BR BR112013013636A patent/BR112013013636A2/pt not_active IP Right Cessation
- 2011-11-18 EP EP11810917.2A patent/EP2646034A1/en not_active Withdrawn
- 2011-11-18 RU RU2013129748/15A patent/RU2013129748A/ru not_active Application Discontinuation
- 2011-11-18 CN CN2011800652550A patent/CN103327981A/zh active Pending
- 2011-11-18 AU AU2011336976A patent/AU2011336976A1/en not_active Abandoned
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- 2015-04-27 US US14/696,789 patent/US9561234B2/en not_active Expired - Fee Related
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| US5744468A (en) * | 1996-10-23 | 1998-04-28 | Tong-Ho Lin | Hypotensive intraocular pressure activity of clozapine and sulpiride |
| WO2003070249A1 (de) * | 2002-02-19 | 2003-08-28 | Nowak Goetz | Kombination von trapidil mit serotoninantagonisten wie cyproheptadin oder pizotifen zur hemmung der angiogenese |
| WO2004103263A2 (en) * | 2003-05-22 | 2004-12-02 | Yeda Research And Development Co. Ltd. | Dopamine and agonists and antagonists thereof for treatment of neurodegenerative diseases |
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Also Published As
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| US9018202B2 (en) | 2015-04-28 |
| CA2819616A1 (en) | 2012-06-07 |
| AU2011336976A1 (en) | 2013-07-11 |
| JP2013544838A (ja) | 2013-12-19 |
| US9561234B2 (en) | 2017-02-07 |
| BR112013013636A2 (pt) | 2016-11-08 |
| EP2646034A1 (en) | 2013-10-09 |
| RU2013129748A (ru) | 2015-01-10 |
| WO2012074788A1 (en) | 2012-06-07 |
| KR20130122958A (ko) | 2013-11-11 |
| US20150290215A1 (en) | 2015-10-15 |
| US20120142675A1 (en) | 2012-06-07 |
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