CN103142504A - 一种甘糖酯缓释颗粒及其制备方法 - Google Patents
一种甘糖酯缓释颗粒及其制备方法 Download PDFInfo
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- CN103142504A CN103142504A CN2013100933273A CN201310093327A CN103142504A CN 103142504 A CN103142504 A CN 103142504A CN 2013100933273 A CN2013100933273 A CN 2013100933273A CN 201310093327 A CN201310093327 A CN 201310093327A CN 103142504 A CN103142504 A CN 103142504A
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1h | 2h | 4h | 8h | 12h | 16h | 20h | 24h |
实施例1 | 15.8% | 29.9% | 46.7% | 61.2% | 75.4% | 88.9% | 100.0% | |
实施例2 | 17.1% | 35.6% | 54.8% | 70.7% | 85.0% | 100.1% | ||
实施例3 | 17.8% | 34.2% | 55.3% | 73.6% | 90.0% | 100.0% | ||
实施例4 | 19.5% | 37.8% | 57.4% | 75.5% | 91.4% | 100.0% |
实施例5 | 实施例6 | 实施例7 | ||
甘糖酯 | 110g | 110g | 110g | |
填充剂 | 微晶纤维素 | 590g | 590g | 590g |
缓释材料 | 羟丙纤维素 | 208.3g | 200g | 187.5g |
增塑剂 | 乙酰柠檬酸三丁酯 | 50g | 50g | 50g |
致孔剂 | 乳糖 | 41.7g | 50g | 62.5g |
抗粘剂 | 滑石粉 | 100g | 100g | 100g |
1h | 2h | 4h | 8h | 12h | 16h | 20h | 24h | |
实施例5 | 18.6% | 37.2% | 56.8% | 72.5% | 84.6% | 93.3% | 100.0% | |
实施例6 | 14.2% | 28.8% | 43.6% | 58.4% | 71.1% | 82.9% | 91.5% | 100.1% |
实施例7 | 16.8% | 33.2% | 48.7% | 63.6% | 79.0% | 91.1% | 100.0% |
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CN201310093327.3A CN103142504B (zh) | 2013-03-21 | 2013-03-21 | 一种甘糖酯缓释颗粒及其制备方法 |
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CN201310093327.3A CN103142504B (zh) | 2013-03-21 | 2013-03-21 | 一种甘糖酯缓释颗粒及其制备方法 |
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CN103142504A true CN103142504A (zh) | 2013-06-12 |
CN103142504B CN103142504B (zh) | 2014-07-23 |
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Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN105434364A (zh) * | 2015-12-07 | 2016-03-30 | 青岛正大海尔制药有限公司 | 一种托匹司他缓释颗粒及其制备方法 |
CN106075610A (zh) * | 2016-08-12 | 2016-11-09 | 陈旭东 | 一种介入穿刺用止血粒子及其制备方法 |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN101006989A (zh) * | 2005-09-26 | 2007-08-01 | 刘凤鸣 | 藻酸双酯钠的缓释制剂 |
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Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
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CN101006989A (zh) * | 2005-09-26 | 2007-08-01 | 刘凤鸣 | 藻酸双酯钠的缓释制剂 |
Non-Patent Citations (2)
Title |
---|
李红兵: "海藻酸作为活性药物和新型药用敷料的开发", 《海洋技术》 * |
陈娥功: "甘糖酯薄膜衣片的制备及稳定性试验", 《中国海洋药物》 * |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN105434364A (zh) * | 2015-12-07 | 2016-03-30 | 青岛正大海尔制药有限公司 | 一种托匹司他缓释颗粒及其制备方法 |
CN105434364B (zh) * | 2015-12-07 | 2018-07-03 | 青岛正大海尔制药有限公司 | 一种托匹司他缓释颗粒及其制备方法 |
CN106075610A (zh) * | 2016-08-12 | 2016-11-09 | 陈旭东 | 一种介入穿刺用止血粒子及其制备方法 |
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Address after: 266103 Qingdao economic and Technological Development Zone, unity Road, No. 3601, Shandong Applicant after: Qingdao Zhengda Haier Pharmaceutical Co., Ltd. Address before: 266103 Haier Road, Shandong, Qingdao, No. 1 Applicant before: Qingdao Zhengda Haier Pharmaceutical Co., Ltd. |
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Address after: 266103 3601 Tuen Jie Road, Qingdao economic and Technological Development Zone, Shandong Patentee after: Zhengda Pharmaceutical (Qingdao) Co., Ltd. Address before: 266103 3601 Tuen Jie Road, Qingdao economic and Technological Development Zone, Shandong Patentee before: Qingdao Zhengda Haier Pharmaceutical Co., Ltd. |
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