CN101296731A - 作为钾通道开启剂的苯并吡喃和吡喃并吡啶衍生物 - Google Patents

作为钾通道开启剂的苯并吡喃和吡喃并吡啶衍生物 Download PDF

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Publication number
CN101296731A
CN101296731A CNA2006800401602A CN200680040160A CN101296731A CN 101296731 A CN101296731 A CN 101296731A CN A2006800401602 A CNA2006800401602 A CN A2006800401602A CN 200680040160 A CN200680040160 A CN 200680040160A CN 101296731 A CN101296731 A CN 101296731A
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alkyl
amino
halogen
alkoxy
phenyl
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Chinese (zh)
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X·张
X·李
Z·隋
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Janssen Pharmaceutica NV
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Janssen Pharmaceutica NV
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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
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    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
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    • C07D311/62—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4 with aryl radicals attached in position 2 with oxygen atoms directly attached in position 3, e.g. anthocyanidins
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    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
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  • Chemical & Material Sciences (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pulmonology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Otolaryngology (AREA)
  • Vascular Medicine (AREA)
  • Dermatology (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrane Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CNA2006800401602A 2005-09-01 2006-08-30 作为钾通道开启剂的苯并吡喃和吡喃并吡啶衍生物 Pending CN101296731A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US71355005P 2005-09-01 2005-09-01
US60/713,550 2005-09-01

Publications (1)

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CN101296731A true CN101296731A (zh) 2008-10-29

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CNA2006800401602A Pending CN101296731A (zh) 2005-09-01 2006-08-30 作为钾通道开启剂的苯并吡喃和吡喃并吡啶衍生物

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Country Link
US (1) US7812183B2 (enExample)
EP (1) EP1940516A2 (enExample)
JP (1) JP2009509927A (enExample)
CN (1) CN101296731A (enExample)
AU (1) AU2006284860A1 (enExample)
CA (1) CA2620846A1 (enExample)
WO (1) WO2007027780A2 (enExample)

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Publication number Priority date Publication date Assignee Title
EP1937669B9 (en) * 2005-09-01 2012-07-18 Janssen Pharmaceutica NV Novel benzopyran derivatives as potassium channel openers
CN101296731A (zh) * 2005-09-01 2008-10-29 詹森药业有限公司 作为钾通道开启剂的苯并吡喃和吡喃并吡啶衍生物
WO2009022633A1 (ja) * 2007-08-10 2009-02-19 Astellas Pharma Inc. 二環式アシルグアニジン誘導体
EP2817877A4 (en) 2012-02-22 2016-01-27 Int Electronic Machines Corp ENERGY
JP6409004B2 (ja) * 2013-01-28 2018-10-17 ハー・ルンドベック・アクチエゼルスカベット ソルチリン阻害剤としてのｎ置換された５置換フタルアミド酸
US9573921B2 (en) * 2013-09-30 2017-02-21 Polfarmex S.A. Substituted N, N-dimethylaminoalkyl ethers of isoflavanone oximes as H1-receptor antagonists
JP6996032B1 (ja) * 2020-04-24 2022-01-17 大日本住友製薬株式会社 ２－ヘテロアリールアミノキナゾリノン誘導体

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CN101296731A (zh) * 2005-09-01 2008-10-29 詹森药业有限公司 作为钾通道开启剂的苯并吡喃和吡喃并吡啶衍生物
EP1937669B9 (en) 2005-09-01 2012-07-18 Janssen Pharmaceutica NV Novel benzopyran derivatives as potassium channel openers

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EP1940516A2 (en) 2008-07-09
US20070072832A1 (en) 2007-03-29
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