CN101180071A - 抑制蛋白酶体的组合物 - Google Patents

抑制蛋白酶体的组合物 Download PDF

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Publication number
CN101180071A
CN101180071A CNA2005800478775A CN200580047877A CN101180071A CN 101180071 A CN101180071 A CN 101180071A CN A2005800478775 A CNA2005800478775 A CN A2005800478775A CN 200580047877 A CN200580047877 A CN 200580047877A CN 101180071 A CN101180071 A CN 101180071A
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China
Prior art keywords
alkyl
hydrogen
aryl
pharmaceutical composition
independently selected
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Pending
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CNA2005800478775A
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English (en)
Chinese (zh)
Inventor
E·R·路易斯
M·N·侯
F·N·丰塞卡
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Onyx Pharmaceuticals Inc
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Proteolix Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36143200&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CN101180071(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Proteolix Inc filed Critical Proteolix Inc
Publication of CN101180071A publication Critical patent/CN101180071A/zh
Pending legal-status Critical Current

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CNA2005800478775A 2004-12-07 2005-12-07 抑制蛋白酶体的组合物 Pending CN101180071A (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US63436604P 2004-12-07 2004-12-07
US60/634,366 2004-12-07
US65593005P 2005-02-23 2005-02-23
US60/655,930 2005-02-23

Related Child Applications (1)

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CN2012103747120A Division CN102847136A (zh) 2004-12-07 2005-12-07 抑制蛋白酶体的组合物

Publications (1)

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CN101180071A true CN101180071A (zh) 2008-05-14

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CNA2005800478775A Pending CN101180071A (zh) 2004-12-07 2005-12-07 抑制蛋白酶体的组合物
CN2012103747120A Pending CN102847136A (zh) 2004-12-07 2005-12-07 抑制蛋白酶体的组合物

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CN2012103747120A Pending CN102847136A (zh) 2004-12-07 2005-12-07 抑制蛋白酶体的组合物

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Country Link
US (1) US7737112B2 (https=)
EP (3) EP2261236B1 (https=)
JP (1) JP4990155B2 (https=)
KR (1) KR101299821B1 (https=)
CN (2) CN101180071A (https=)
AT (1) ATE499109T1 (https=)
AU (1) AU2005313975B2 (https=)
CA (1) CA2589921C (https=)
CY (1) CY1111489T1 (https=)
DE (1) DE602005026556D1 (https=)
DK (1) DK1819353T3 (https=)
ES (2) ES2408216T3 (https=)
HU (1) HUE027850T2 (https=)
IL (1) IL183607A (https=)
PL (3) PL2260835T3 (https=)
PT (3) PT2260835E (https=)
WO (1) WO2006063154A1 (https=)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103570806A (zh) * 2012-07-26 2014-02-12 圣特莱国际公司 多肽环氧酮化合物
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CN104411334A (zh) * 2012-05-08 2015-03-11 欧尼斯治疗公司 用于配制肽蛋白酶体抑制剂的环糊精络合法
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CN103570806A (zh) * 2012-07-26 2014-02-12 圣特莱国际公司 多肽环氧酮化合物
CN109096370A (zh) * 2012-07-26 2018-12-28 圣特莱国际公司 多肽环氧酮化合物
CN109180780A (zh) * 2012-07-26 2019-01-11 圣特莱国际公司 多肽环氧酮化合物
CN103570806B (zh) * 2012-07-26 2020-04-07 圣特莱国际公司 多肽环氧酮化合物
CN109180780B (zh) * 2012-07-26 2022-03-18 圣特莱国际公司 多肽环氧酮化合物
CN109096370B (zh) * 2012-07-26 2022-03-18 圣特莱国际公司 多肽环氧酮化合物
CN104797591A (zh) * 2012-08-14 2015-07-22 弗洛伊诺制药公司 氟化环氧酮系化合物及其作为蛋白酶体抑制剂的用途
CN109415353A (zh) * 2016-05-24 2019-03-01 美国安进公司 聚乙二醇化卡非佐米化合物
CN109415353B (zh) * 2016-05-24 2023-01-10 美国安进公司 聚乙二醇化卡非佐米化合物
WO2025092827A1 (zh) * 2023-10-30 2025-05-08 上海汇伦医药股份有限公司 一种环氧类化合物及其应用

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