CY1111489T1 - Ενωσεις για την αναστολη του πρωτεασωματος - Google Patents

Ενωσεις για την αναστολη του πρωτεασωματος

Info

Publication number
CY1111489T1
CY1111489T1 CY20111100410T CY111100410T CY1111489T1 CY 1111489 T1 CY1111489 T1 CY 1111489T1 CY 20111100410 T CY20111100410 T CY 20111100410T CY 111100410 T CY111100410 T CY 111100410T CY 1111489 T1 CY1111489 T1 CY 1111489T1
Authority
CY
Cyprus
Prior art keywords
compositions
suspension
compounds
proteasome inhibitors
cyclodextrin
Prior art date
Application number
CY20111100410T
Other languages
Greek (el)
English (en)
Inventor
Evan R Lewis
Mark Nguyen Ho
Fabiana N Fonseca
Original Assignee
Proteolix, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36143200&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1111489(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Proteolix, Inc. filed Critical Proteolix, Inc.
Publication of CY1111489T1 publication Critical patent/CY1111489T1/el

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    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/336Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having three-membered rings, e.g. oxirane, fumagillin
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/396Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having three-membered rings, e.g. aziridine
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0802Tripeptides with the first amino acid being neutral
    • C07K5/0812Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Organic Chemistry (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
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  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Virology (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Inorganic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Psychology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Hospice & Palliative Care (AREA)
CY20111100410T 2004-12-07 2011-04-21 Ενωσεις για την αναστολη του πρωτεασωματος CY1111489T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US63436604P 2004-12-07 2004-12-07
US65593005P 2005-02-23 2005-02-23
EP05853385A EP1819353B1 (en) 2004-12-07 2005-12-07 Composition for proteasome inhibition

Publications (1)

Publication Number Publication Date
CY1111489T1 true CY1111489T1 (el) 2014-02-12

Family

ID=36143200

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20111100410T CY1111489T1 (el) 2004-12-07 2011-04-21 Ενωσεις για την αναστολη του πρωτεασωματος

Country Status (17)

Country Link
US (1) US7737112B2 (https=)
EP (3) EP2261236B1 (https=)
JP (1) JP4990155B2 (https=)
KR (1) KR101299821B1 (https=)
CN (2) CN101180071A (https=)
AT (1) ATE499109T1 (https=)
AU (1) AU2005313975B2 (https=)
CA (1) CA2589921C (https=)
CY (1) CY1111489T1 (https=)
DE (1) DE602005026556D1 (https=)
DK (1) DK1819353T3 (https=)
ES (2) ES2408216T3 (https=)
HU (1) HUE027850T2 (https=)
IL (1) IL183607A (https=)
PL (3) PL2260835T3 (https=)
PT (3) PT2260835E (https=)
WO (1) WO2006063154A1 (https=)

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US8198270B2 (en) * 2004-04-15 2012-06-12 Onyx Therapeutics, Inc. Compounds for proteasome enzyme inhibition
US8129346B2 (en) 2004-04-15 2012-03-06 Onyx Therapeutics, Inc. Compounds for enzyme inhibition
EP2030981B1 (en) * 2004-05-10 2014-07-09 Onyx Therapeutics, Inc. Compounds for proteasome enzyme inhibition
US9034846B2 (en) * 2004-10-10 2015-05-19 Universite De Liege Use of cyclodextrin for treatment and prevention of bronchial inflammatory diseases
MY171061A (en) * 2005-11-09 2019-09-24 Onyx Therapeutics Inc Compounds for enzyme inhibition
CA2657213C (en) 2006-06-19 2017-01-03 Proteolix, Inc. Peptide epoxyketones for proteasome inhibition
KR20170125413A (ko) 2007-10-04 2017-11-14 오닉스 세라퓨틱스, 인크. 결정형 펩티드 에폭시 케톤 프로테아제 저해제 및 아미노산 케토-에폭시드의 합성
US7635773B2 (en) 2008-04-28 2009-12-22 Cydex Pharmaceuticals, Inc. Sulfoalkyl ether cyclodextrin compositions
EA201170527A1 (ru) * 2008-10-01 2011-10-31 Др. Редди'С Лабораторис Лтд. Фармацевтические композиции, включающие соединения бороновой кислоты
EP3090737A1 (en) * 2008-10-21 2016-11-09 Onyx Therapeutics, Inc. Combination therapy with peptide epoxyketones
TWI504598B (zh) 2009-03-20 2015-10-21 Onyx Therapeutics Inc 結晶性三肽環氧酮蛋白酶抑制劑
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