CL2023001325A1 - Compuestos y su uso en el tratamiento de trastornos mediados por receptores de taquicinina - Google Patents

Compuestos y su uso en el tratamiento de trastornos mediados por receptores de taquicinina

Info

Publication number
CL2023001325A1
CL2023001325A1 CL2023001325A CL2023001325A CL2023001325A1 CL 2023001325 A1 CL2023001325 A1 CL 2023001325A1 CL 2023001325 A CL2023001325 A CL 2023001325A CL 2023001325 A CL2023001325 A CL 2023001325A CL 2023001325 A1 CL2023001325 A1 CL 2023001325A1
Authority
CL
Chile
Prior art keywords
compounds
treatment
disorders mediated
tachykinin receptors
tachykinin
Prior art date
Application number
CL2023001325A
Other languages
English (en)
Spanish (es)
Inventor
Bernt Fredrik Gustafsson Magnus
Madsen Johnny
Mulvad Olivia
Frederik Johan Hogendorf Wouter
Bondo HANSEN Jakob
Original Assignee
Embark Biotech Aps
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Embark Biotech Aps filed Critical Embark Biotech Aps
Publication of CL2023001325A1 publication Critical patent/CL2023001325A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/22Tachykinins, e.g. Eledoisins, Substance P; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/542Carboxylic acids, e.g. a fatty acid or an amino acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2319/00Fusion polypeptide

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Obesity (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Emergency Medicine (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
CL2023001325A 2020-11-09 2023-05-08 Compuestos y su uso en el tratamiento de trastornos mediados por receptores de taquicinina CL2023001325A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP20206509 2020-11-09

Publications (1)

Publication Number Publication Date
CL2023001325A1 true CL2023001325A1 (es) 2023-12-15

Family

ID=73198203

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2023001325A CL2023001325A1 (es) 2020-11-09 2023-05-08 Compuestos y su uso en el tratamiento de trastornos mediados por receptores de taquicinina

Country Status (13)

Country Link
US (1) US20230406883A1 (https=)
EP (1) EP4240749A1 (https=)
JP (1) JP2023551122A (https=)
KR (1) KR20230106616A (https=)
CN (1) CN116745310A (https=)
AU (1) AU2021374843A1 (https=)
CA (1) CA3197916A1 (https=)
CL (1) CL2023001325A1 (https=)
CO (1) CO2023007404A2 (https=)
IL (1) IL302745A (https=)
MX (1) MX2023005408A (https=)
PE (1) PE20231952A1 (https=)
WO (1) WO2022096736A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA3204051A1 (en) 2021-01-20 2022-07-28 Brian Lian Compositions and methods for the treatment of metabolic and liver disorders
JP7642830B2 (ja) 2021-09-15 2025-03-10 バイキング・セラピューティクス・インコーポレイテッド 代謝及び肝臓障害の処置のための組成物及び方法
WO2023118263A1 (en) * 2021-12-21 2023-06-29 Embark Biotech Aps Agonists for treatment of eating disorder
CN117384258B (zh) * 2023-10-12 2024-07-26 湖南中晟全肽生物科技股份有限公司 一种神经激肽受体2(nk2r)激动剂及其应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2427475T3 (pl) * 2009-05-08 2021-07-19 Techfields Biochem Co., Ltd. Kompozycje proleku o wysokim przenikaniu peptydów i związków powiązanych z peptydami
CN105722526B (zh) * 2013-11-15 2020-12-08 诺和诺德股份有限公司 选择性pyy化合物及其用途
TWI694082B (zh) * 2015-06-12 2020-05-21 丹麥商諾佛 儂迪克股份有限公司 選擇性pyy化合物及其用途
WO2019059963A1 (en) * 2017-09-21 2019-03-28 Dignify Therapeutics, Llc COMPOSITIONS FOR INDUCING MICTION AND DEFECATION
US11633459B2 (en) * 2018-05-04 2023-04-25 Novo Nordisk A/S GIP derivatives and uses thereof
MX2022004566A (es) * 2019-10-17 2022-07-21 Univ Copenhagen Agonista del receptor de taquiquinina 2 (tacr2).

Also Published As

Publication number Publication date
CO2023007404A2 (es) 2023-07-10
EP4240749A1 (en) 2023-09-13
WO2022096736A1 (en) 2022-05-12
MX2023005408A (es) 2023-07-25
KR20230106616A (ko) 2023-07-13
IL302745A (en) 2023-07-01
US20230406883A1 (en) 2023-12-21
AU2021374843A9 (en) 2024-08-08
JP2023551122A (ja) 2023-12-07
CN116745310A (zh) 2023-09-12
CA3197916A1 (en) 2022-05-12
AU2021374843A1 (en) 2023-06-08
PE20231952A1 (es) 2023-12-06

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