CL2017002255A1 - Procesos para preparar fluorocetólidos. - Google Patents

Procesos para preparar fluorocetólidos.

Info

Publication number
CL2017002255A1
CL2017002255A1 CL2017002255A CL2017002255A CL2017002255A1 CL 2017002255 A1 CL2017002255 A1 CL 2017002255A1 CL 2017002255 A CL2017002255 A CL 2017002255A CL 2017002255 A CL2017002255 A CL 2017002255A CL 2017002255 A1 CL2017002255 A1 CL 2017002255A1
Authority
CL
Chile
Prior art keywords
processes
fluorocetolides
prepare
fluorocetolide
intermediates
Prior art date
Application number
CL2017002255A
Other languages
English (en)
Spanish (es)
Inventor
David Eugene Pereira
Stephen E Schneider
Keshav Deo
Original Assignee
Cempra Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cempra Pharmaceuticals Inc filed Critical Cempra Pharmaceuticals Inc
Publication of CL2017002255A1 publication Critical patent/CL2017002255A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)
CL2017002255A 2015-03-06 2017-09-06 Procesos para preparar fluorocetólidos. CL2017002255A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562129305P 2015-03-06 2015-03-06

Publications (1)

Publication Number Publication Date
CL2017002255A1 true CL2017002255A1 (es) 2018-05-11

Family

ID=56880477

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2017002255A CL2017002255A1 (es) 2015-03-06 2017-09-06 Procesos para preparar fluorocetólidos.

Country Status (19)

Country Link
US (2) US20180044365A1 (OSRAM)
EP (1) EP3265100A4 (OSRAM)
JP (1) JP6773672B2 (OSRAM)
KR (1) KR20170133377A (OSRAM)
CN (1) CN107405355A (OSRAM)
AU (1) AU2016230027A1 (OSRAM)
BR (1) BR112017019176A2 (OSRAM)
CA (1) CA2978731A1 (OSRAM)
CL (1) CL2017002255A1 (OSRAM)
CO (1) CO2017010143A2 (OSRAM)
HK (1) HK1247097A1 (OSRAM)
IL (1) IL254306A0 (OSRAM)
MX (2) MX2017011454A (OSRAM)
PE (1) PE20180219A1 (OSRAM)
RU (1) RU2017131253A (OSRAM)
SG (2) SG11201707215XA (OSRAM)
TW (1) TW201638102A (OSRAM)
WO (1) WO2016144833A1 (OSRAM)
ZA (1) ZA201706505B (OSRAM)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2703475A1 (en) 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
EP2358379B1 (en) 2008-10-24 2015-12-16 Cempra Pharmaceuticals, Inc. Biodefenses using triazole-containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
KR20140139083A (ko) 2012-03-27 2014-12-04 셈프라 파마슈티컬스, 인크. 마크롤라이드계 항생제를 투여하기 위한 비경구 제제
RU2015138796A (ru) 2013-03-14 2017-04-19 Семпра Фармасьютикалс, Инк. Способы и составы для лечения респираторных заболеваний

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668282A (en) * 1970-05-08 1972-06-06 Stauffer Chemical Co Stabilized mixture employing n-(beta-0,0-dialkyldithiophosphoryl) aryl sulfonamides
EP1638549A4 (en) * 2003-03-10 2011-06-15 Optimer Pharmaceuticals Inc NEW ANTIBACTERIAL AGENTS
US7595300B2 (en) * 2005-12-13 2009-09-29 Kosan Biosciences Incorporated 7-quinolyl ketolide antibacterial agents
CA2703475A1 (en) * 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
US8376805B2 (en) * 2008-07-24 2013-02-19 Ideo Llc Printable pre-sewn stuffed toy composite sheets
JP5718488B2 (ja) * 2011-03-01 2015-05-13 ウォックハート リミテッド ケトライド中間体の調製方法
RU2015138796A (ru) * 2013-03-14 2017-04-19 Семпра Фармасьютикалс, Инк. Способы и составы для лечения респираторных заболеваний
JP6675973B2 (ja) * 2013-03-15 2020-04-08 センプラ ファーマシューティカルズ,インコーポレイテッド マクロライド抗菌薬を調製するための集束的な方法
AU2014248014B2 (en) * 2013-04-04 2018-11-08 President And Fellows Of Harvard College Macrolides and methods of their preparation and use

Also Published As

Publication number Publication date
SG10201908248PA (en) 2019-10-30
MX2020007742A (es) 2020-09-25
SG11201707215XA (en) 2017-10-30
KR20170133377A (ko) 2017-12-05
US20180044365A1 (en) 2018-02-15
CO2017010143A2 (es) 2018-02-28
ZA201706505B (en) 2021-04-28
HK1247097A1 (zh) 2018-09-21
US20210070797A1 (en) 2021-03-11
CA2978731A1 (en) 2016-09-15
AU2016230027A1 (en) 2017-09-28
TW201638102A (zh) 2016-11-01
JP2018508537A (ja) 2018-03-29
PE20180219A1 (es) 2018-01-31
BR112017019176A2 (pt) 2018-04-24
IL254306A0 (en) 2017-11-30
EP3265100A4 (en) 2019-01-09
JP6773672B2 (ja) 2020-10-21
MX2017011454A (es) 2018-01-23
CN107405355A (zh) 2017-11-28
WO2016144833A1 (en) 2016-09-15
RU2017131253A (ru) 2019-04-08
EP3265100A1 (en) 2018-01-10

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