PE20180219A1 - Procesos para preparar fluorocetolidos - Google Patents

Procesos para preparar fluorocetolidos

Info

Publication number
PE20180219A1
PE20180219A1 PE2017001500A PE2017001500A PE20180219A1 PE 20180219 A1 PE20180219 A1 PE 20180219A1 PE 2017001500 A PE2017001500 A PE 2017001500A PE 2017001500 A PE2017001500 A PE 2017001500A PE 20180219 A1 PE20180219 A1 PE 20180219A1
Authority
PE
Peru
Prior art keywords
processes
fluorocetolides
prepare
fluoroketolide
intermediates
Prior art date
Application number
PE2017001500A
Other languages
English (en)
Spanish (es)
Inventor
David Eugene Pereira
Stephen E Schneider
Keshav Deo
Original Assignee
Cempra Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cempra Pharmaceuticals Inc filed Critical Cempra Pharmaceuticals Inc
Publication of PE20180219A1 publication Critical patent/PE20180219A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Pyrane Compounds (AREA)
PE2017001500A 2015-03-06 2016-03-05 Procesos para preparar fluorocetolidos PE20180219A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562129305P 2015-03-06 2015-03-06

Publications (1)

Publication Number Publication Date
PE20180219A1 true PE20180219A1 (es) 2018-01-31

Family

ID=56880477

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2017001500A PE20180219A1 (es) 2015-03-06 2016-03-05 Procesos para preparar fluorocetolidos

Country Status (19)

Country Link
US (2) US20180044365A1 (OSRAM)
EP (1) EP3265100A4 (OSRAM)
JP (1) JP6773672B2 (OSRAM)
KR (1) KR20170133377A (OSRAM)
CN (1) CN107405355A (OSRAM)
AU (1) AU2016230027A1 (OSRAM)
BR (1) BR112017019176A2 (OSRAM)
CA (1) CA2978731A1 (OSRAM)
CL (1) CL2017002255A1 (OSRAM)
CO (1) CO2017010143A2 (OSRAM)
HK (1) HK1247097A1 (OSRAM)
IL (1) IL254306A0 (OSRAM)
MX (2) MX2017011454A (OSRAM)
PE (1) PE20180219A1 (OSRAM)
RU (1) RU2017131253A (OSRAM)
SG (2) SG11201707215XA (OSRAM)
TW (1) TW201638102A (OSRAM)
WO (1) WO2016144833A1 (OSRAM)
ZA (1) ZA201706505B (OSRAM)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2703475A1 (en) 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
EP2358379B1 (en) 2008-10-24 2015-12-16 Cempra Pharmaceuticals, Inc. Biodefenses using triazole-containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
KR20140139083A (ko) 2012-03-27 2014-12-04 셈프라 파마슈티컬스, 인크. 마크롤라이드계 항생제를 투여하기 위한 비경구 제제
RU2015138796A (ru) 2013-03-14 2017-04-19 Семпра Фармасьютикалс, Инк. Способы и составы для лечения респираторных заболеваний

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3668282A (en) * 1970-05-08 1972-06-06 Stauffer Chemical Co Stabilized mixture employing n-(beta-0,0-dialkyldithiophosphoryl) aryl sulfonamides
EP1638549A4 (en) * 2003-03-10 2011-06-15 Optimer Pharmaceuticals Inc NEW ANTIBACTERIAL AGENTS
US7595300B2 (en) * 2005-12-13 2009-09-29 Kosan Biosciences Incorporated 7-quinolyl ketolide antibacterial agents
CA2703475A1 (en) * 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
US8376805B2 (en) * 2008-07-24 2013-02-19 Ideo Llc Printable pre-sewn stuffed toy composite sheets
JP5718488B2 (ja) * 2011-03-01 2015-05-13 ウォックハート リミテッド ケトライド中間体の調製方法
RU2015138796A (ru) * 2013-03-14 2017-04-19 Семпра Фармасьютикалс, Инк. Способы и составы для лечения респираторных заболеваний
JP6675973B2 (ja) * 2013-03-15 2020-04-08 センプラ ファーマシューティカルズ,インコーポレイテッド マクロライド抗菌薬を調製するための集束的な方法
AU2014248014B2 (en) * 2013-04-04 2018-11-08 President And Fellows Of Harvard College Macrolides and methods of their preparation and use

Also Published As

Publication number Publication date
SG10201908248PA (en) 2019-10-30
MX2020007742A (es) 2020-09-25
SG11201707215XA (en) 2017-10-30
KR20170133377A (ko) 2017-12-05
US20180044365A1 (en) 2018-02-15
CO2017010143A2 (es) 2018-02-28
ZA201706505B (en) 2021-04-28
HK1247097A1 (zh) 2018-09-21
US20210070797A1 (en) 2021-03-11
CA2978731A1 (en) 2016-09-15
AU2016230027A1 (en) 2017-09-28
TW201638102A (zh) 2016-11-01
JP2018508537A (ja) 2018-03-29
BR112017019176A2 (pt) 2018-04-24
IL254306A0 (en) 2017-11-30
CL2017002255A1 (es) 2018-05-11
EP3265100A4 (en) 2019-01-09
JP6773672B2 (ja) 2020-10-21
MX2017011454A (es) 2018-01-23
CN107405355A (zh) 2017-11-28
WO2016144833A1 (en) 2016-09-15
RU2017131253A (ru) 2019-04-08
EP3265100A1 (en) 2018-01-10

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