CH626872A5 - - Google Patents

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Publication number
CH626872A5
CH626872A5 CH678277A CH678277A CH626872A5 CH 626872 A5 CH626872 A5 CH 626872A5 CH 678277 A CH678277 A CH 678277A CH 678277 A CH678277 A CH 678277A CH 626872 A5 CH626872 A5 CH 626872A5
Authority
CH
Switzerland
Prior art keywords
formula
group
alanyl
phenyl
compound
Prior art date
Application number
CH678277A
Other languages
German (de)
English (en)
Inventor
Cedric Herbert Hassall
William Henry Johnson
Noel Allan Roberts
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB25645/76A external-priority patent/GB1581543A/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH626872A5 publication Critical patent/CH626872A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06008Dipeptides with the first amino acid being neutral
    • C07K5/06017Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Rheumatology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CH678277A 1976-06-21 1977-06-02 CH626872A5 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB25645/76A GB1581543A (en) 1976-06-21 1976-06-21 Dipeptide derivatives
GB3249676 1976-08-04
GB1199777 1977-03-22

Publications (1)

Publication Number Publication Date
CH626872A5 true CH626872A5 (fi) 1981-12-15

Family

ID=27256763

Family Applications (1)

Application Number Title Priority Date Filing Date
CH678277A CH626872A5 (fi) 1976-06-21 1977-06-02

Country Status (17)

Country Link
US (1) US4176116A (fi)
JP (1) JPS52156811A (fi)
AT (1) AT355741B (fi)
AU (1) AU510077B2 (fi)
CA (1) CA1095027A (fi)
CH (1) CH626872A5 (fi)
DE (1) DE2727670A1 (fi)
DK (1) DK271977A (fi)
FR (1) FR2361346A1 (fi)
IE (1) IE45095B1 (fi)
IL (1) IL52307A (fi)
IT (1) IT1203108B (fi)
LU (1) LU77580A1 (fi)
NL (1) NL7706827A (fi)
NZ (1) NZ184394A (fi)
PH (1) PH14589A (fi)
SE (1) SE7707129L (fi)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU78804A1 (de) * 1977-12-30 1979-07-20 Byk Gulden Lomberg Chem Fab N-substituierte w-aminoalkanoyl-w-aminoalkansaeuren,ihre verwendung und verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel
US4277395A (en) * 1980-06-16 1981-07-07 Richardson-Merrell Inc. Novel enzyme inhibitors
US4309342A (en) * 1980-07-03 1982-01-05 Abbott Laboratories Antibacterial peptides
US4462943A (en) * 1980-11-24 1984-07-31 E. R. Squibb & Sons, Inc. Carboxyalkyl amino acid derivatives of various substituted prolines
US4820729A (en) * 1981-03-30 1989-04-11 Rorer Pharmaceutical Corporation N-substituted-amido-amino acids
CS226907B1 (en) * 1981-08-07 1984-04-16 Kasafirek Evzen Alkylamides of carboxyalkanoylpeptides
EP0132441A1 (en) * 1983-01-26 1985-02-06 University Patents, Inc. Antibacterial peptides
JPH0513980U (ja) * 1991-07-29 1993-02-23 アラコ株式会社 ツールバツグ
JPH05345754A (ja) * 1992-06-15 1993-12-27 Suntory Ltd ジペプチド誘導体およびそれを有効成分とする骨疾患の予防または治療剤
FR2733995B1 (fr) * 1995-05-09 1997-07-25 Inst Nat Sante Rech Med Inhibiteurs de l'inactivation de neuropeptides endogenes notamment la cholecystokinine, leurs procedes de preparation leur utilisation comme medicaments et procede de criblage de medicaments
WO2008060621A2 (en) * 2006-11-17 2008-05-22 Abbott Laboratories Aminopyrrolidines as chemokine receptor antagonists
WO2024044098A2 (en) * 2022-08-23 2024-02-29 Alexion Pharmaceuticals, Inc. Pharmaceutical compounds for the treatment of complement mediated disorders

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5255593A (en) * 1975-10-30 1977-05-07 Ajinomoto Kk Measuring method of enzyme activity

Also Published As

Publication number Publication date
JPS52156811A (en) 1977-12-27
DE2727670A1 (de) 1977-12-29
AT355741B (de) 1980-03-25
DK271977A (da) 1977-12-22
AU510077B2 (en) 1980-06-05
NL7706827A (nl) 1977-12-23
NZ184394A (en) 1980-08-26
IE45095B1 (en) 1982-06-16
IT1203108B (it) 1989-02-15
ATA432877A (de) 1979-08-15
AU2610777A (en) 1978-12-21
FR2361346B1 (fi) 1980-04-04
IL52307A0 (en) 1977-08-31
US4176116A (en) 1979-11-27
PH14589A (en) 1981-09-29
FR2361346A1 (fr) 1978-03-10
CA1095027A (en) 1981-02-03
SE7707129L (sv) 1977-12-22
IL52307A (en) 1980-11-30
IE45095L (en) 1977-12-21
LU77580A1 (fi) 1978-07-11

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Legal Events

Date Code Title Description
PL Patent ceased