CH626050A5 - - Google Patents

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Publication number
CH626050A5
CH626050A5 CH1600076A CH1600076A CH626050A5 CH 626050 A5 CH626050 A5 CH 626050A5 CH 1600076 A CH1600076 A CH 1600076A CH 1600076 A CH1600076 A CH 1600076A CH 626050 A5 CH626050 A5 CH 626050A5
Authority
CH
Switzerland
Prior art keywords
group
azaalanyl
amino
radical
methyl
Prior art date
Application number
CH1600076A
Other languages
German (de)
English (en)
Inventor
Conrad Peter Dorn
Shu Shu Yang
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of CH626050A5 publication Critical patent/CH626050A5/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0821Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
    • C07K5/0823Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp and Pro-amino acid; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0802Tripeptides with the first amino acid being neutral
    • C07K5/0804Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/0806Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
CH1600076A 1975-12-23 1976-12-20 CH626050A5 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/643,721 US4064236A (en) 1975-12-23 1975-12-23 Peptide carbazates and pharmaceutical composition

Publications (1)

Publication Number Publication Date
CH626050A5 true CH626050A5 (es) 1981-10-30

Family

ID=24582010

Family Applications (1)

Application Number Title Priority Date Filing Date
CH1600076A CH626050A5 (es) 1975-12-23 1976-12-20

Country Status (9)

Country Link
US (1) US4064236A (es)
JP (1) JPS5278829A (es)
CH (1) CH626050A5 (es)
DE (1) DE2658254A1 (es)
DK (1) DK551276A (es)
FR (1) FR2336139A1 (es)
GB (1) GB1520830A (es)
NL (1) NL7613661A (es)
SE (1) SE7613855L (es)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1592552A (en) * 1976-12-10 1981-07-08 Inst Nat Sante Rech Med Pseudopeptides used as medicaments
CS226907B1 (en) * 1981-08-07 1984-04-16 Kasafirek Evzen Alkylamides of carboxyalkanoylpeptides
US5464739A (en) 1994-08-22 1995-11-07 Bayer Corporation Composition method for determining the presence of leukocyte cells, esterase or protease in a test sample
DE19612644A1 (de) * 1996-03-29 1997-10-02 Bayer Ag Oxadiazin-Derivate
US8394813B2 (en) 2000-11-14 2013-03-12 Shire Llc Active agent delivery systems and methods for protecting and administering active agents
US7169752B2 (en) 2003-09-30 2007-01-30 New River Pharmaceuticals Inc. Compounds and compositions for prevention of overdose of oxycodone
US20060014697A1 (en) 2001-08-22 2006-01-19 Travis Mickle Pharmaceutical compositions for prevention of overdose or abuse
US7105486B2 (en) * 2002-02-22 2006-09-12 New River Pharmaceuticals Inc. Abuse-resistant amphetamine compounds
US7659253B2 (en) 2002-02-22 2010-02-09 Shire Llc Abuse-resistant amphetamine prodrugs
US7700561B2 (en) * 2002-02-22 2010-04-20 Shire Llc Abuse-resistant amphetamine prodrugs
US20060233863A1 (en) 2003-02-10 2006-10-19 Enzymotec Ltd. Oils enriched with diacylglycerols and phytosterol esters and unit dosage forms thereof for use in therapy
IL155136A0 (en) 2003-02-10 2003-10-31 Enzymotec Ltd A composition for reducing blood cholesterol and triglycerides
AU2004251647B2 (en) 2003-05-29 2010-01-14 Takeda Pharmaceutical Company Limited Abuse resistant amphetamine compounds
CN101035594B (zh) * 2004-08-09 2013-10-23 酶学技术有限公司 用于糖尿病患者的食品
JP5118965B2 (ja) 2004-08-10 2013-01-16 エンジモテック リミテッド 植物成分を必要とする治療方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3904593A (en) * 1973-02-07 1975-09-09 American Home Prod Peptide derivatives having an ' -hydrazide linkage and preparation thereof
US3888840A (en) * 1973-02-07 1975-06-10 American Home Prod Novel hydrazinocarboxamide derivatives and preparation thereof

Also Published As

Publication number Publication date
SE7613855L (sv) 1977-06-24
GB1520830A (en) 1978-08-09
DK551276A (da) 1977-06-24
JPS5278829A (en) 1977-07-02
US4064236A (en) 1977-12-20
NL7613661A (nl) 1977-06-27
DE2658254A1 (de) 1977-07-07
FR2336139B1 (es) 1979-07-13
FR2336139A1 (fr) 1977-07-22

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Legal Events

Date Code Title Description
PL Patent ceased