CH576921A5 - - Google Patents
Info
- Publication number
- CH576921A5 CH576921A5 CH395572A CH395572A CH576921A5 CH 576921 A5 CH576921 A5 CH 576921A5 CH 395572 A CH395572 A CH 395572A CH 395572 A CH395572 A CH 395572A CH 576921 A5 CH576921 A5 CH 576921A5
- Authority
- CH
- Switzerland
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
- C07F9/6571—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms
- C07F9/6574—Esters of oxyacids of phosphorus
- C07F9/65744—Esters of oxyacids of phosphorus condensed with carbocyclic or heterocyclic rings or ring systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Braiding, Manufacturing Of Bobbin-Net Or Lace, And Manufacturing Of Nets By Knotting (AREA)
- Hydrogenated Pyridines (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT49167/71A IT951631B (it) | 1971-03-18 | 1971-03-18 | Composti utili per la separazione di isomeri ottici geometrici e strutturali e relativo procedimen to di sintesi |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH576921A5 true CH576921A5 (enExample) | 1976-06-30 |
Family
ID=11269830
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH395572A CH576921A5 (enExample) | 1971-03-18 | 1972-03-17 |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US3848030A (enExample) |
| JP (1) | JPS5547013B1 (enExample) |
| AU (1) | AU462431B2 (enExample) |
| BE (1) | BE780887A (enExample) |
| CA (1) | CA961500A (enExample) |
| CH (1) | CH576921A5 (enExample) |
| DE (1) | DE2212660C3 (enExample) |
| DK (1) | DK139944B (enExample) |
| ES (1) | ES400862A1 (enExample) |
| FR (1) | FR2129741A5 (enExample) |
| GB (1) | GB1360946A (enExample) |
| IL (1) | IL38860A (enExample) |
| IT (1) | IT951631B (enExample) |
| NL (1) | NL7203574A (enExample) |
| NO (1) | NO136357C (enExample) |
| PH (1) | PH10768A (enExample) |
| SE (1) | SE409323B (enExample) |
| ZA (1) | ZA721297B (enExample) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4143028A (en) * | 1977-12-05 | 1979-03-06 | Ciba-Geigy Corporation | Alkylated 1,1'-biphenyl-2,2'-diyl phosphonites and stabilized compositions |
| US5288914A (en) * | 1984-08-27 | 1994-02-22 | The Dow Chemical Company | Poly(arylcyclobutenes) |
| NL8403224A (nl) * | 1984-10-24 | 1986-05-16 | Oce Andeno Bv | Dioxafosforinanen, de bereiding ervan en de toepassing voor het splitsen van optisch actieve verbindingen. |
| DE3940765A1 (de) * | 1989-12-09 | 1991-06-13 | Hoechst Ag | Verfahren zur herstellung reiner cyclischer phosphorsaeurediarylester |
| EP0759904B1 (en) * | 1994-05-16 | 2000-07-05 | Merrell Pharmaceuticals Inc. | Process and diastereomeric salts useful for the optical resolution of racemic 4-[4-[-4-(hydroxydiphenylmethyl)-1-piperidinyl]-1-hydroxybutyl]-alpha,alpha-dimethylbenzene acetic acid. |
| JP4725757B2 (ja) * | 1999-03-24 | 2011-07-13 | 東ソー株式会社 | ビナフトールリン酸誘導体及びその利用 |
| EP1038877B1 (en) * | 1999-03-24 | 2004-03-10 | Tosoh Corporation | Binaphthol monophosphoric acid derivative and its use |
| AU7949900A (en) * | 1999-10-22 | 2001-05-08 | Takeda Chemical Industries Ltd. | Process for producing optically active naphthalene derivative and optical resolver therefor |
| EP1229019A4 (en) * | 1999-11-10 | 2004-08-18 | Takeda Chemical Industries Ltd | METHOD FOR THE PRODUCTION OF OPTICALLY ACTIVE, CYCLIC ENAMINONE DERIVATIVES |
| US6391926B2 (en) * | 2000-03-13 | 2002-05-21 | Tosoh Corporation | Optically active phosphate derivative |
| CA2453337C (en) | 2001-07-09 | 2012-08-28 | Zonagen, Inc. | Methods and materials for the treatment of testosterone deficiency in men |
| CN100410234C (zh) * | 2003-04-25 | 2008-08-13 | 东亚合成株式会社 | 利用手性布朗斯台德酸的不对称合成用催化剂和使用该催化剂的不对称合成方法 |
| US7229557B2 (en) * | 2004-02-04 | 2007-06-12 | Konec, Inc. | Method to separate stereoisomers |
| EP2486032A4 (en) * | 2009-10-09 | 2013-03-27 | Hetero Research Foundation | RACEMATSPALTUNG SUBSTITUTED 2- (2-PYRIDINYLMETHYLSULFINYL) -1H-BENZIMIDAZOLE |
| UA113291C2 (xx) | 2011-08-04 | 2017-01-10 | Метаболіти транскломіфену і їх застосування | |
| AU2013306393A1 (en) | 2012-08-21 | 2015-02-19 | Repros Therapeutics Inc. | Trans-clomiphene formulations and uses thereof |
| CN104994877A (zh) | 2012-11-02 | 2015-10-21 | 利普生物药剂公司 | 用于癌症治疗的反式-克罗米芬 |
| CN106068121A (zh) * | 2014-03-11 | 2016-11-02 | 利普生物药剂公司 | 使用单一溶剂进行克罗米芬合成 |
| UA121971C2 (uk) | 2014-07-24 | 2020-08-25 | Аспен Парк Фармасутікалс, Інк. | Лікування викликаних антиандрогенною терапією припливів та остеопорозу із застосуванням цис-кломіфену |
| EP3015453B1 (en) | 2014-10-28 | 2016-10-12 | F.I.S.- Fabbrica Italiana Sintetici S.p.A. | Process for the preparation of Clomiphene |
| EP3015454A1 (en) * | 2014-10-28 | 2016-05-04 | F.I.S.- Fabbrica Italiana Sintetici S.p.A. | Stable solid form of trans-Clomiphene citrate |
| CN108463453A (zh) * | 2016-04-22 | 2018-08-28 | 意大利合成制造有限公司 | 用于制备具有针状晶体习性的柠檬酸恩氯米芬的方法 |
| KR20200052349A (ko) | 2017-09-11 | 2020-05-14 | 아토사 테라퓨틱스, 인크. | 엔독시펜을 제조 및 사용하는 방법 |
| FR3082842A1 (fr) * | 2018-06-21 | 2019-12-27 | Veru Inc. | Polymorphe de cis-clomiphene (zuclomiphene) et procedes d'utilisation de celui-ci |
| US12201591B2 (en) | 2019-07-03 | 2025-01-21 | Atossa Therapeutics, Inc. | Sustained release compositions of endoxifen |
| CA3098552A1 (en) | 2019-11-14 | 2021-05-14 | Apotex Inc. | Processes for the preparation of zuclomiphene and intermediates thereof |
| CA3098725A1 (en) | 2019-11-14 | 2021-05-14 | Apotex Inc. | Zuclpomiphene salts and crystalline forms thereof |
| CA3105944A1 (en) | 2020-01-22 | 2021-07-22 | Apotex Inc. | Crystalline forms of zuclomiphene citrate |
| EP3907213A1 (en) | 2020-05-04 | 2021-11-10 | Pcas | Processes for the production of isomerically pure or enriched cis-clomiphene |
| US11578025B2 (en) | 2020-10-19 | 2023-02-14 | Apotex Inc. | Processes for the preparation of zuclomiphene intermediates |
-
1971
- 1971-03-18 IT IT49167/71A patent/IT951631B/it active
-
1972
- 1972-02-28 ZA ZA721297A patent/ZA721297B/xx unknown
- 1972-02-29 IL IL38860A patent/IL38860A/xx unknown
- 1972-03-03 PH PH13312A patent/PH10768A/en unknown
- 1972-03-03 AU AU39611/72A patent/AU462431B2/en not_active Expired
- 1972-03-09 CA CA136,671A patent/CA961500A/en not_active Expired
- 1972-03-09 GB GB1104172A patent/GB1360946A/en not_active Expired
- 1972-03-10 US US00233793A patent/US3848030A/en not_active Expired - Lifetime
- 1972-03-15 SE SE7203303A patent/SE409323B/xx unknown
- 1972-03-16 DE DE2212660A patent/DE2212660C3/de not_active Expired
- 1972-03-17 DK DK127372AA patent/DK139944B/da unknown
- 1972-03-17 NL NL7203574A patent/NL7203574A/xx not_active Application Discontinuation
- 1972-03-17 BE BE780887A patent/BE780887A/xx unknown
- 1972-03-17 FR FR7209350A patent/FR2129741A5/fr not_active Expired
- 1972-03-17 JP JP2661472A patent/JPS5547013B1/ja active Pending
- 1972-03-17 NO NO880/72A patent/NO136357C/no unknown
- 1972-03-17 ES ES400862A patent/ES400862A1/es not_active Expired
- 1972-03-17 CH CH395572A patent/CH576921A5/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| IT951631B (it) | 1973-07-10 |
| DK139944B (da) | 1979-05-21 |
| IL38860A (en) | 1975-06-25 |
| FR2129741A5 (enExample) | 1972-10-27 |
| DK139944C (enExample) | 1979-10-22 |
| CA961500A (en) | 1975-01-21 |
| DE2212660C3 (de) | 1981-09-24 |
| AU3961172A (en) | 1973-09-06 |
| JPS5547013B1 (enExample) | 1980-11-27 |
| NL7203574A (enExample) | 1972-09-20 |
| IL38860A0 (en) | 1972-04-27 |
| AU462431B2 (en) | 1975-06-09 |
| DE2212660B2 (de) | 1980-07-10 |
| SE409323B (sv) | 1979-08-13 |
| GB1360946A (en) | 1974-07-24 |
| US3848030A (en) | 1974-11-12 |
| ZA721297B (en) | 1973-03-28 |
| NO136357B (enExample) | 1977-05-16 |
| PH10768A (en) | 1977-09-05 |
| DE2212660A1 (de) | 1972-09-28 |
| BE780887A (fr) | 1972-07-17 |
| NO136357C (no) | 1977-08-24 |
| ES400862A1 (es) | 1976-04-16 |
Similar Documents
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PL | Patent ceased | ||
| PL | Patent ceased |