CH571001A5 - - Google Patents

Info

Publication number
CH571001A5
CH571001A5 CH581473A CH581473A CH571001A5 CH 571001 A5 CH571001 A5 CH 571001A5 CH 581473 A CH581473 A CH 581473A CH 581473 A CH581473 A CH 581473A CH 571001 A5 CH571001 A5 CH 571001A5
Authority
CH
Switzerland
Prior art keywords
formula
acid
lower alkyl
derivatives
halogen atom
Prior art date
Application number
CH581473A
Other languages
English (en)
French (fr)
Original Assignee
Centre Etd Ind Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority to FR7314310A priority Critical patent/FR2183716A1/fr
Application filed by Centre Etd Ind Pharma filed Critical Centre Etd Ind Pharma
Priority to CH581473A priority patent/CH571001A5/fr
Priority to BE130386A priority patent/BE798677A/xx
Priority to DE2321705A priority patent/DE2321705A1/de
Priority to CA170,487A priority patent/CA999860A/en
Priority to JP48051065A priority patent/JPS4947391A/ja
Publication of CH571001A5 publication Critical patent/CH571001A5/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CH581473A 1972-05-05 1973-04-24 CH571001A5 (enExample)

Priority Applications (6)

Application Number Priority Date Filing Date Title
FR7314310A FR2183716A1 (en) 1972-05-05 1973-04-19 Substd-6-phenyl-4h-imidazo (1,2-a)-1,4-benzo diazepines - - tranquillisers anxiolytics,sedatives and muscle-relaxants
CH581473A CH571001A5 (enExample) 1972-05-05 1973-04-24
BE130386A BE798677A (fr) 1972-05-05 1973-04-25 Derives de benzodiazepine, leur preparation et leurs applications
DE2321705A DE2321705A1 (de) 1972-05-05 1973-04-28 Benzodiazepinderivate, ihre herstellung und verwendung
CA170,487A CA999860A (en) 1972-05-05 1973-05-04 Imidazo-(1,2-a)-(benzodiazepine-1,4) compounds
JP48051065A JPS4947391A (enExample) 1972-05-05 1973-05-07

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB2114172 1972-05-05
CH581473A CH571001A5 (enExample) 1972-05-05 1973-04-24

Publications (1)

Publication Number Publication Date
CH571001A5 true CH571001A5 (enExample) 1975-12-31

Family

ID=25698412

Family Applications (1)

Application Number Title Priority Date Filing Date
CH581473A CH571001A5 (enExample) 1972-05-05 1973-04-24

Country Status (6)

Country Link
JP (1) JPS4947391A (enExample)
BE (1) BE798677A (enExample)
CA (1) CA999860A (enExample)
CH (1) CH571001A5 (enExample)
DE (1) DE2321705A1 (enExample)
FR (1) FR2183716A1 (enExample)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ZA755418B (en) * 1974-09-11 1977-06-29 Hoffmann La Roche Diazepine derivatives
US3910946A (en) * 1974-09-12 1975-10-07 Upjohn Co 4H-Imidazo{8 1,2-a{9 {8 1,4{9 benzodiazepines
DE2547652A1 (de) * 1974-11-15 1976-05-20 Upjohn Co Pharmazeutische zubereitung
US4044142A (en) 1975-02-03 1977-08-23 Roussel Uclaf 1,2-Dihydro-6-phenyl-1H,4H-imidazobenzodiazepin-1-ones
US4134976A (en) * 1975-02-15 1979-01-16 Roussel Uclaf 1,2-Dihydro-6-phenyl-1H,4H-imidazobenzodiazepin-1-ones
SE422580B (sv) * 1975-08-07 1982-03-15 Hoffmann La Roche Analogiforfarande for framstellning av imidazo (1,5-a)(1,4)diazepin-foreningar
US4185102A (en) 1975-11-04 1980-01-22 Roussel Uclaf 1,2-Dihydro-6-phenyl-1H,4H-imidazobenzodiazepin-1-ones
JPS60202096A (ja) * 1984-03-22 1985-10-12 日産自動車株式会社 フオ−クリフトのフオ−ク移動装置
DE3610848A1 (de) * 1986-04-01 1987-10-15 Boehringer Ingelheim Kg Neue 1,4-diazepine
SU1681729A3 (ru) * 1986-07-25 1991-09-30 Берингер Ингельгейм Кг (Фирма) Способ получени производных 1,4-бензодиазепина
CA2068500A1 (en) * 1991-05-14 1992-11-15 Roger M. Freidinger 1,4-benzodiazepines with 5- and 6-membered heterocyclic rings
WO1994026723A2 (en) * 1993-05-14 1994-11-24 Genentech, Inc. ras FARNESYL TRANSFERASE INHIBITORS
GB9911152D0 (en) * 1999-05-14 1999-07-14 Glaxo Group Ltd Short-acting benzodiazepines
US7160880B1 (en) 1999-05-14 2007-01-09 Cenes Limited Short-acting benzodiazepines
KR20150081370A (ko) 2006-07-10 2015-07-13 파이온 유케이 리미티드 속효형 벤조디아제핀 염 및 이의 중합체 형태
EP2450039A1 (en) 2010-11-08 2012-05-09 PAION UK Ltd. Dosing regimen for sedation with CNS 7056 (Remimazolam)
CN108033964B (zh) * 2017-12-28 2021-02-09 杭州奥默医药股份有限公司 一种吡啶基咪唑并苯并二氮杂卓丙酸酯化合物及其合成和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE787251A (fr) * 1971-08-04 1973-02-05 Upjohn Co Nouvelles benzodiazepines et leur preparation

Also Published As

Publication number Publication date
BE798677A (fr) 1973-08-16
FR2183716B1 (enExample) 1976-12-03
JPS4947391A (enExample) 1974-05-08
DE2321705A1 (de) 1973-11-15
CA999860A (en) 1976-11-16
FR2183716A1 (en) 1973-12-21

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Legal Events

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