CA2872021C - Glucokinase activator compositions for the treatment of diabetes - Google Patents
Glucokinase activator compositions for the treatment of diabetes Download PDFInfo
- Publication number
- CA2872021C CA2872021C CA2872021A CA2872021A CA2872021C CA 2872021 C CA2872021 C CA 2872021C CA 2872021 A CA2872021 A CA 2872021A CA 2872021 A CA2872021 A CA 2872021A CA 2872021 C CA2872021 C CA 2872021C
- Authority
- CA
- Canada
- Prior art keywords
- insulin
- diabetes
- pharmaceutically acceptable
- glucose
- glucokinase activator
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261648110P | 2012-05-17 | 2012-05-17 | |
| US61/648,110 | 2012-05-17 | ||
| PCT/US2013/041076 WO2013173417A2 (en) | 2012-05-17 | 2013-05-15 | Glucokinase activator compositions for the treatment of diabetes |
Publications (2)
| Publication Number | Publication Date |
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| CA2872021A1 CA2872021A1 (en) | 2013-11-21 |
| CA2872021C true CA2872021C (en) | 2022-08-16 |
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| Application Number | Title | Priority Date | Filing Date |
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| CA2872021A Active CA2872021C (en) | 2012-05-17 | 2013-05-15 | Glucokinase activator compositions for the treatment of diabetes |
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| KR101878252B1 (ko) | 2010-05-26 | 2018-07-13 | 브이티브이 테라퓨틱스 엘엘씨 | 글루코키나아제 활성화제와 병용되는 메트포르민의 용도, 및 메트포르민과 글루코키나아제 활성화제를 포함하는 조성물 |
| IN2014DN09554A (esLanguage) | 2012-05-17 | 2015-07-17 | Transtech Pharma Llc | |
| KR102408480B1 (ko) | 2018-05-30 | 2022-06-10 | 이삼구 | 당뇨질환의 치료용 조성물 |
| US20210214312A1 (en) * | 2018-05-31 | 2021-07-15 | Hua Medicine (Shanghai) Ltd. | Pharmaceutical combination, composition and formulation containing glucokinase activator and a-glucosidase inhibitor, prepraration methods therefor and uses thereof |
| EP4487909A3 (en) * | 2018-06-12 | 2025-03-19 | vTv Therapeutics LLC | Therapeutic uses of glucokinase activators in combination with insulin or insulin analogs |
| US11872221B2 (en) | 2020-01-31 | 2024-01-16 | Hua Medicine (Shanghai) Ltd. | Treating untreated or treatment-resistant diabetes with glucokinase activator |
| WO2021151251A1 (en) * | 2020-01-31 | 2021-08-05 | Hua Medicine (Shanghai) Ltd. | Treating treatment-resistant diabetes with glucokinase activator |
| WO2021167840A1 (en) | 2020-02-18 | 2021-08-26 | Vtv Therapeutics Llc | Sulfoxide and sulfone glucokinase activators and methods of use thereof |
| CA3185834A1 (en) * | 2020-06-04 | 2021-12-09 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with hepatic impairment |
| WO2021243645A1 (en) * | 2020-06-04 | 2021-12-09 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with renal impairment |
| US11857536B2 (en) | 2020-06-04 | 2024-01-02 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with renal impairment |
| CN116056760A (zh) * | 2020-06-08 | 2023-05-02 | 维特卫治疗有限责任公司 | {2-[3-环己基-3-(反式-4-丙氧基-环己基)-脲基]-噻唑-5-基硫烷基}-乙酸的结晶形式及其用途 |
| KR20230048502A (ko) * | 2020-06-08 | 2023-04-11 | 브이티브이 테라퓨틱스 엘엘씨 | ｛2-[3-사이클로헥실-3-(트랜스-4-프로폭시-사이클로헥실)-우레이도]-티아졸-5-일설파닐｝-아세트산의 염 또는 공결정 및 그의 용도 |
| CN115350268B (zh) * | 2022-08-24 | 2025-02-11 | 深圳青澜生物技术有限公司 | 一种用于治疗糖尿病的制剂、微针及其制备工艺 |
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| KR101878252B1 (ko) * | 2010-05-26 | 2018-07-13 | 브이티브이 테라퓨틱스 엘엘씨 | 글루코키나아제 활성화제와 병용되는 메트포르민의 용도, 및 메트포르민과 글루코키나아제 활성화제를 포함하는 조성물 |
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| CA2903440C (en) | 2013-03-04 | 2021-04-13 | Vtv Therapeutics Llc | Solid compositions comprising a glucokinase activator and methods of making and using the same |
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2013
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Also Published As
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| KR20210027547A (ko) | 2021-03-10 |
| MX360304B (es) | 2018-10-29 |
| IN2014DN09554A (esLanguage) | 2015-07-17 |
| AU2013262895A1 (en) | 2014-11-13 |
| ES2878001T3 (es) | 2021-11-18 |
| US10004782B2 (en) | 2018-06-26 |
| SG11201406987UA (en) | 2014-12-30 |
| KR102371364B1 (ko) | 2022-03-07 |
| AU2017203835B2 (en) | 2018-11-22 |
| IL235484A0 (en) | 2014-12-31 |
| JP6234443B2 (ja) | 2017-11-22 |
| EP2849776A2 (en) | 2015-03-25 |
| CN118453592A (zh) | 2024-08-09 |
| BR112014028622A2 (pt) | 2017-06-27 |
| MX2014013105A (es) | 2015-04-08 |
| EP2849776B1 (en) | 2021-04-21 |
| US20140066372A1 (en) | 2014-03-06 |
| AU2017203835A1 (en) | 2017-06-22 |
| SG10201609644UA (en) | 2017-01-27 |
| EA201492109A1 (ru) | 2015-07-30 |
| US10980861B2 (en) | 2021-04-20 |
| JP2015517525A (ja) | 2015-06-22 |
| CA2872021A1 (en) | 2013-11-21 |
| WO2013173417A3 (en) | 2014-02-20 |
| US10588943B2 (en) | 2020-03-17 |
| HK1202458A1 (en) | 2015-10-02 |
| US20200138909A1 (en) | 2020-05-07 |
| CN104349790A (zh) | 2015-02-11 |
| US20180311314A1 (en) | 2018-11-01 |
| KR20150013838A (ko) | 2015-02-05 |
| WO2013173417A2 (en) | 2013-11-21 |
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