CA2844742A1 - Kinase inhibitor polymorphs - Google Patents
Kinase inhibitor polymorphs Download PDFInfo
- Publication number
- CA2844742A1 CA2844742A1 CA2844742A CA2844742A CA2844742A1 CA 2844742 A1 CA2844742 A1 CA 2844742A1 CA 2844742 A CA2844742 A CA 2844742A CA 2844742 A CA2844742 A CA 2844742A CA 2844742 A1 CA2844742 A1 CA 2844742A1
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Classifications
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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- Nitrogen Condensed Heterocyclic Rings (AREA)
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| US201161522624P | 2011-08-11 | 2011-08-11 | |
| US61/522,624 | 2011-08-11 | ||
| PCT/US2012/050453 WO2013023184A1 (en) | 2011-08-11 | 2012-08-10 | Kinase inhibitor polymorphs |
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| CA2844742A1 true CA2844742A1 (en) | 2013-02-14 |
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| US9365634B2 (en) | 2007-05-29 | 2016-06-14 | Angiochem Inc. | Aprotinin-like polypeptides for delivering agents conjugated thereto to tissues |
| EP2346896A4 (en) | 2008-10-15 | 2014-06-25 | Angiochem Inc | ETOPOSID AND DOXORUBICIN CONJUGATES FOR ACTIVITY EXTRACTION |
| US8921314B2 (en) | 2008-10-15 | 2014-12-30 | Angiochem, Inc. | Conjugates of GLP-1 agonists and uses thereof |
| JP5759379B2 (ja) | 2008-12-05 | 2015-08-05 | アンジオケム インコーポレーテッド | ニューロテンシンまたはニューロテンシンアナログおよびその使用 |
| WO2010069074A1 (en) | 2008-12-17 | 2010-06-24 | Universite Du Quebec A Montreal | Membrane type-1 matrix metalloprotein inhibitors and uses thereof |
| ES2729261T3 (es) | 2009-04-20 | 2019-10-31 | Angiochem Inc | Tratamiento del cáncer de ovario utilizando un agente anticancerígeno conjugado con un análogo de Angiopep-2 |
| CN102596993A (zh) | 2009-07-02 | 2012-07-18 | 安吉奥开米公司 | 多聚体肽结合物以及其应用 |
| CN106924741A (zh) * | 2011-11-08 | 2017-07-07 | 因特利凯有限责任公司 | 使用多种药剂的治疗方案 |
| CN104250250A (zh) * | 2013-06-25 | 2014-12-31 | 苏州科捷生物医药有限公司 | 4-芳香胺基嘧啶类化合物及其抗肿瘤用途 |
| WO2015073644A1 (en) | 2013-11-13 | 2015-05-21 | Novartis Ag | Mtor inhibitors for enhancing the immune response |
| US10640569B2 (en) | 2013-12-19 | 2020-05-05 | Novartis Ag | Human mesothelin chimeric antigen receptors and uses thereof |
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| CN107109419B (zh) | 2014-07-21 | 2020-12-22 | 诺华股份有限公司 | 使用cd33嵌合抗原受体治疗癌症 |
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| KR102804360B1 (ko) | 2014-09-17 | 2025-05-12 | 노파르티스 아게 | 입양 면역요법을 위한 키메라 수용체에 의한 세포독성 세포의 표적화 |
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| SG11201708516YA (en) | 2015-04-17 | 2017-11-29 | David Maxwell Barrett | Methods for improving the efficacy and expansion of chimeric antigen receptor-expressing cells |
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| JP6823055B2 (ja) | 2015-06-15 | 2021-01-27 | アンジオケム インコーポレーテッド | 軟髄膜癌腫症の治療方法 |
| ES2636646B1 (es) * | 2016-04-05 | 2018-08-03 | Universidade De Santiago De Compostela | NUEVOS VEHÍCULOS PARA LA TRANSFECCIÓN DE miRNAs |
| CN116769050A (zh) | 2016-07-20 | 2023-09-19 | 犹他大学研究基金会 | Cd229 car t细胞及其使用方法 |
| MX2019003886A (es) | 2016-10-07 | 2019-08-05 | Novartis Ag | Receptores de antigenos quimericos para el tratamiento del cancer. |
| ES2837396T3 (es) | 2016-11-23 | 2021-06-30 | Bayer Cropscience Ag | Derivados de 2-[3-(alquilsulfonil)-2H-indazol-2-il]-3H-imidazo[4,5-b]piridina y compuestos similares como pesticidas |
| US20200055948A1 (en) | 2017-04-28 | 2020-02-20 | Novartis Ag | Cells expressing a bcma-targeting chimeric antigen receptor, and combination therapy with a gamma secretase inhibitor |
| BR112020013794B1 (pt) * | 2018-01-09 | 2023-05-02 | Halcyon Labs Private Limited | Processo para a preparação de crisaborola de fórmula (i), compostos, uso de um composto de fórmula (iv), (iii) ou (ii), processo para a preparação de crisaborola altamente pura e sal |
| EP3784351A1 (en) | 2018-04-27 | 2021-03-03 | Novartis AG | Car t cell therapies with enhanced efficacy |
| EP3788369A1 (en) | 2018-05-01 | 2021-03-10 | Novartis Ag | Biomarkers for evaluating car-t cells to predict clinical outcome |
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| TW370529B (en) * | 1992-12-17 | 1999-09-21 | Pfizer | Pyrazolopyrimidines |
| US7420084B2 (en) * | 2002-07-18 | 2008-09-02 | Teva Pharmaceutical Industries Ltd. | Polymorphic forms of nateglinide |
| US8476282B2 (en) * | 2008-11-03 | 2013-07-02 | Intellikine Llc | Benzoxazole kinase inhibitors and methods of use |
| AR084824A1 (es) * | 2011-01-10 | 2013-06-26 | Intellikine Inc | Procesos para preparar isoquinolinonas y formas solidas de isoquinolinonas |
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2012
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- 2012-08-10 PE PE2014000191A patent/PE20141358A1/es not_active Application Discontinuation
- 2012-08-10 CA CA2844742A patent/CA2844742A1/en not_active Abandoned
- 2012-08-10 HK HK14112711.7A patent/HK1199203A1/xx unknown
- 2012-08-10 EA EA201490446A patent/EA027970B1/ru not_active IP Right Cessation
- 2012-08-10 MX MX2014001662A patent/MX2014001662A/es unknown
- 2012-08-10 BR BR112014003214A patent/BR112014003214A2/pt not_active Application Discontinuation
- 2012-08-10 MY MYPI2014000363A patent/MY186267A/en unknown
- 2012-08-10 KR KR1020147006105A patent/KR20140079368A/ko not_active Ceased
- 2012-08-10 PH PH1/2014/500331A patent/PH12014500331A1/en unknown
- 2012-08-10 US US14/238,426 patent/US20150065524A1/en not_active Abandoned
- 2012-08-10 SG SG2014009492A patent/SG2014009492A/en unknown
- 2012-08-10 CN CN201280043863.6A patent/CN103957918A/zh active Pending
- 2012-08-10 AU AU2012294202A patent/AU2012294202B2/en active Active
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| KR20140079368A (ko) | 2014-06-26 |
| CL2014000343A1 (es) | 2014-10-17 |
| PE20141358A1 (es) | 2014-10-12 |
| CO6960542A2 (es) | 2014-05-30 |
| EA201490446A1 (ru) | 2014-05-30 |
| IL230850A0 (en) | 2014-03-31 |
| RU2636588C2 (ru) | 2017-11-24 |
| TN2014000063A1 (en) | 2015-07-01 |
| PH12014500331A1 (en) | 2014-03-31 |
| AU2012294202B2 (en) | 2017-02-23 |
| SG2014009492A (en) | 2014-09-26 |
| CR20140082A (es) | 2014-06-03 |
| MY186267A (en) | 2021-07-01 |
| EP2741749A4 (en) | 2015-04-15 |
| AU2012294202A1 (en) | 2014-03-06 |
| EP2741749A1 (en) | 2014-06-18 |
| EA027970B1 (ru) | 2017-09-29 |
| NZ622208A (en) | 2016-04-29 |
| ECSP14013236A (es) | 2014-06-30 |
| WO2013023184A1 (en) | 2013-02-14 |
| DOP2014000027A (es) | 2014-07-15 |
| US20150065524A1 (en) | 2015-03-05 |
| MX2014001662A (es) | 2014-08-26 |
| JP2014521726A (ja) | 2014-08-28 |
| HK1199203A1 (en) | 2015-06-26 |
| SG10201606288TA (en) | 2016-09-29 |
| ZA201401211B (en) | 2015-12-23 |
| RU2014109023A (ru) | 2015-09-20 |
| CN103957918A (zh) | 2014-07-30 |
| BR112014003214A2 (pt) | 2017-03-14 |
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