CA2838055C - Use of 4-((1r,3s)-6-chloro-3-phenyl-indan-1-yl)-1,2,2-trimethyl-piperaz ine and the salts thereof in the treatment of psychosis - Google Patents
Use of 4-((1r,3s)-6-chloro-3-phenyl-indan-1-yl)-1,2,2-trimethyl-piperaz ine and the salts thereof in the treatment of psychosis Download PDFInfo
- Publication number
- CA2838055C CA2838055C CA2838055A CA2838055A CA2838055C CA 2838055 C CA2838055 C CA 2838055C CA 2838055 A CA2838055 A CA 2838055A CA 2838055 A CA2838055 A CA 2838055A CA 2838055 C CA2838055 C CA 2838055C
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- Prior art keywords
- compound
- pharmaceutically acceptable
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- acceptable salt
- weekly
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- A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
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- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
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- Life Sciences & Earth Sciences (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| DKPA201100465 | 2011-06-20 | ||
| PCT/EP2012/061779 WO2012175531A1 (en) | 2011-06-20 | 2012-06-20 | Method of administration of 4-((1r,3s)-6-chloro-3-phenyl-indan-1-yl)-1,2,2-trimethyl-piperazine and the salts thereof in the treatment of schizophrenia |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK55192D0 (da) | 1992-04-28 | 1992-04-28 | Lundbeck & Co As H | 1-piperazino-1,2-dihydroindenderivater |
| PL1658277T3 (pl) | 2003-08-18 | 2012-10-31 | H Lundbeck As | Sól bursztynianowa i malonianowa trans-4-((1R,3S)-6-chloro-3-fenyloindan-1-ylo)-1,2,2-tri-metylopiperazyny i zastosowanie jako lek |
| AU2006269927B2 (en) | 2004-01-12 | 2013-05-16 | The Trustees Of The University Of Pennsylvania | Drug-containing implants and methods of use thereof |
| AU2005235422B2 (en) | 2004-04-22 | 2011-08-11 | Boehringer Ingelheim International Gmbh | New pharmaceutical compositions for the treatment of sexual disorders II |
| CN102065861B (zh) * | 2008-05-07 | 2013-10-16 | H.隆德贝克有限公司 | 反式-4-((1r，3s)-6-氯-3-苯基茚满-1-基)-1，2，2-三甲基哌嗪用于改善认知的用途 |
| CN102170884A (zh) * | 2008-10-03 | 2011-08-31 | H.隆德贝克有限公司 | 口服制剂 |
| MX2012000061A (es) | 2009-06-24 | 2012-06-01 | Msd Oss Bv | Formulaciones inyectables que contienen asenapina, y metodo de tratamiento usando las mismas. |
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| JP6140151B2 (ja) | 2017-05-31 |
| RU2014101482A (ru) | 2015-07-27 |
| RS57944B1 (sr) | 2019-01-31 |
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| EP2720698A1 (en) | 2014-04-23 |
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| BR112013032178A2 (pt) | 2016-12-20 |
| EP2720698B1 (en) | 2018-10-03 |
| AU2012274150B2 (en) | 2016-10-06 |
| PL2720698T3 (pl) | 2019-01-31 |
| US9610287B2 (en) | 2017-04-04 |
| TWI552751B (zh) | 2016-10-11 |
| SI2720698T1 (sl) | 2018-12-31 |
| AU2012274150A1 (en) | 2014-01-09 |
| WO2012175531A1 (en) | 2012-12-27 |
| IL230060A (en) | 2017-10-31 |
| MX349754B (es) | 2017-08-11 |
| US20140194409A1 (en) | 2014-07-10 |
| CN103608015A (zh) | 2014-02-26 |
| RU2613177C2 (ru) | 2017-03-15 |
| ZA201309617B (en) | 2015-04-29 |
| ES2694298T3 (es) | 2018-12-19 |
| JP2014517050A (ja) | 2014-07-17 |
| CA2838055A1 (en) | 2012-12-27 |
| KR101900989B1 (ko) | 2018-09-20 |
| KR20140033419A (ko) | 2014-03-18 |
| DK2720698T3 (en) | 2018-11-26 |
| HRP20181684T1 (hr) | 2018-12-14 |
| MX2013014978A (es) | 2014-04-10 |
| JO3421B1 (ar) | 2019-10-20 |
| SMT201800567T1 (it) | 2018-11-09 |
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