CA2777071A1 - Substituted halophenoxybenzamide derivatives - Google Patents

Substituted halophenoxybenzamide derivatives Download PDF

Info

Publication number
CA2777071A1
CA2777071A1 CA2777071A CA2777071A CA2777071A1 CA 2777071 A1 CA2777071 A1 CA 2777071A1 CA 2777071 A CA2777071 A CA 2777071A CA 2777071 A CA2777071 A CA 2777071A CA 2777071 A1 CA2777071 A1 CA 2777071A1
Authority
CA
Canada
Prior art keywords
general formula
hydrogen atom
compound
compounds
atom
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA2777071A
Other languages
English (en)
French (fr)
Inventor
Marion Hitchcock
Ingo Hartung
Florian Puehler
Gerhard Siemeister
Roland Neuhaus
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer Intellectual Property GmbH
Original Assignee
Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of CA2777071A1 publication Critical patent/CA2777071A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C307/00Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C307/04Diamides of sulfuric acids
    • C07C307/06Diamides of sulfuric acids having nitrogen atoms of the sulfamide groups bound to acyclic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/095Sulfur, selenium, or tellurium compounds, e.g. thiols
    • A61K31/10Sulfides; Sulfoxides; Sulfones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/136Amines having aromatic rings, e.g. ketamine, nortriptyline having the amino group directly attached to the aromatic ring, e.g. benzeneamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/145Amines having sulfur, e.g. thiurams (>N—C(S)—S—C(S)—N< and >N—C(S)—S—S—C(S)—N<), Sulfinylamines (—N=SO), Sulfonylamines (—N=SO2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/18Sulfonamides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA2777071A 2009-10-21 2010-10-12 Substituted halophenoxybenzamide derivatives Abandoned CA2777071A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP09075470 2009-10-21
EP09075470.6 2009-10-21
PCT/EP2010/006235 WO2011047796A1 (en) 2009-10-21 2010-10-12 Substituted halophenoxybenzamide derivatives

Publications (1)

Publication Number Publication Date
CA2777071A1 true CA2777071A1 (en) 2011-04-28

Family

ID=43086963

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2777071A Abandoned CA2777071A1 (en) 2009-10-21 2010-10-12 Substituted halophenoxybenzamide derivatives

Country Status (6)

Country Link
US (1) US20120263714A1 (https=)
EP (1) EP2491014A1 (https=)
JP (1) JP2013508320A (https=)
CN (1) CN102574782B (https=)
CA (1) CA2777071A1 (https=)
WO (1) WO2011047796A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
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CN115803024B (zh) * 2020-07-22 2025-01-10 中外制药株式会社 包含芳基酰胺衍生物的组合物
CN116930478A (zh) * 2022-04-02 2023-10-24 迈克生物股份有限公司 一种甲状腺素荧光偶联物及其制备方法和应用
CN121511080A (zh) * 2023-07-06 2026-02-10 华健未来(成都)科技股份有限公司 一类芳香酰胺类衍生物及其用途
WO2025146040A1 (zh) * 2024-01-01 2025-07-10 华健未来(成都)科技股份有限公司 芳香酰肼类衍生物及其医药用途

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Also Published As

Publication number Publication date
EP2491014A1 (en) 2012-08-29
HK1173134A1 (en) 2013-05-10
CN102574782B (zh) 2014-10-08
JP2013508320A (ja) 2013-03-07
WO2011047796A1 (en) 2011-04-28
CN102574782A (zh) 2012-07-11
US20120263714A1 (en) 2012-10-18

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Legal Events

Date Code Title Description
EEER Examination request

Effective date: 20151009

FZDE Dead

Effective date: 20171012