CA2565101A1 - Novel use of peptide compounds for treating pain in trigeminal neuralgia - Google Patents
Novel use of peptide compounds for treating pain in trigeminal neuralgia Download PDFInfo
- Publication number
- CA2565101A1 CA2565101A1 CA002565101A CA2565101A CA2565101A1 CA 2565101 A1 CA2565101 A1 CA 2565101A1 CA 002565101 A CA002565101 A CA 002565101A CA 2565101 A CA2565101 A CA 2565101A CA 2565101 A1 CA2565101 A1 CA 2565101A1
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- Prior art keywords
- lower alkyl
- use according
- unsubstituted
- aryl
- heterocyclic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Neurology (AREA)
- Gastroenterology & Hepatology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biomedical Technology (AREA)
- Psychology (AREA)
- Rheumatology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US57806204P | 2004-06-09 | 2004-06-09 | |
| US60/578,062 | 2004-06-09 | ||
| EP04013635A EP1604655A1 (en) | 2004-06-09 | 2004-06-09 | Novel use of peptide compounds for treating pain in trigeminal neuralgia |
| EP04013635.0 | 2004-06-09 | ||
| PCT/EP2005/006202 WO2005120539A2 (en) | 2004-06-09 | 2005-06-09 | Novel use of peptide compounds for treating pain in trigeminal neuralgia |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2565101A1 true CA2565101A1 (en) | 2005-12-22 |
Family
ID=34925315
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002565101A Abandoned CA2565101A1 (en) | 2004-06-09 | 2005-06-09 | Novel use of peptide compounds for treating pain in trigeminal neuralgia |
Country Status (13)
| Country | Link |
|---|---|
| US (2) | US7820857B2 (https=) |
| EP (2) | EP1604655A1 (https=) |
| JP (1) | JP2008501760A (https=) |
| CN (1) | CN1964708A (https=) |
| AU (1) | AU2005251465B2 (https=) |
| BR (1) | BRPI0511995A (https=) |
| CA (1) | CA2565101A1 (https=) |
| EA (1) | EA200602221A1 (https=) |
| MX (1) | MXPA06014193A (https=) |
| TW (1) | TW200701982A (https=) |
| UA (1) | UA88169C2 (https=) |
| WO (1) | WO2005120539A2 (https=) |
| ZA (1) | ZA200608745B (https=) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK1243262T3 (da) * | 2001-03-20 | 2006-10-02 | Sanol Arznei Schwarz Gmbh | Hidtil ukendt anvendelse af en peptidklasse af forbindelser til behandling af ikke-neuropatiske, inflammatoriske smerter |
| ES2185606T3 (es) | 2001-03-21 | 2003-05-01 | Sanol Arznei Schwarz Gmbh | Nuevo uso de una clase de compuestos peptidicos para tratamiento de la alodinia u otros tipos diferentes de dolor cronico o fantasma. |
| JP4664924B2 (ja) | 2003-12-02 | 2011-04-06 | ウーツェーベー ファルマ ゲーエムベーハー | 中枢神経因性疼痛の治療のためのペプチド化合物の新規使用 |
| US20070042969A1 (en) * | 2004-03-26 | 2007-02-22 | Srz Properties, Inc. | Combination therapy for pain in painful diabetic neuropathy |
| US20100256179A1 (en) * | 2004-03-26 | 2010-10-07 | Ucb Pharma Gmbh | Combination therapy for pain in painful diabetic neuropathy |
| KR20070007931A (ko) | 2004-04-16 | 2007-01-16 | 쉬바르츠파르마에이지 | 만성 두통의 예방 및 치료를 위한 펩티드 화합물의 용도 |
| EP1604655A1 (en) | 2004-06-09 | 2005-12-14 | Schwarz Pharma Ag | Novel use of peptide compounds for treating pain in trigeminal neuralgia |
| PL1781276T3 (pl) * | 2004-08-27 | 2010-11-30 | Ucb Pharma Gmbh | Zastosowanie związków peptydowych do leczenia bólu związanego z rakiem kości, bólu indukowanego przez chemioterapię oraz nukleozydy |
| EP1642889A1 (en) * | 2004-10-02 | 2006-04-05 | Schwarz Pharma Ag | Improved synthesis scheme for lacosamide |
| US20060252749A1 (en) * | 2005-01-28 | 2006-11-09 | Srz Properties, Inc. | Lacosamide for add-on therapy of psychosis |
| US20070043120A1 (en) * | 2005-08-18 | 2007-02-22 | Bettina Beyreuther | Therapeutic combination for painful medical conditions |
| US20070048372A1 (en) * | 2005-08-18 | 2007-03-01 | Srz Properties, Inc. | Method for treating non-inflammatory osteoarthritic pain |
| EP1754476A1 (en) * | 2005-08-18 | 2007-02-21 | Schwarz Pharma Ag | Lacosamide (SPM 927) for treating myalgia, e.g. fibromyalgia |
| JP5276982B2 (ja) * | 2005-08-26 | 2013-08-28 | ボード オブ トラスティーズ オブ ザ レランド スタンフォード ジュニア ユニバーシティ | オキシトシンの投与による頭痛の処置のための方法 |
| WO2007144195A2 (en) | 2006-06-15 | 2007-12-21 | Schwarz Pharma Ag | Pharmaceutical composition with synergistic anticonvulsant effect |
| EP1873527A1 (en) * | 2006-06-30 | 2008-01-02 | Schwarz Pharma Ag | Method for identifying CRMP modulators |
| CN101466390B (zh) | 2006-06-15 | 2014-03-12 | 优时比制药有限公司 | 用于治疗难治性癫痫持续状态的肽类化合物 |
| EP1920780A1 (en) * | 2006-10-12 | 2008-05-14 | Schwarz Pharma Ag | Peptide compounds for the treatment of hyperexcitability disorders |
| CA2774569A1 (en) * | 2009-09-23 | 2011-03-31 | The University Of North Carolina At Chapel Hill | Novel n-benzylamide substituted derivatives of 2-(acylamido)acetic acid and 2-(acylamido)propionic acids: potent neurological agents |
| MX350056B (es) | 2009-11-03 | 2017-08-25 | Lupin Ltd | Formulacion de liberacion modificada de lacosamida. |
| MX2013005974A (es) | 2010-12-02 | 2013-07-29 | Ucb Pharma Gmbh | Formulacion de lacosamida de administracion una vez al dia. |
| EP2468261A1 (en) | 2010-12-02 | 2012-06-27 | UCB Pharma GmbH | Formulation of lacosamide |
| SG11201705591PA (en) | 2015-01-07 | 2017-08-30 | Trigemina Inc | Magnesium-containing oxytocin formulations and methods of use |
| CN109069480A (zh) | 2015-12-30 | 2018-12-21 | 阿达玛斯医药公司 | 用于治疗与癫痫相关的病症的方法和组合物 |
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-
2004
- 2004-06-09 EP EP04013635A patent/EP1604655A1/en not_active Withdrawn
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2005
- 2005-06-09 UA UAA200700160A patent/UA88169C2/ru unknown
- 2005-06-09 CA CA002565101A patent/CA2565101A1/en not_active Abandoned
- 2005-06-09 WO PCT/EP2005/006202 patent/WO2005120539A2/en not_active Ceased
- 2005-06-09 EP EP05754667.3A patent/EP1753415B1/en not_active Expired - Lifetime
- 2005-06-09 MX MXPA06014193A patent/MXPA06014193A/es not_active Application Discontinuation
- 2005-06-09 CN CNA2005800185740A patent/CN1964708A/zh active Pending
- 2005-06-09 JP JP2007526303A patent/JP2008501760A/ja not_active Withdrawn
- 2005-06-09 AU AU2005251465A patent/AU2005251465B2/en not_active Ceased
- 2005-06-09 BR BRPI0511995-2A patent/BRPI0511995A/pt not_active IP Right Cessation
- 2005-06-09 US US11/148,429 patent/US7820857B2/en not_active Expired - Fee Related
- 2005-06-09 EA EA200602221A patent/EA200602221A1/ru unknown
- 2005-07-11 TW TW094123448A patent/TW200701982A/zh unknown
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2006
- 2006-10-19 ZA ZA200608745A patent/ZA200608745B/en unknown
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2010
- 2010-06-16 US US12/816,753 patent/US8338641B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| UA88169C2 (ru) | 2009-09-25 |
| ZA200608745B (en) | 2008-04-30 |
| JP2008501760A (ja) | 2008-01-24 |
| AU2005251465B2 (en) | 2009-07-09 |
| EA200602221A1 (ru) | 2007-04-27 |
| EP1753415A2 (en) | 2007-02-21 |
| WO2005120539A2 (en) | 2005-12-22 |
| US20100256241A1 (en) | 2010-10-07 |
| TW200701982A (en) | 2007-01-16 |
| MXPA06014193A (es) | 2007-03-12 |
| US8338641B2 (en) | 2012-12-25 |
| CN1964708A (zh) | 2007-05-16 |
| EP1604655A1 (en) | 2005-12-14 |
| WO2005120539A3 (en) | 2006-01-26 |
| BRPI0511995A (pt) | 2008-01-22 |
| EP1753415B1 (en) | 2013-04-17 |
| US20060135437A1 (en) | 2006-06-22 |
| US7820857B2 (en) | 2010-10-26 |
| AU2005251465A1 (en) | 2005-12-22 |
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