CA2478918A1 - Angiogenesis inhibitors - Google Patents
Angiogenesis inhibitors Download PDFInfo
- Publication number
- CA2478918A1 CA2478918A1 CA002478918A CA2478918A CA2478918A1 CA 2478918 A1 CA2478918 A1 CA 2478918A1 CA 002478918 A CA002478918 A CA 002478918A CA 2478918 A CA2478918 A CA 2478918A CA 2478918 A1 CA2478918 A1 CA 2478918A1
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- CA
- Canada
- Prior art keywords
- furyl
- phenyl
- compound
- cancer
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Landscapes
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Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
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| US36889202P | 2002-03-29 | 2002-03-29 | |
| US60/368,892 | 2002-03-29 | ||
| US10/147,445 | 2002-05-16 | ||
| US10/147,445 US7166293B2 (en) | 2002-03-29 | 2002-05-16 | Angiogenesis inhibitors |
| PCT/US2003/009968 WO2003082274A1 (en) | 2002-03-29 | 2003-03-31 | Angiogenesis inhibitors |
Publications (1)
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| CA2478918A1 true CA2478918A1 (en) | 2003-10-09 |
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| TW (1) | TWI296524B (enExample) |
| WO (1) | WO2003082274A1 (enExample) |
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| US7166293B2 (en) * | 2002-03-29 | 2007-01-23 | Carlsbad Technology, Inc. | Angiogenesis inhibitors |
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| US20050096370A1 (en) * | 2003-04-07 | 2005-05-05 | Bizbiotech Co., Ltd. | Method for inhibiting tumor angiogenesis and tumor growth |
| US20040198798A1 (en) * | 2003-04-07 | 2004-10-07 | Park Jong-Wan | Method for inhibiting tumor angiogenesis and tumor growth |
| US7429596B2 (en) * | 2003-06-20 | 2008-09-30 | The Regents Of The University Of California | 1H-pyrrolo [2,3-D] pyrimidine derivatives and methods of use thereof |
| EP1646382A4 (en) * | 2003-06-30 | 2010-07-21 | Hif Bio Inc | COMPOUNDS, COMPOSITIONS AND METHODS |
| CN100516049C (zh) | 2004-11-16 | 2009-07-22 | 永信药品工业股份有限公司 | 抗血管生成药n2-(取代的芳基甲基)-3-(取代的苯基)吲唑的合成 |
| EP1831225A2 (en) * | 2004-11-19 | 2007-09-12 | The Regents of the University of California | Anti-inflammatory pyrazolopyrimidines |
| TW200732305A (en) * | 2005-12-23 | 2007-09-01 | Yung Shin Pharmaceutical Ind | Cancer chemotherapy |
| KR20150038395A (ko) * | 2006-04-04 | 2015-04-08 | 더 리젠트스 오브 더 유니이버시티 오브 캘리포니아 | 키나제 길항물질 |
| US20080252028A1 (en) * | 2007-04-16 | 2008-10-16 | Ming-Tai Huang | Shock absorbing device for toy stroller |
| WO2009046448A1 (en) | 2007-10-04 | 2009-04-09 | Intellikine, Inc. | Chemical entities and therapeutic uses thereof |
| US8193182B2 (en) | 2008-01-04 | 2012-06-05 | Intellikine, Inc. | Substituted isoquinolin-1(2H)-ones, and methods of use thereof |
| KR101653842B1 (ko) | 2008-01-04 | 2016-09-02 | 인텔리카인, 엘엘씨 | 특정 화학 물질, 조성물 및 방법 |
| WO2009114874A2 (en) * | 2008-03-14 | 2009-09-17 | Intellikine, Inc. | Benzothiazole kinase inhibitors and methods of use |
| WO2009114870A2 (en) * | 2008-03-14 | 2009-09-17 | Intellikine, Inc. | Kinase inhibitors and methods of use |
| US20110224223A1 (en) * | 2008-07-08 | 2011-09-15 | The Regents Of The University Of California, A California Corporation | MTOR Modulators and Uses Thereof |
| JP5788316B2 (ja) * | 2008-07-08 | 2015-09-30 | インテリカイン， エルエルシー | キナーゼインヒビターおよび使用方法 |
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| WO2010045542A2 (en) | 2008-10-16 | 2010-04-22 | The Regents Of The University Of California | Fused ring heteroaryl kinase inhibitors |
| US8476282B2 (en) * | 2008-11-03 | 2013-07-02 | Intellikine Llc | Benzoxazole kinase inhibitors and methods of use |
| CA2760791C (en) | 2009-05-07 | 2017-06-20 | Intellikine, Inc. | Heterocyclic compounds and uses thereof |
| US8980899B2 (en) | 2009-10-16 | 2015-03-17 | The Regents Of The University Of California | Methods of inhibiting Ire1 |
| JP5951600B2 (ja) | 2010-05-21 | 2016-07-13 | インフィニティー ファーマシューティカルズ， インコーポレイテッド | キナーゼ調節のための、化合物、組成物および方法 |
| CN103298474B (zh) | 2010-11-10 | 2016-06-29 | 无限药品股份有限公司 | 杂环化合物及其用途 |
| CN102485724B (zh) * | 2010-12-06 | 2015-08-12 | 中国人民解放军军事医学科学院毒物药物研究所 | 取代噻吩基吡唑并吡啶类化合物及其医药用途 |
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| UA111754C2 (uk) | 2011-10-06 | 2016-06-10 | Байєр Фарма Акцієнгезелльшафт | Заміщені бензиліндазоли для застосування як інгібіторів bub1-кінази для лікування гіперпроліферативних захворювань |
| WO2013092512A1 (en) | 2011-12-21 | 2013-06-27 | Bayer Intellectual Property Gmbh | Substituted benzylpyrazoles |
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| US20050119278A1 (en) * | 2002-05-16 | 2005-06-02 | Che-Ming Teng | Anti-angiogenesis methods |
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| AU2003222148B2 (en) | 2008-10-09 |
| JP2005521713A (ja) | 2005-07-21 |
| KR20100102746A (ko) | 2010-09-24 |
| AU2003222148A1 (en) | 2003-10-13 |
| TWI296524B (en) | 2008-05-11 |
| EP1496894A4 (en) | 2007-06-06 |
| US7166293B2 (en) | 2007-01-23 |
| WO2003082274A1 (en) | 2003-10-09 |
| US20030186996A1 (en) | 2003-10-02 |
| CN1642542A (zh) | 2005-07-20 |
| AU2003222148C1 (en) | 2009-05-21 |
| KR20040095342A (ko) | 2004-11-12 |
| US20050107406A1 (en) | 2005-05-19 |
| NZ535990A (en) | 2006-10-27 |
| CN1642542B (zh) | 2012-01-11 |
| HK1080745A1 (zh) | 2006-05-04 |
| KR100997174B1 (ko) | 2010-11-29 |
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